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Vishal Verma
Vishal Verma
在 gene.com 的电子邮件经过验证
标题
引用次数
引用次数
年份
Function-oriented synthesis, step economy, and drug design
PA Wender, VA Verma, TJ Paxton, TH Pillow
Accounts of chemical research 41 (1), 40-49, 2008
12482008
Structural basis for dual-mode inhibition of the ABC transporter MsbA
H Ho, A Miu, MK Alexander, NK Garcia, A Oh, I Zilberleyb, M Reichelt, ...
Nature 557 (7704), 196-201, 2018
1642018
Design, synthesis, and evaluation of potent bryostatin analogs that modulate PKC translocation selectivity
PA Wender, JL Baryza, SE Brenner, BA DeChristopher, BA Loy, ...
Proceedings of the National Academy of Sciences 108 (17), 6721-6726, 2011
1222011
Pharmacological inhibition of fatty acid synthase (FAS): a novel therapeutic approach for breast cancer chemoprevention through its ability to suppress Her‐2/neu (erbB‐2 …
JA Menendez, I Mehmi, VA Verma, PK Teng, R Lupu
Molecular Carcinogenesis: Published in cooperation with the University of …, 2004
1072004
Actin is the primary cellular receptor of bistramide A
AV Statsuk, R Bai, JL Baryza, VA Verma, E Hamel, PA Wender, ...
Nature Chemical Biology 1 (7), 383-388, 2005
1012005
Discovery of peptidomimetic antibody–drug conjugate linkers with enhanced protease specificity
BQ Wei, J Gunzner-Toste, H Yao, T Wang, J Wang, Z Xu, J Chen, J Wai, ...
Journal of medicinal chemistry 61 (3), 989-1000, 2018
942018
A TRPA1 inhibitor suppresses neurogenic inflammation and airway contraction for asthma treatment
A Balestrini, V Joseph, M Dourado, RM Reese, SD Shields, L Rougé, ...
Journal of Experimental Medicine 218 (4), 2021
862021
A cellular model of Alzheimer's disease therapeutic efficacy: PKC activation reverses Aβ-induced biomarker abnormality on cultured fibroblasts
TK Khan, TJ Nelson, VA Verma, PA Wender, DL Alkon
Neurobiology of disease 34 (2), 332-339, 2009
842009
The cryptophycins as potent payloads for antibody drug conjugates
VA Verma, TH Pillow, L DePalatis, G Li, GL Phillips, AG Polson, HE Raab, ...
Bioorganic & medicinal chemistry letters 25 (4), 864-868, 2015
692015
Disrupting gram-negative bacterial outer membrane biosynthesis through inhibition of the lipopolysaccharide transporter MsbA
MK Alexander, A Miu, A Oh, M Reichelt, H Ho, C Chalouni, S Labadie, ...
Antimicrobial Agents and Chemotherapy 62 (11), 10.1128/aac. 01142-18, 2018
672018
2′-azido substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
V Girijavallabhan, FG Njoroge, S Bogen, F Bennett, V Verma, ...
US Patent 9,156,872, 2015
672015
The design, synthesis, and evaluation of C7 diversified bryostatin analogs reveals a hot spot for PKC affinity
PA Wender, VA Verma
Organic letters 10 (15), 3331-3334, 2008
652008
Inhibition of tumor-associated fatty acid synthase activity antagonizes estradiol-and tamoxifen-induced agonist transactivation of estrogen receptor (ER) in human endometrial …
JA Menendez, BP Oza, E Atlas, VA Verma, I Mehmi, R Lupu
Oncogene 23 (28), 4945-4958, 2004
622004
2′-substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
V Girijavallabhan, FG Njoroge, S Bogen, V Verma, F Bennett, A Kerekes, ...
US Patent 9,061,041, 2015
592015
Total synthesis and initial biological evaluation of new B-ring-modified bryostatin analogs
PA Wender, JC Horan, VA Verma
Organic Letters 8 (23), 5299-5302, 2006
522006
Curse or cure? A perspective on the developability of aldehydes as active pharmaceutical ingredients
C Gampe, VA Verma
Journal of Medicinal Chemistry 63 (23), 14357-14381, 2020
472020
Design, synthesis, and biological evaluation of a potent, PKC selective, B-ring analog of bryostatin
PA Wender, VA Verma
Organic Letters 8 (9), 1893-1896, 2006
432006
Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
A Arasappan, FG Njoroge, CD Kwong, S Ananthan, F Bennett, J Clark, ...
US Patent 8,697,694, 2014
422014
Discovery of a Potent (4R,5S)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug …
H Chen, M Volgraf, S Do, A Kolesnikov, DG Shore, VA Verma, E Villemure, ...
Journal of Medicinal Chemistry 61 (8), 3641-3659, 2018
412018
Peptidomimetic compounds and antibody-drug conjugates thereof
J Flygare, J Gunzner-Toste, T Pillow, B Safina, V Verma, BQ Wei, G Zhao, ...
US Patent 10,533,058, 2020
322020
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