Kinetically guided radical-based synthesis of C(sp3)−C(sp3) linkages on DNA J Wang, H Lundberg, S Asai, P Martín-Acosta, JS Chen, S Brown, ... Proceedings of the National Academy of Sciences 115 (28), E6404-E6410, 2018 | 150 | 2018 |
PROTACs to address the challenges facing small molecule inhibitors P Martín-Acosta, X Xiao European journal of medicinal chemistry 210, 112993, 2021 | 98 | 2021 |
Microwave-Assisted Organocatalytic Intramolecular Knoevenagel/Hetero Diels–Alder Reaction with O-(Arylpropynyloxy)-Salicylaldehydes: Synthesis of Polycyclic … P Martín-Acosta, G Feresin, A Tapia, A Estévez-Braun The Journal of Organic Chemistry 81 (20), 9738-9756, 2016 | 39 | 2016 |
Domino synthesis of embelin derivatives with antibacterial activity R Peña, P Martín, GE Feresin, A Tapia, F Machín, A Estévez-Braun Journal of natural products 79 (4), 970-977, 2016 | 31 | 2016 |
A new family of densely functionalized fused-benzoquinones as potent human protein kinase CK2 inhibitors P Martin-Acosta, S Haider, A Amesty, D Aichele, J Jose, A Estévez-Braun European Journal of Medicinal Chemistry 144, 410-423, 2018 | 21 | 2018 |
Design, synthesis and biological evaluation of new embelin derivatives as CK2 inhibitors S Oramas-Royo, S Haidar, A Amesty, P Martin-Acosta, G Feresin, A Tapia, ... Bioorganic Chemistry 95, 103520, 2020 | 15 | 2020 |
JKST6, a novel multikinase modulator of the BCR-ABL1/STAT5 signaling pathway that potentiates direct BCR-ABL1 inhibition and overcomes imatinib resistance in chronic … H Aranda-Tavío, C Recio, P Martín-Acosta, M Guerra-Rodríguez, ... Biomedicine & Pharmacotherapy 144, 112330, 2021 | 10 | 2021 |
5-Ethynylarylnaphthalimides as antitumor agents: Synthesis and biological evaluation P Quintana-Espinoza, P Martin-Acosta, Á Amesty, P Martin-Rodriguez, ... Bioorganic & Medicinal Chemistry 25 (6), 1976-1983, 2017 | 9 | 2017 |
Synthesis of Quinoline and Dihydroquinoline Embelin Derivatives as Cardioprotective Agents P Martín-Acosta, I Cuadrado, L González-Cofrade, R Pestano, ... Journal of Natural Products 86 (2), 317-329, 2023 | 7 | 2023 |
Modular Synthesis and Antiproliferative Activity of New Dihydro-1H-pyrazolo[1,3-b]pyridine Embelin Derivatives P Martín-Acosta, Á Amesty, M Guerra-Rodríguez, B Guerra, ... Pharmaceuticals 14 (10), 1026, 2021 | 7 | 2021 |
A clickable photoaffinity probe of betulinic acid identifies tropomyosin as a target P Martín-Acosta, Q Meng, J Klimek, AP Reddy, L David, SK Petrie, BX Li, ... Acta Pharmaceutica Sinica B 12 (5), 2406-2416, 2022 | 6 | 2022 |
Efficient multicomponent synthesis of diverse antibacterial embelin-privileged structure conjugates P Martín-Acosta, R Peña, G Feresin, A Tapia, I Lorenzo-Castrillejo, ... Molecules 25 (14), 3290, 2020 | 4 | 2020 |
Mechanistic insights into the activation of ester prodrugs of 666-15 F Xie, P Martín-Acosta, BX Li, X Xiao Bioorganic & medicinal chemistry letters 30 (19), 127455, 2020 | 3 | 2020 |
Síntesis dominó de compuestos quinónicos con potencial actividad frente a dianas de interés farmacológico P Martín Acosta Síntesis dominó de compuestos quinónicos con potencial actividad frente a …, 2019 | 2 | 2019 |
Síntesis dominó de compuestos quinónicos con potencial actividad frente a dianas de interés farmacológico PM Acosta Universidad de La Laguna, 2019 | | 2019 |
Design, synthesis and biological evaluation of new embelin derivatives as CK2 Inhibitors AM Estévez Braun, SM Oramas-Royo, S Haidar, ÁE Amesty Arrieta, ... | | |