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Yaser A. Mostafa
Yaser A. Mostafa
Associate Professor of Pharmaceutical Organic Chemistry, Assiut University
在 pharm.aun.edu.eg 的电子邮件经过验证
标题
引用次数
引用次数
年份
Thiohydantoin derivatives incorporating a pyrazole core: Design, synthesis and biological evaluation as dual inhibitors of topoisomerase-I and cycloxygenase-2 with anti-cancer …
KRA Abdellatif, WAA Fadaly, YA Mostafa, DM Zaher, HA Omar
Bioorganic Chemistry 91, 103132, 2019
502019
Synthesis and antimicrobial activity of certain new 1, 2, 4-triazolo [1, 5-a] pyrimidine derivatives
YAH Mostafa, MA Hussein, AA Radwan, AEHN Kfafy
Archives of pharmacal research 31, 279-293, 2008
422008
Steroid derivatives as inhibitors of steroid sulfatase
YAM Abdel-Karem
Journal of Steroid Biochemistry & Molecular Biology 137, 183– 198, 2013
40*2013
Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives
CM Phan, Y Liu, B Kim, Y Mostafa, SD Taylor
Bioorganic & medicinal chemistry 19 (20), 5999-6005, 2011
372011
Discovery of new pyrimido [5, 4-c] quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studies
RA Mekheimer, SMR Allam, MA Al-Sheikh, MS Moustafa, SM Al-Mousawi, ...
Bioorganic Chemistry 121, 105693, 2022
332022
Antioxidant and Wound Healing Potential of Vitis vinifera Seeds Supported by Phytochemical Characterization and Docking Studies
T Al-Warhi, EM Zahran, S Selim, MM Al-Sanea, MM Ghoneim, SA Maher, ...
Antioxidants 11 (5), 881, 2022
312022
A first-in-class anticancer dual HDAC2/FAK inhibitors bearing hydroxamates/benzamides capped by pyridinyl-1, 2, 4-triazoles
M Mustafa, AA Abd El-Hafeez, D Abdelhamid, GD Katkar, YA Mostafa, ...
European journal of medicinal chemistry 222, 113569, 2021
262021
17β-Arylsulfonamides of 17β-aminoestra-1, 3, 5 (10)-trien-3-ol as highly potent inhibitors of steroid sulfatase
YA Mostafa, SD Taylor
Bioorganic & medicinal chemistry 20 (4), 1535-1544, 2012
242012
A facile synthesis, drug-likeness, and in silico molecular docking of certain new azidosulfonamide–chalcones and their in vitro antimicrobial activity
M Mustafa, YA Mostafa
Monatshefte für Chemie-Chemical Monthly 151, 417-427, 2020
212020
Novel piperine-carboximidamide hybrids: Design, synthesis, and antiproliferative activity via a multi-targeted inhibitory pathway
LH Al-Wahaibi, MA Mahmoud, YA Mostafa, AE Raslan, BGM Youssif
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 376-386, 2023
192023
Wound Healing and Antioxidant Capabilities of Zizyphus mauritiana Fruits: In-Vitro, In-Vivo, and Molecular Modeling Study
NH Shady, R Soltane, SA Maher, EA Saber, MA Elrehany, YA Mostafa, ...
Plants 11 (11), 1392, 2022
192022
Antimicrobial pyridazines: synthesis, characterization, cytotoxicity, substrate promiscuity, and molecular docking
M Mustafa, YA Mostafa
Chemistry & Biodiversity 17 (6), e2000100, 2020
192020
Synthesis and biological evaluation of indole-2-carboxamides with potent apoptotic antiproliferative activity as egfr/cdk2 dual inhibitors
LH Al-Wahaibi, YA Mostafa, MH Abdelrahman, AH El-Bahrawy, ...
Pharmaceuticals 15 (8), 1006, 2022
182022
Novel urea linked ciprofloxacin-chalcone hybrids having antiproliferative topoisomerases I/II inhibitory activities and caspases-mediated apoptosis
HHH Mohammed, SH Abbas, AM Hayallah, GEDA Abuo-Rahma, ...
Bioorganic Chemistry 106, 104422, 2021
182021
Novel 1, 5-diaryl pyrazole-3-carboxamides as selective COX-2/sEH inhibitors with analgesic, anti-inflammatory, and lower cardiotoxicity effects
OM Hendawy, HAM Gomaa, SI Alzarea, MS Alshammari, FAM Mohamed, ...
Bioorganic Chemistry 116, 105302, 2021
162021
FAK inhibitors as promising anticancer targets: present and future directions
M Mustafa, AA Abd El-Hafeez, DA Abdelhafeez, D Abdelhamid, ...
Future medicinal chemistry 13 (18), 1559-1590, 2021
152021
A-ring substituted 17β-arylsulfonamides of 17β-aminoestra-1, 3, 5 (10)-trien-3-ol as highly potent reversible inhibitors of steroid sulfatase
YA Mostafa, B Kralt, PPN Rao, SD Taylor
Bioorganic & Medicinal Chemistry 23 (17), 5681-5692, 2015
142015
Discovery of novel oxazole-based macrocycles as anti-coronaviral agents targeting SARS-CoV-2 main protease
LH Al-Wahaibi, A Mostafa, YA Mostafa, OF Abou-Ghadir, AH Abdelazeem, ...
Bioorganic Chemistry 116, 105363, 2021
132021
Discovery of new cyanopyridine/chalcone hybrids as dual inhibitors of EGFR/BRAFV600E with promising antiproliferative properties
HA Abou‐Zied, EAM Beshr, HAM Gomaa, YA Mostafa, BGM Youssif, ...
Archiv der Pharmazie 356 (4), 2200464, 2023
122023
Novel indazole derivatives as potent apoptotic antiproliferative agents by multi-targeted mechanism: Synthesis and biological evaluation
FOA Frejat, H Zhai, Y Cao, L Wang, YA Mostafa, HAM Gomaa, ...
Bioorganic Chemistry 126, 105922, 2022
102022
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