| Macrocycles in drug discovery─ learning from the past for the future D Garcia Jimenez, V Poongavanam, J Kihlberg Journal of Medicinal Chemistry 66 (8), 5377-5396, 2023 | 67 | 2023 |
| Designing soluble PROTACs: strategies and preliminary guidelines D García Jiménez, M Rossi Sebastiano, M Vallaro, V Mileo, D Pizzirani, ... Journal of Medicinal Chemistry 65 (19), 12639-12649, 2022 | 41 | 2022 |
| Rational control of molecular properties is mandatory to exploit the potential of PROTACs as oral drugs G Ermondi, D Garcia Jimenez, M Rossi Sebastiano, G Caron ACS Medicinal Chemistry Letters 12 (7), 1056-1060, 2021 | 29 | 2021 |
| Protacs and building blocks: the 2d chemical space in very early drug discovery G Ermondi, D Garcia-Jimenez, G Caron Molecules 26 (3), 672, 2021 | 29 | 2021 |
| Are we ready to design oral PROTACs®? DG Jimenez, J Sebastiano, M Rossi, G Caron, G Ermondi ADMET and DMPK 9 (4), 243-254, 2021 | 19 | 2021 |
| Refinement of computational access to molecular physicochemical properties: From Ro5 to bRo5 M Rossi Sebastiano, D Garcia Jimenez, M Vallaro, G Caron, G Ermondi Journal of Medicinal Chemistry 65 (18), 12068-12083, 2022 | 11 | 2022 |
| Chamelogk: A chromatographic Chameleonicity quantifier to design orally bioavailable beyond-rule-of-5 drugs D Garcia Jimenez, M Vallaro, M Rossi Sebastiano, G Apprato, ... Journal of Medicinal Chemistry 66 (15), 10681-10693, 2023 | 8 | 2023 |
| Conformational sampling deciphers the chameleonic properties of a VHL-based degrader G Ermondi, DG Jimenez, M Rossi Sebastiano, J Kihlberg, G Caron Pharmaceutics 15 (1), 272, 2023 | 7 | 2023 |
| Exploring the chemical space of orally bioavailable PROTACs G Apprato, V Poongavanam, DG Jimenez, Y Atilaw, M Erdelyi, G Ermondi, ... Drug Discovery Today, 103917, 2024 | 3 | 2024 |
| IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs D Garcia Jimenez, M Rossi Sebastiano, M Vallaro, G Ermondi, G Caron Journal of Medicinal Chemistry, 2024 | | 2024 |
| IMHB-Mediated Chameleonicity in Drug Design: A Focus on Structurally Related PROTACs DG Jimenez, MR Sebastiano, M Vallaro, G Ermondi, G Caron Journal of medicinal chemistry, 0 | | |
