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Vladlen Klochkov
Vladlen Klochkov
ассистент, кафедра фармакологии, ВолгГМУ
在 volgmed.ru 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Synthesis, in vitro and in vivo evaluation of 2-aryl-4H-chromene and 3-aryl-1H-benzo [f] chromene derivatives as novel α-glucosidase inhibitors
AA Spasov, DA Babkov, DV Osipov, VG Klochkov, DR Prilepskaya, ...
Bioorganic & medicinal chemistry letters 29 (1), 119-123, 2019
472019
Neural network modeling of the multitarget rage inhibitory activity
PM Vassiliev, AA Spasov, LR Yanaliyeva, AN Kochetkov, ...
Biochemistry (Moscow), Supplement Series B: Biomedical Chemistry 13, 256-263, 2019
212019
Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3, 5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors
VG Klochkov, EN Bezsonova, M Dubar, DD Melekhina, VV Temnov, ...
Bioorganic & Medicinal Chemistry Letters 55, 128449, 2022
122022
Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors
A Spasov, A Ozerov, P Vassiliev, V Kosolapov, N Gurova, ...
Scientific reports 11 (1), 24380, 2021
112021
Discovery of nitro-azolo [1, 5-a] pyrimidines with anti-inflammatory and protective activity against LPS-induced acute lung injury
A Spasov, V Kosolapov, D Babkov, V Klochkov, E Sokolova, ...
Pharmaceuticals 15 (5), 537, 2022
52022
3-Arylidene-2-oxindoles as potent NRH: quinone oxidoreductase 2 inhibitors
NA Lozinskaya, EN Bezsonova, M Dubar, DD Melekhina, DR Bazanov, ...
Molecules 28 (3), 1174, 2023
42023
ИНГИБИТОРЫ РЕЦЕПТОРОВ КОНЕЧНЫХ ПРОДУКТОВ ГЛИКИРОВАНИЯ
КВГ Васильев П.М., Яналиева Л.Р., Спасов А.А., Кочетков А.Н., Ворфоломеева В.В.
RU Patent RU 2,019,620,160, 2019
42019
База данных 3D-моделей релевантных белков-мишеней сигнального пути RAGE-NF-kB
ПМ Васильев, ЛР Яналиева, АН Кочетков, ВВ Ворфоломеева, ...
Вестник Волгоградского государственного медицинского университета, 133-138, 2018
42018
Нейросетевое моделирование мультитаргетной RAGE-ингибирующей активности
ПМ Васильев, АА Спасов, ЛР Яналиева, АН Кочетков, ...
Биомедицинская химия 65 (2), 91-98, 2019
32019
Amino derivatives of diaryl pyrimidines and azolopyrimidines as protective agents against LPS-induced acute lung injury
A Spasov, I Ovchinnikova, O Fedorova, Y Titova, D Babkov, V Kosolapov, ...
Molecules 28 (2), 741, 2023
22023
Design, Synthesis and Pharmacological Evaluation of Novel C2,C3-Quinoxaline Derivatives as Promising Anxiolytic Agents
DV Maltsev, MO Skripka, AA Spasov, PM Vassiliev, MA Perfiliev, ...
International Journal of Molecular Sciences 23 (22), 14401, 2022
22022
Guanidine Derivatives of Quinazoline-2,4(1H,3H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents
A Spasov, A Ozerov, V Kosolapov, N Gurova, A Kucheryavenko, ...
Life 12 (10), 1647, 2022
22022
DATABASE OF 3D MODELS OF RELEVANT PROTEIN-TARGETS OF THE RAGE-NF-KB SIGNSLING PATHWAY
PM Vassiliev, LR Ianalieva, AN Kochetkov, VV Vorfolomeeva, ...
Journal of Volgograd State Medical University 15 (3), 133-138, 2018
22018
Литолиз конкрементов мочевыделительной системы животных органическими соединениями с выраженной комплексообразующей способностью
АК Брель, СВ Лисина, ВГ Клочков
22014
СПОСОБ ЛЕЧЕНИЯ САХАРНОГО ДИАБЕТА
НА Лозинская, ЕВ Зарянова, ДА Бабков, ВГ Клочков, АА Спасов, ...
12020
БИОМИШЕНИ СИГНАЛЬНЫХ ПУТЕЙ RAGE–NF-KB
АН Кочетков, ЛР Яналиева, ПМ Васильев, ВГ Клочков
XXV Российский национальный конгресс" Человек и лекарство", 73-73, 2018
12018
NLRX1 Inhibits LPS-Induced Microglial Death via Inducing p62-Dependent HO-1 Expression, Inhibiting MLKL and Activating PARP-1
YL Huang, DY Huang, V Klochkov, CM Chan, YS Chen, WW Lin
Antioxidants 13 (4), 481, 2024
2024
3-Arylidene-2-oxindoles as GSK3β inhibitors and anti-thrombotic agents
D Babkov, E Bezsonova, V Sirotenko, E Othman, V Klochkov, S Sosonyuk, ...
Bioorganic & Medicinal Chemistry Letters 87, 129283, 2023
2023
3-ARILIDENE-2-OXYNDOLE DERIVATIVES AS MELATONIN ANALOGUES WITH ANTIOXIDANT AND INTRAOCULAR PRESSURE LOWERING PROPERTIES
AA Spasov, LV Naumenko, DS Yakovlev, AS Taran, EV Sokolova, ...
Journal of Volgograd State Medical University 19 (4), 94-103, 2022
2022
PROCEEDING OF INTERNATIONAL CONFERENCE ON POST-COVID HEALTHCARE, MEDICAL RESEARCH AND EDUCATION 2022 (pS1-S102) & PROCEEDING OF 35TH ANNUAL SCIENTIFIC MEETING OF THE MALAYSIAN …
NAA Nasir
Journal of Clinical and Health Sciences 7 (2 (S)), 1-199, 2022
2022
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