Recent updates of fluoroquinolones as antibacterial agents HAA Ezelarab, SH Abbas, HA Hassan, GEDA Abuo‐Rahma Archiv der Pharmazie 351 (9), 1800141, 2018 | 170 | 2018 |
Design and synthesis of novel quinoline/chalcone/1, 2, 4-triazole hybrids as potent antiproliferative agent targeting EGFR and BRAFV600E kinases AM Mohassab, HA Hassan, D Abdelhamid, AM Gouda, BGM Youssif, ... Bioorganic chemistry 106, 104510, 2021 | 71 | 2021 |
New quinoline/chalcone hybrids as anti-cancer agents: Design, synthesis, and evaluations of cytotoxicity and PI3K inhibitory activity SH Abbas, AA Abd El-Hafeez, ME Shoman, MM Montano, HA Hassan Bioorganic chemistry 82, 360-377, 2019 | 55 | 2019 |
Novel quinoline incorporating 1, 2, 4-triazole/oxime hybrids: synthesis, molecular docking, anti-inflammatory, COX inhibition, ulceroginicity and histopathological investigations AM Mohassab, HA Hassan, D Abdelhamid, M Abdel-Aziz, KN Dalby, ... Bioorganic chemistry 75, 242-259, 2017 | 51 | 2017 |
STAT3 transcription factor as target for anti-cancer therapy AM Mohassab, HA Hassan, D Abdelhamid, M Abdel-Aziz Pharmacological Reports 72, 1101-1124, 2020 | 50 | 2020 |
Design, synthesis, molecular docking, anti-Proteus mirabilis and urease inhibition of new fluoroquinolone carboxylic acid derivatives MAA Abdullah, GEDAA Abuo-Rahma, ESMN Abdelhafez, HA Hassan, ... Bioorganic Chemistry 70, 1-11, 2017 | 46 | 2017 |
NO-releasing STAT3 inhibitors suppress BRAF-mutant melanoma growth TS Kaoud, AM Mohassab, HA Hassan, C Yan, SX Van Ravenstein, ... European Journal of Medicinal Chemistry 186, 111885, 2020 | 32 | 2020 |
JNK signaling as a target for anticancer therapy KS Abdelrahman, HA Hassan, SA Abdel-Aziz, AA Marzouk, A Narumi, ... Pharmacological Reports 73, 405-434, 2021 | 27 | 2021 |
1-Malonyl-1, 4-dihydropyridine as a novel carrier for specific delivery of drugs to the brain HA Hassan, M Abdel-Aziz, GEDAA Abuo-Rahma, HH Farag Bioorganic & Medicinal Chemistry 17 (4), 1681-1692, 2009 | 27 | 2009 |
Novel 4-(piperazin-1-yl) quinolin-2 (1H)-one bearing thiazoles with antiproliferative activity through VEGFR-2-TK inhibition A Hassan, M Badr, HA Hassan, D Abdelhamid, GEDA Abuo‐Rahma Bioorganic & Medicinal Chemistry 40, 116168, 2021 | 25 | 2021 |
New acyloxy nitroso compounds with improved water solubility and nitroxyl (HNO) release kinetics and inhibitors of platelet aggregation HAH Mohamed, M Abdel-Aziz, GEDAA Abuo-Rahma, SB King Bioorganic & medicinal chemistry 23 (17), 6069-6077, 2015 | 24 | 2015 |
Structure-based design, synthesis and antiproliferative action of new quinazoline-4-one/chalcone hybrids as EGFR inhibitors M Hisham, HA Hassan, HAM Gomaa, BGM Youssif, AM Hayallah, ... Journal of Molecular Structure 1254, 132422, 2022 | 23 | 2022 |
Design, synthesis, anticonvulsant activity, and pharmacophore study of new 1,5-diaryl-1H-1,2,4-triazole-3-carboxamide derivatives AH Abuelhassan, MM Badran, HA Hassan, D Abdelhamed, S Elnabtity, ... Medicinal Chemistry Research 27, 928-938, 2018 | 20 | 2018 |
New quinoline/1, 2, 4-triazole hybrids as dual inhibitors of COX-2/5-LOX and inflammatory cytokines: Design, synthesis, and docking study AM Mohassab, HA Hassan, D Abdelhamid, AM Gouda, HAM Gomaa, ... Journal of Molecular Structure 1244, 130948, 2021 | 19 | 2021 |
Fluoroquinolones as urease inhibitors: anti-Proteus mirabilis activity and molecular docking studies MA Abdullah, RMA El-Baky, HA Hassan, ESMN Abdelhafez, ... Am J Microbiol Res 4 (3), 81-84, 2016 | 18 | 2016 |
Recent prospectives of anticancer histone deacetylase inhibitors SA Abbass, HA Hassan, MFA Mohamed, GAI Moustafa, ... Journal of advanced Biomedical and Pharmaceutical Sciences 2 (4), 135-151, 2019 | 17 | 2019 |
Facile one-pot three-component synthesis of 4,6-diaryl-3,4-dihydropyrimidine-2(1H)-thiones under ultrasonic irradiation SA Abbass, GAI Moustafa, HA Hassan, GEDA Abuo-Rahma Synthetic Communications 49 (21), 2995-3000, 2019 | 12 | 2019 |
Design, synthesis, in vitro antiproliferative evaluation and in silico studies of new VEGFR-2 inhibitors based on 4-piperazinylquinolin-2 (1H)-one scaffold A Hassan, M Badr, D Abdelhamid, HA Hassan, MAS Abourehab, ... Bioorganic Chemistry 120, 105631, 2022 | 11 | 2022 |
Design, synthesis and antifungal activity of 1, 2, 4-triazole/or 1, 3, 4-oxadiazole-ciprofloxacin hybrids HAA Ezelarab, HA Hassan, SH Abbas, A El-Baky, M Rehab, ... Journal of advanced Biomedical and Pharmaceutical Sciences 1 (2), 78-84, 2018 | 9 | 2018 |
Nicotinonitrile as an essential scaffold in medicinal chemistry: an updated review (2015–present) H Hassan, M Hisham, M Osman, A Hayallah Journal of advanced Biomedical and Pharmaceutical Sciences 6 (1), 1-11, 2023 | 7 | 2023 |