作者
MO Chekanov, AR Synyugin, SS Lukashov, SM Yarmoluk
发表日期
2009/12/1
期刊
Ukrainica Bioorganica Acta
卷号
7
期号
1
简介
Abstract Several 2-phenylisothiazolidine-3-one dioxide derivatives were synthesized and their in vitro activity against protein kinase CK2 was measured. The most active compound N-(3-acetylphenyl)-2-chloro-4-(4-methyl-1, 1-dioxido-3-phenylisothiazolidin-2-yl) benzamide showed IC50 value 20 μM.
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