关注
Samer Haidar
Samer Haidar
Professor of Pharmaceutical and Medicinal chemistry Damascus University, Syria
在 damascusuniversity.edu.sy 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Effects of novel 17α-hydroxylase/C17, 20-lyase (P450 17, CYP 17) inhibitors on androgen biosynthesis in vitro and in vivo
S Haidar, PB Ehmer, S Barassin, C Batzl-Hartmann, RW Hartmann
The Journal of steroid biochemistry and molecular biology 84 (5), 555-562, 2003
1322003
Synthesis and evaluation of novel steroidal oxime inhibitors of P450 17 (17α-hydroxylase/C17− 20-lyase) and 5α-reductase types 1 and 2
RW Hartmann, M Hector, S Haidar, PB Ehmer, W Reichert, J Jose
Journal of medicinal chemistry 43 (22), 4266-4277, 2000
1202000
Preclinical Efficacy of the MDM2 Inhibitor RG7112 in MDM2-Amplified and TP53 Wild-type Glioblastomas
M Verreault, C Schmitt, L Goldwirt, K Pelton, S Haidar, C Levasseur, ...
Clinical Cancer Research 22 (5), 1185-1196, 2016
1062016
Inhibition of CYP 17, a new strategy for the treatment of prostate cancer
RW Hartmann, PB Ehmer, S Haidar, M Hector, J Jose, CDP Klein, ...
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2002
882002
Novel steroidal pyrimidyl inhibitors of P 450 17(17 α-hydroxylase/C 17-20-lyase)
S Haidar, PB Ehmer, RW Hartmann
Archiv der Pharmazie 334 (12), 373-374, 2001
412001
Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining
S Haidar, Z Bouaziz, C Marminon, T Laitinen, A Poso, M Le Borgne, ...
Pharmaceuticals 10 (1), 8, 2017
342017
Determination of levocetirizine configurational stability in tablets using chiral HPLC method
R Hommoss, H Elzein, S Haidar
International Journal of Pharmacy and Pharmaceutical Sciences 3 (2), 103-107, 2011
232011
In vitro and in silico evaluation of bikaverin as a potent inhibitor of human protein kinase CK2
S Haidar, D Aichele, R Birus, J Hielscher, T Laitinen, A Poso, J Jose
Molecules 24 (7), 1380, 2019
212019
C16 and C17 Substituted Derivatives of Pregnenolone and Progesterone as Inhibitors of 17α‐Hydroxylase‐C17, 20‐lyase: Synthesis and Biological Evaluation
S Haidar, RW Hartmann
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2002
192002
Synthesis and Evaluation of Steroidal Hydroxamic Acids as Inhibitors of P450 17 (17α‐Hydroxylase/C17‐20‐Lyase)
S Haidar, CDP Klein, RW Hartmann
Archiv der Pharmazie 334 (4), 138-140, 2001
182001
Separation and assay of antiprotozoal imidazole derivatives (metronidazole, tinidazole and secnidazole) by RPHPLC
Z Alhalabi, MA Al-Khayat, S Haidar
International Journal of Pharmaceutical Sciences Review and Research 13 (1 …, 2012
172012
Design, synthesis and biological evaluation of new embelin derivatives as CK2 inhibitors
S Oramas-Royo, S Haidar, A Amesty, P Martin-Acosta, G Feresin, A Tapia, ...
Bioorganic Chemistry 95, 103520, 2020
142020
Human αS1-casein induces IL-8 secretion by binding to the ecto-domain of the TLR4/MD2 receptor complex
T Saenger, S Vordenbäumen, S Genich, S Haidar, M Schulte, C Nienberg, ...
Biochimica et Biophysica Acta (BBA)-General Subjects 1863 (3), 632-643, 2019
122019
Development and validation of RP-HPLC method for determination of clopidogrel in tablets
MA Al-Khayat, S Haidar, H Mando
Int. J. Pharm. Sci. Rev. Res 14, 1-5, 2012
122012
QSAR Model of Indeno[1,2-b]indole Derivatives and Identification of N-isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3-b]furan-3-carboxamide as a Potent …
S Haidar, C Marminon, D Aichele, A Nacereddine, W Zeinyeh, A Bouzina, ...
Molecules 25 (1), 97, 2019
102019
Development and validation of RP-HPLC method for analysis of four UV filters in sunscreen products
N Yousef Agha, S Haidar, MA Al-Khayat
Int. J. Pharm. Sci. Rev. Res 23 (2), 254-258, 2013
92013
Autodisplay of human PIP5K1α lipid kinase on Escherichia coli and inhibitor testing
K Strätker, S Haidar, M Dubiel, A Estévez-Braun, J Jose
Enzyme and Microbial Technology 143, 109717, 2021
72021
Synthesis and biological evaluation of 2, 6-di (furan-3-yl) anthracene-9, 10-dione as an inhibitor of human protein kinase CK2
S Haidar, A Meyers, A Bollacke, J Jose
Die Pharmazie-An International Journal of Pharmaceutical Sciences 70 (12 …, 2015
72015
Development of an in vitro screening assay for PIP5K1α lipid kinase and identification of potent inhibitors
K Strätker, S Haidar, Á Amesty, E El‐Awaad, C Götz, A Estévez‐Braun, ...
The FEBS Journal 287 (14), 3042-3064, 2020
62020
Computational prediction of new CYP17 inhibitors based on pharmacophore modeling, virtual screening and docking approach
S Haidar, RW Hartmann
Die Pharmazie-An International Journal of Pharmaceutical Sciences 72 (9 …, 2017
32017
系统目前无法执行此操作,请稍后再试。
文章 1–20