关注
Vangelis Agouridas
Vangelis Agouridas
Centrale Lille Institut
在 centralelille.fr 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Native chemical ligation and extended methods: mechanisms, catalysis, scope, and limitations
V Agouridas, O El Mahdi, V Diemer, M Cargoet, JCM Monbaliu, O Melnyk
Chemical reviews 119 (12), 7328-7443, 2019
4762019
A statistical view of protein chemical synthesis using NCL and extended methodologies
V Agouridas, O El Mahdi, M Cargoët, O Melnyk
Bioorganic & Medicinal Chemistry 25 (18), 4938-4945, 2017
762017
Total synthesis of discodermolide: optimization of the effective synthetic route
E de Lemos, FH Porée, A Bourin, J Barbion, E Agouridas, MI Lannou, ...
Chemistry–A European Journal 14 (35), 11092-11112, 2008
572008
Design and synthesis of ansamycin antibiotics
IE Wrona, V Agouridas, JS Panek
Comptes Rendus Chimie 11 (11-12), 1483-1522, 2008
452008
From protein total synthesis to peptide transamidation and metathesis: playing with the reversibility of N, S-acyl or N, Se-acyl migration reactions
O Melnyk, V Agouridas
Current Opinion in Chemical Biology 22, 137-145, 2014
362014
Chemical Protein Synthesis in Medicinal Chemistry: Miniperspective
V Agouridas, O El Mahdi, O Melnyk
Journal of Medicinal Chemistry 63 (24), 15140-15152, 2020
282020
M. Cargo t, J.-CM Monbaliu, O. Melnyk
V Agouridas, O El Mahdi, V Diemer
Chem. Rev 119, 7328-7443, 2019
272019
A cysteine selenosulfide redox switch for protein chemical synthesis
V Diemer, N Ollivier, B Leclercq, H Drobecq, J Vicogne, V Agouridas, ...
Nature Communications 11 (1), 2558, 2020
252020
Catalysis of Thiol–Thioester Exchange by Water-Soluble Alkyldiselenols Applied to the Synthesis of Peptide Thioesters and SEA-Mediated Ligation
M Cargoët, V Diemer, B Snella, R Desmet, A Blanpain, H Drobecq, ...
The Journal of organic chemistry 83 (20), 12584-12594, 2018
252018
Cyclic Sulfamidates as Vehicles for the Synthesis of Poly- and Diversely Substituted Benzosultams via Unusual S(O)2−O Bond Cleavage
M Lorion, V Agouridas, A Couture, E Deniau, P Grandclaudon
Organic Letters 12 (6), 1356-1359, 2010
242010
Loss of antagonistic activity of tamoxifen by replacement of one N-methyl of its side chain by fluorinated residues
V Agouridas, I Laı, A Cleeren, E Kizilian, E Magnier, JC Blazejewski, ...
Bioorganic & medicinal chemistry 14 (22), 7531-7538, 2006
222006
Strategies and open questions in solid-phase protein chemical synthesis
V Agouridas, V Diemer, O Melnyk
Current Opinion in Chemical Biology 58, 1-9, 2020
212020
Native chemical ligation at serine revisited
B Snella, V Diemer, H Drobecq, V Agouridas, O Melnyk
Organic Letters 20 (23), 7616-7619, 2018
162018
Pedal to the metal: The homogeneous catalysis of the native chemical ligation reaction
V Diemer, O Firstova, V Agouridas, O Melnyk
Chemistry–A European Journal 28 (16), e202104229, 2022
152022
Conception, synthesis, and biological evaluation of original discodermolide analogues
E de Lemos, E Agouridas, G Sorin, A Guerreiro, A Commerçon, ...
Chemistry–A European Journal 17 (36), 10123-10134, 2011
152011
Effect of fluorination on the pharmacological profile of 11β isomers of fulvestrant in breast carcinoma cells
V Agouridas, E Magnier, JC Blazejewski, I Laïos, A Cleeren, D Nonclercq, ...
Journal of medicinal chemistry 52 (3), 883-887, 2009
152009
Cesium carbonate mediated aryl triflate esters’ deprotection
AE Green, V Agouridas, E Deniau
Tetrahedron Letters 54 (51), 7078-7079, 2013
142013
A highly diastereoselective synthesis of isoindolinone-centered Meyers’ tetracyclic lactams. Application to the asymmetric synthesis of 3-alkylisoindolinones
V Agouridas, F Capet, A Couture, E Deniau, P Grandclaudon
Tetrahedron: Asymmetry 22 (13), 1441-1447, 2011
142011
Total chemical synthesis of proteins
A Brik, P Dawson, L Liu
John Wiley & Sons, 2021
132021
Synthesis and cytotoxic evaluation of cis-locked and constrained analogues of combretastatin and combretastatin A4
M Lorion, V Agouridas, A Couture, E Deniau, P Grandclaudon
Tetrahedron Letters 51 (39), 5146-5149, 2010
122010
系统目前无法执行此操作,请稍后再试。
文章 1–20