关注
Abdulmalik S. AlTamimi
Abdulmalik S. AlTamimi
Prince Sattam Bin Abdulaziz University - PhD Associate prof. - Head of Pharmaceutical Chemistry
在 psau.edu.sa 的电子邮件经过验证
标题
引用次数
引用次数
年份
Synthesis and antimicrobial activity of novel 5-(1-adamantyl)-2-aminomethyl-4-substituted-1, 2, 4-triazoline-3-thiones
AA El-Emam, AMS Al-Tamimi, MA Al-Omar, KA Alrashood, EE Habib
European journal of medicinal chemistry 68, 96-102, 2013
1022013
Carbonic anhydrase inhibition and the management of glaucoma: a literature and patent review 2013-2019
CT Supuran, ASA Altamimi, F Carta
Expert opinion on therapeutic patents 29 (10), 781-792, 2019
632019
Discovery of novel nonsteroidal anti-inflammatory drugs and carbonic anhydrase inhibitors hybrids (NSAIDs–CAIs) for the management of rheumatoid arthritis
O Akgul, L Di Cesare Mannelli, D Vullo, A Angeli, C Ghelardini, ...
Journal of Medicinal Chemistry 61 (11), 4961-4977, 2018
532018
Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae
AM Alafeefy, M Ceruso, AMS Al-Tamimi, S Del Prete, C Capasso, ...
Bioorganic & Medicinal Chemistry 22 (19), 5133-5140, 2014
502014
Inhibition of carbonic anhydrases from the extremophilic bacteria Sulfurihydrogenibium yellostonense (SspCA) and S. azorense (SazCA) with a new series of sulfonamides …
AM Alafeefy, HA Abdel-Aziz, D Vullo, AMS Al-Tamimi, NA Al-Jaber, ...
Bioorganic & medicinal chemistry 22 (1), 141-147, 2014
472014
Inhibition studies of quinazoline-sulfonamide derivatives against the γ-CA (PgiCA) from the pathogenic bacterium, Porphyromonas gingivalis
AM Alafeefy, M Ceruso, AMS Al-Tamimi, SD Prete, CT Supuran, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 30 (4), 592-596, 2015
462015
Structural and spectroscopic characterization of a novel potential chemotherapeutic agent 3-(1-adamantyl)-1-{[4-(2-methoxyphenyl) piperazin-1-yl] methyl}-4-methyl-1H-1, 2, 4 …
AA El-Emam, AMS Al-Tamimi, KA Al-Rashood, HN Misra, V Narayan, ...
Journal of Molecular Structure 1022, 49-60, 2012
422012
A review on epidermal growth factor receptor's role in breast and non-small cell lung cancer
V Subramaniyan, S Fuloria, G Gupta, DH Kumar, M Sekar, KV Sathasivam, ...
Chemico-biological interactions 351, 109735, 2022
412022
Development of certain new 2-substituted-quinazolin-4-yl-aminobenzenesulfonamide as potential antitumor agents
AM Alafeefy, R Ahmad, M Abdulla, WM Eldehna, AMS Al-Tamimi, ...
European Journal of Medicinal Chemistry 109, 247-253, 2016
412016
Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-,[1, 2, 4] triazolo [3, 4-b][1, 3, 4 …
AM Alafeefy, HA Abdel-Aziz, D Vullo, AMS Al-Tamimi, AS Awaad, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 30 (1), 52-56, 2015
412015
Discovery of new organoselenium compounds as antileishmanial agents
AMS Al-Tamimi, M Etxebeste-Mitxeltorena, C Sanmartin, A Jimenez-Ruiz, ...
Bioorganic Chemistry 86, 339-345, 2019
352019
Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity
M Bozdag, AM Alafeefy, AM Altamimi, D Vullo, F Carta, CT Supuran
Bioorganic & Medicinal Chemistry 25 (2), 677-683, 2017
352017
Carbonic anhydrase inhibitors based on sorafenib scaffold: design, synthesis, crystallographic investigation and effects on primary breast cancer cells
M Bozdag, M Ferraroni, C Ward, F Carta, S Bua, A Angeli, SP Langdon, ...
European Journal of Medicinal Chemistry 182, 111600, 2019
292019
Synthesis and Antimicrobial Activity of N′-Heteroarylidene-1-adamantylcarbohydrazides and (±)-2-(1-Adamantyl)-4-acetyl-5-[5-(4-substituted phenyl-3-isoxazolyl …
AA El-Emam, KA Alrashood, MA Al-Omar, AMS Al-Tamimi
Molecules 17 (3), 3475-3483, 2012
292012
Cationic solid lipid nanoparticles of resveratrol for hepatocellular carcinoma treatment: systematic optimization, in vitro characterization and preclinical investigation
M Rahman, WH Almalki, O Afzal, AS Alfawaz Altamimi, I Kazmi, ...
International Journal of Nanomedicine, 9283-9299, 2020
282020
3-(1-Adamantyl)-1-{[4-(2-methoxyphenyl) piperazin-1-yl] methyl}-4-methyl-1H-1, 2, 4-triazole-5 (4H)-thione
A Al-Tamimi, A Bari, MA Al-Omar, KA Alrashood, AA El-Emam
Acta Crystallographica Section E: Structure Reports Online 66 (7), o1756-o1756, 2010
282010
Sodium alginate based drug delivery in management of breast cancer
MAJ Shaikh, KS Alharbi, WH Almalki, SS Imam, M Albratty, AM Meraya, ...
Carbohydrate polymers 292, 119689, 2022
262022
Drug delivery challenges and current progress in nanocarrier-based ocular therapeutic system
MH Akhter, I Ahmad, MY Alshahrani, AI Al-Harbi, H Khalilullah, O Afzal, ...
Gels 8 (2), 82, 2022
242022
Investigation of potential anti-malarial lead candidate 2-(4-fluorobenzylthio)-5-(5-bromothiophen-2-yl)-1, 3, 4-oxadiazole: Insights from crystal structure, DFT, QTAIM and …
LH Al-Wahaibi, NS Kumar, AA El-Emam, NS Venkataramanan, ...
Journal of Molecular Structure 1175, 230-240, 2019
242019
Neuroprotective role of chrysin‐loaded poly (lactic‐co‐glycolic acid) nanoparticle against kindling‐induced epilepsy through Nrf2/ARE/HO‐1 pathway
Y Zhang, J Zhao, O Afzal, I Kazmi, FA Al‐Abbasi, ASA Altamimi, Z Yang
Journal of Biochemical and Molecular Toxicology 35 (2), e22634, 2021
232021
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