| Structure–activity relationship of purine and pyrimidine nucleotides as ecto-5′-nucleotidase (CD73) inhibitors A Junker, C Renn, C Dobelmann, V Namasivayam, S Jain, K Losenkova, ... Journal of medicinal chemistry 62 (7), 3677-3695, 2019 | 61 | 2019 |
| Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists A Junker, R Balasubramanian, A Ciancetta, E Uliassi, E Kiselev, ... Journal of Medicinal Chemistry 59 (13), 6149-6168, 2016 | 43 | 2016 |
| Synthesis of thiophene-based TAK-779 analogues by C–H arylation A Junker, J Yamaguchi, K Itami, B Wünsch The Journal of Organic Chemistry 78 (11), 5579-5586, 2013 | 34 | 2013 |
| Synthesis and Structure− Activity Relationships of Imidazopyridine/Pyrimidine‐and Furopyridine‐Based Anti‐infective Agents against Trypanosomiases DG Silva, A Junker, SMG de Melo, F Fumagalli, JR Gillespie, N Molasky, ... ChemMedChem 16 (6), 966-975, 2021 | 18 | 2021 |
| Synthesis, binding affinity and structure–activity relationships of novel, selective and dual targeting CCR2 and CCR5 receptor antagonists A Junker, AK Kokornaczyk, AJM Zweemer, B Frehland, D Schepmann, ... Organic & Biomolecular Chemistry 13 (8), 2407-2422, 2015 | 18 | 2015 |
| Discovery of potent cholinesterase inhibition-based multi-target-directed lead compounds for synaptoprotection in Alzheimer’s disease B Turgutalp, P Bhattarai, T Ercetin, C Luise, R Reis, EE Gurdal, A Isaak, ... Journal of medicinal chemistry 65 (18), 12292-12318, 2022 | 17 | 2022 |
| Automated counting of cancer cells by ensembling deep features Q Liu, A Junker, K Murakami, P Hu Cells 8 (9), 1019, 2019 | 17 | 2019 |
| Synthesis and biological evaluation of chemokine receptor ligands with 2-benzazepine scaffold S Thum, AK Kokornaczyk, T Seki, M De Maria, NVO Zacarias, H de Vries, ... European Journal of Medicinal Chemistry 135, 401-413, 2017 | 16 | 2017 |
| Selective and dual targeting of CCR2 and CCR5 receptors: a current overview A Junker, AK Kokornaczyk, AK Strunz, B Wünsch Chemokines: Chemokines and Their Receptors in Drug Discovery, 187-241, 2015 | 16 | 2015 |
| Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2) AK Strunz, AJM Zweemer, C Weiss, D Schepmann, A Junker, LH Heitman, ... Bioorganic & Medicinal Chemistry 23 (14), 4034-4049, 2015 | 13 | 2015 |
| A novel convolutional regression network for cell counting Q Liu, A Junker, K Murakami, P Hu 2019 IEEE 7th International Conference on Bioinformatics and Computational …, 2019 | 12 | 2019 |
| Diverse modifications of the 4-methylphenyl moiety of TAK-779 by late-stage Suzuki–Miyaura cross-coupling A Junker, D Schepmann, J Yamaguchi, K Itami, A Faust, K Kopka, ... Organic & Biomolecular Chemistry 12 (1), 177-186, 2014 | 10 | 2014 |
| Spotlight on P2X7 Receptor PET Imaging: A Bright Target or a Failing Star? S Schmidt, A Isaak, A Junker International journal of molecular sciences 24 (2), 1374, 2023 | 9 | 2023 |
| Structure–Activity Relationship of 3-Methylcytidine-5′-α, β-methylenediphosphates as CD73 Inhibitors M Scortichini, RM Idris, S Moschütz, A Keim, V Salmaso, C Dobelmann, ... Journal of medicinal chemistry 65 (3), 2409-2433, 2022 | 8 | 2022 |
| Structure-activity relationships of pyrimidine nucleotides containing a 5′-α, β-methylene diphosphonate at the P2Y6 receptor P Oliva, M Scortichini, C Dobelmann, S Jain, V Gopinatth, KS Toti, ... Bioorganic & medicinal chemistry letters 45, 128137, 2021 | 8 | 2021 |
| Piperazine squaric acid diamides, a novel class of allosteric P2X7 receptor antagonists M Patberg, A Isaak, F Füsser, NVO Zacarías, L Vinnenberg, J Schulte, ... European Journal of Medicinal Chemistry 226, 113838, 2021 | 7 | 2021 |
| Development of the first potential nonpeptidic positron emission tomography tracer for the imaging of CCR2 receptors S Wagner, F de Moura Gatti, DG Silva, NV Ortiz Zacarias, AJM Zweemer, ... ChemMedChem 16 (4), 640-645, 2021 | 7 | 2021 |
| Effects of axonal demyelination, inflammatory cytokines and divalent cation chelators on thalamic HCN channels and oscillatory bursting T Oniani, L Vinnenberg, R Chaudhary, JA Schreiber, K Riske, B Williams, ... International Journal of Molecular Sciences 23 (11), 6285, 2022 | 5 | 2022 |
| Microwave-Assisted Synthesis, Structure, and Preliminary Biological Evaluation of Novel 6-Methoxy-5, 6-dihydro-5-azapurines AI Siutkina, S Kalinina, R Liu, LH Heitman, A Junker, CG Daniliuc, ... ACS omega 8 (15), 14097-14112, 2023 | 4 | 2023 |
| Unveiling the Structure–Activity Relationships at the Orthosteric Binding Site of P2X Ion Channels: The Route to Selectivity A Isaak, C Dobelmann, FT Fusser, KS Erlitz, O Koch, A Junker Journal of Medicinal Chemistry 65 (16), 11291-11308, 2022 | 3 | 2022 |
