Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ... Science signaling 13 (625), eaaz3140, 2020 | 262 | 2020 |
Morphine‐induced respiratory depression is independent of β‐arrestin2 signalling A Kliewer, A Gillis, R Hill, F Schmiedel, C Bailey, E Kelly, G Henderson, ... British journal of pharmacology 177 (13), 2923-2931, 2020 | 224 | 2020 |
Critical assessment of G protein-biased agonism at the μ-opioid receptor A Gillis, A Kliewer, E Kelly, G Henderson, MJ Christie, S Schulz, M Canals Trends in pharmacological sciences 41 (12), 947-959, 2020 | 128 | 2020 |
Intrinsic efficacy of opioid ligands and its importance for apparent bias, operational analysis, and therapeutic window A Gillis, V Sreenivasan, MJ Christie Molecular pharmacology 98 (4), 410-424, 2020 | 67 | 2020 |
A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor Z Dekan, S Sianati, A Yousuf, KJ Sutcliffe, A Gillis, C Mallet, P Singh, ... Proceedings of the National Academy of Sciences 116 (44), 22353-22358, 2019 | 42 | 2019 |
Opioid overdose and tolerance: is the recruitment of β-arrestin to the µ-receptor involved? A Gillis, MJ Christie Neuropsychopharmacology 46 (13), 2226-2227, 2021 | 6 | 2021 |
Peripheral administration of selective glycine transporter-2 inhibitor, oleoyl-d-lysine, reverses chronic neuropathic pain but not acute or inflammatory pain in male mice BS Wilson, J Peiser-Oliver, A Gillis, S Evans, C Alamein, SN Mostyn, ... Journal of Pharmacology and Experimental Therapeutics 382 (3), 246-255, 2022 | 2 | 2022 |
Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists (vol 13, eaaz3140, 2020) A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ... SCIENCE SIGNALING 14 (670), 2021 | 1 | 2021 |
Peripheral administration of selective GlyT2 inhibitor, oleoyl-D-lysine, is analgesic in neuropathic but not acute or inflammatory pain models in mice B Wilson, J Peiser-Oliver, A Gillis, S Evans, C Alamein, S Mostyn, ... Authorea Preprints, 2021 | | 2021 |
µ-opioid receptor ligand pharmacology in cell and animal models A Gillis University of Sydney, 2020 | | 2020 |
View metadata, citation and similar papers at core. ac. uk A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ... | | |