| Evaluation of 3-Carboxy-4(1H)-quinolones as Inhibitors of Human Protein Kinase CK2 AG Golub, OY Yakovenko, VG Bdzhola, VM Sapelkin, P Zien, ... Journal of medicinal chemistry 49 (22), 6443-6450, 2006 | 87 | 2006 |
| Synthesis and biological evaluation of substituted (thieno [2, 3-d] pyrimidin-4-ylthio) carboxylic acids as inhibitors of human protein kinase CK2 AG Golub, VG Bdzhola, NV Briukhovetska, AO Balanda, OP Kukharenko, ... European journal of medicinal chemistry 46 (3), 870-876, 2011 | 79 | 2011 |
| Identification of 3H-Naphtho[1,2,3-de]quinoline-2,7-diones as Inhibitors of Apoptosis Signal-Regulating Kinase 1 (ASK1) GP Volynets, MO Chekanov, AR Synyugin, AG Golub, OP Kukharenko, ... Journal of medicinal chemistry 54 (8), 2680-2686, 2011 | 67 | 2011 |
| Evaluation of 4, 5, 6, 7-tetrahalogeno-1H-isoindole-1, 3 (2H)-diones as inhibitors of human protein kinase CK2 AG Golub, OY Yakovenko, AO Prykhod'Ko, SS Lukashov, VG Bdzhola, ... Biochimica et Biophysica Acta (BBA)-Proteins and Proteomics 1784 (1), 143-149, 2008 | 61 | 2008 |
| Discovery of potent anti-tuberculosis agents targeting leucyl-tRNA synthetase OI Gudzera, AG Golub, VG Bdzhola, GP Volynets, SS Lukashov, ... Bioorganic & Medicinal Chemistry 24 (5), 1023-1031, 2016 | 42 | 2016 |
| Design, synthesis and biological evaluation of N-phenylthieno [2, 3-d] pyrimidin-4-amines as inhibitors of FGFR1 AA Gryshchenko, VG Bdzhola, AO Balanda, NV Briukhovetska, IM Kotey, ... Bioorganic & Medicinal Chemistry 23 (9), 2287-2293, 2015 | 38 | 2015 |
| Discovery and characterization of synthetic 4′-hydroxyflavones—New CK2 inhibitors from flavone family AG Golub, VG Bdzhola, OV Ostrynska, IV Kyshenia, VM Sapelkin, ... Bioorganic & medicinal chemistry 21 (21), 6681-6689, 2013 | 37 | 2013 |
| Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1, 5-dihydro-pyrrol-2-one SA Starosyla, GP Volynets, SS Lukashov, OB Gorbatiuk, AG Golub, ... Bioorganic & Medicinal Chemistry 23 (10), 2489-2497, 2015 | 35 | 2015 |
| Kirchhoff atomic charges fitted to multipole moments: implementation for a virtual screening system O Yakovenko, AA Oliferenko, VG Bdzhola, VA Palyulin, NS Zefirov Journal of computational chemistry 29 (8), 1332-1343, 2008 | 35 | 2008 |
| Structure-based discovery of novel flavonol inhibitors of human protein kinase CK2 AG Golub, VG Bdzhola, YV Kyshenia, VM Sapelkin, AO Prykhod’ko, ... Molecular and cellular biochemistry 356, 107-115, 2011 | 34 | 2011 |
| Design, synthesis and evaluation of 3-quinoline carboxylic acids as new inhibitors of protein kinase CK2 AR Syniugin, OV Ostrynska, MO Chekanov, GP Volynets, SA Starosyla, ... Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup4), 160-169, 2016 | 29 | 2016 |
| Treatment of cultured human astrocytes and vascular endothelial cells with protein kinase CK2 inhibitors induces early changes in cell shape and cytoskeleton AA Kramerov, AG Golub, VG Bdzhola, SM Yarmoluk, K Ahmed, M Bretner, ... Molecular and cellular biochemistry 349, 125-137, 2011 | 29 | 2011 |
| Identification of novel PARP-1 inhibitors by structure-based virtual screening K Hannigan, SS Kulkarni, VG Bdzhola, AG Golub, SM Yarmoluk, ... Bioorganic & medicinal chemistry letters 23 (21), 5790-5794, 2013 | 28 | 2013 |
| A note of caution on the role of halogen bonds for protein kinase/inhibitor recognition suggested by high-and low-salt CK2α complex structures B Guerra, N Bischoff, VG Bdzhola, SM Yarmoluk, OG Issinger, AG Golub, ... ACS Chemical Biology 10 (7), 1654-1660, 2015 | 26 | 2015 |
| Rational design of apoptosis signal-regulating kinase 1 inhibitors: discovering novel structural scaffold GP Volynets, VG Bdzhola, AG Golub, AR Synyugin, MA Chekanov, ... European Journal of Medicinal Chemistry 61, 104-115, 2013 | 26 | 2013 |
| Identification of Mycobacterium tuberculosis leucyl-tRNA synthetase (LeuRS) inhibitors among the derivatives of 5-phenylamino-2H-[1,2,4]triazin-3-one OI Gudzera, AG Golub, VG Bdzhola, GP Volynets, OP Kovalenko, ... Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup2), 201-207, 2016 | 25 | 2016 |
| Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno [2, 3-d] pyrimidines OV Ostrynska, AO Balanda, VG Bdzhola, AG Golub, IM Kotey, ... European Journal of Medicinal Chemistry 115, 148-160, 2016 | 25 | 2016 |
| Dual-target inhibitors of mycobacterial aminoacyl-tRNA synthetases among N-benzylidene-N′-thiazol-2-yl-hydrazines OP Kovalenko, GP Volynets, MY Rybak, SA Starosyla, OI Gudzera, ... Medchemcomm 10 (12), 2161-2169, 2019 | 20 | 2019 |
| Design, synthesis and biological evaluation of 5-amino-4-(1H-benzoimidazol-2-yl)-phenyl-1, 2-dihydro-pyrrol-3-ones as inhibitors of protein kinase FGFR1 AA Gryshchenko, SS Tarnavskiy, KV Levchenko, VG Bdzhola, ... Bioorganic & Medicinal Chemistry 24 (9), 2053-2059, 2016 | 19 | 2016 |
| The new method of distribution integrals evaluations for high throughput virtual screening OY Yakovenko, AA Oliferenko, AG Golub, VG Bdzhola, SM Yarmoluk Ukr. Bioorg. Acta 1, 52-62, 2007 | 19 | 2007 |
