Water structure recovery in chaotropic anion recognition: high‐affinity binding of dodecaborate clusters to γ‐cyclodextrin KI Assaf, MS Ural, F Pan, T Georgiev, S Simova, K Rissanen, D Gabel, ... Angewandte Chemie International Edition 54 (23), 6852-6856, 2015 | 257 | 2015 |
Cross-reactivity to glutamate carboxypeptidase III causes undesired salivary gland and kidney uptake of PSMA-targeted small-molecule radionuclide therapeutics L Lucaroni, T Georgiev, E Prodi, S Puglioli, C Pellegrino, N Favalli, L Prati, ... European Journal of Nuclear Medicine and Molecular Imaging 50 (3), 957-961, 2023 | 25 | 2023 |
Mn-and Co-catalyzed aminocyclizations of unsaturated hydrazones providing a broad range of functionalized pyrazolines M Balkenhohl, S Kölbl, T Georgiev, EM Carreira JACS Au 1 (7), 919-924, 2021 | 24 | 2021 |
Carboxylate Salt Bridge‐Mediated Enamine Catalysis: Expanded Michael Reaction Substrate Scope and Facile Access to Antidepressant (R)‐Pristiq TC Nugent, HAED Hussein, S Ahmed, FT Najafian, I Hussain, T Georgiev, ... Advanced Synthesis & Catalysis 359 (16), 2824-2831, 2017 | 12 | 2017 |
Cobalt-Catalyzed Aerobic Aminocyclization of Unsaturated Amides for the Synthesis of Functionalized γ-and δ-Lactams M Freis, M Balkenhohl, DM Fischer, T Georgiev, RC Sarott, EM Carreira Organic Letters 25 (34), 6380-6384, 2023 | 1 | 2023 |
Response to: GCP III is not the “off-target” for urea-based PSMA-ligands G Bassi, S Cazzamalli, S Oehler, L Lucaroni, T Georgiev, N Favalli, D Neri European Journal of Nuclear Medicine and Molecular Imaging 50 (10), 2947-2949, 2023 | 1 | 2023 |
Targeted interleukin-2 enhances the in vivo anti-cancer activity of Pluvicto™ T Georgiev, L Principi, A Galbiati, E Gilardoni, D Neri, S Cazzamalli European Journal of Nuclear Medicine and Molecular Imaging 51 (8), 2332-2337, 2024 | | 2024 |
First-in-class ACP3 high-affinity ligands isolated from DNA-Encoded Chemical Libraries for the delivery of radionuclides against prostate cancer S Cazzamalli, T Georgiev, F Migliorini, A Ciamarone, M Müller, ... Journal of Nuclear Medicine 65 (supplement 2), 241120-241120, 2024 | | 2024 |
DNA-encoded chemical libraries enable the discovery of potent PSMA-ligands with substantially reduced affinity towards the GCPIII anti-target L Lucaroni, S Oehler, T Georgiev, M Müller, M Bocci, R De Luca, N Favalli, ... Chemical Science 15 (18), 6789-6799, 2024 | | 2024 |
Biomimetic Synthesis of Nor‐Cedrene and Nor‐Isozizaene Sesquiterpenoids and Exploration of Their Olfactive Properties T Georgiev, N Armanino Chemistry–A European Journal 28 (46), e202201037, 2022 | | 2022 |