5-HT2C receptor structures reveal the structural basis of GPCR polypharmacology Y Peng, JD McCorvy, K Harpsøe, K Lansu, S Yuan, P Popov, L Qu, M Pu, ... Cell 172 (4), 719-730. e14, 2018 | 234 | 2018 |
The importance of the excitatory amino acid transporter 3 (EAAT3) WE Bjørn-Yoshimoto, SM Underhill Neurochemistry international 98, 4-18, 2016 | 94 | 2016 |
Excitatory amino acid transporters: recent insights into molecular mechanisms, novel modes of modulation and new therapeutic possibilities AA Jensen, C Fahlke, WE Bjørn-Yoshimoto, L Bunch Current opinion in pharmacology 20, 116-123, 2015 | 94 | 2015 |
Postendocytic sorting of constitutively internalized dopamine transporter in cell lines and dopaminergic neurons J Eriksen, WE Bjørn-Yoshimoto, TN Jørgensen, AH Newman, U Gether Journal of Biological Chemistry 285 (35), 27289-27301, 2010 | 77 | 2010 |
Improving heterologous production of phenylpropanoids in Saccharomyces cerevisiae by tackling an unwanted side reaction of Tsc13, an endogenous double … BJ Lehka, M Eichenberger, WE Bjørn-Yoshimoto, KG Vanegas, N Buijs, ... FEMS Yeast Research 17 (1), fox004, 2017 | 58 | 2017 |
Curses or cures: A review of the numerous benefits versus the biosecurity concerns of conotoxin research WE Bjørn-Yoshimoto, IBL Ramiro, M Yandell, JM McIntosh, BM Olivera, ... Biomedicines 8 (8), 235, 2020 | 29 | 2020 |
Somatostatin venom analogs evolved by fish-hunting cone snails: From prey capture behavior to identifying drug leads IBL Ramiro, WE Bjørn-Yoshimoto, JS Imperial, J Gajewiak, PF Salcedo, ... Science Advances 8 (12), eabk1410, 2022 | 22 | 2022 |
Identification of a new class of selective excitatory amino acid transporter subtype 1 (EAAT1) inhibitors followed by a structure–activity relationship study SW Hansen, MN Erichsen, B Fu, WE Bjørn-Yoshimoto, B Abrahamsen, ... Journal of Medicinal Chemistry 59 (19), 8757-8770, 2016 | 18 | 2016 |
New 4-functionalized glutamate analogues are selective agonists at metabotropic glutamate receptor subtype 2 or selective agonists at metabotropic glutamate receptor group III THV Huynh, MN Erichsen, AS Tora, C Goudet, E Sagot, Z Assaf, ... Journal of Medicinal Chemistry 59 (3), 914-924, 2016 | 15 | 2016 |
Identification and Structure–Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype … P Wu, WE Bjørn-Yoshimoto, M Staudt, AA Jensen, L Bunch ACS Chemical Neuroscience 10 (10), 4414-4429, 2019 | 13 | 2019 |
Reconstructing the origins of the somatostatin and allatostatin-C signaling systems using the accelerated evolution of biodiverse cone snail toxins TL Koch, IBL Ramiro, P Flórez Salcedo, E Engholm, KJ Jensen, K Chase, ... Molecular Biology and Evolution 39 (4), msac075, 2022 | 12 | 2022 |
β-Sulfonamido functionalized aspartate analogues as excitatory amino acid transporter inhibitors: distinct subtype selectivity profiles arising from subtle structural differences JC Hansen, WE Bjørn-Yoshimoto, N Bisballe, B Nielsen, AA Jensen, ... Journal of Medicinal Chemistry 59 (19), 8771-8786, 2016 | 12 | 2016 |
Biosynthesis of phenylpropanoids and phenylpropanoid derivatives M Naesby, ES VECILLA, M Eichenberger, BJ Lehka, WE Bjørn-yoshimoto, ... US Patent 10,760,062, 2020 | 11 | 2020 |
Bioavailability Studies and in vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH‐102 I Haym, THV Huynh, SW Hansen, MHF Pedersen, JA Ruiz, MN Erichsen, ... ChemMedChem 11 (4), 403-419, 2016 | 10 | 2016 |
Ligand selectivity hotspots in serotonin GPCRs IA Simon, WE Bjørn-Yoshimoto, K Harpsøe, S Iliadis, B Svensson, ... Trends in Pharmacological Sciences, 2023 | 7 | 2023 |
New Insight into the Structure–Activity Relationships of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors UCPH‐101 and UCPH‐102 SW Hansen, MN Erichsen, THV Huynh, JA Ruiz, I Haym, ... ChemMedChem 11 (4), 382-402, 2016 | 6 | 2016 |
Design and Synthesis of 2,3-trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters CBM Poulie, A Alcaide, M Krell-Jørgensen, Y Larsen, E Astier, ... ACS chemical neuroscience 10 (6), 2989-3007, 2019 | 4 | 2019 |
(S)-2-Mercaptohistidine: A First Selective Orthosteric GluK3 Antagonist CBM Poulie, Y Larsen, C Leteneur, G Barthet, WE Bjørn-Yoshimoto, ... ACS Chemical Neuroscience 13 (10), 1580-1587, 2022 | 2 | 2022 |
Reconstructing the Origins of a Neuropeptide Signaling System Using the Accelerated Evolution of Biodiverse Cone Snail Venoms TL Koch, IBL Ramiro, P Flórez-Salcedo, E Engholm, KJ Jensen, K Chase, ... bioRxiv, 2021.11. 05.463867, 2021 | | 2021 |
Molecular determinants in two loops of the glutamate transporter 1 involved in transporter reorganization: MTU07-03 W Bjørn-Yoshimoto, L Bunch, A Jensen Journal of Neurochemistry 134, 154-155, 2015 | | 2015 |