| Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment A Angeli, F Carta, A Nocentini, JY Winum, R Zalubovskis, A Akdemir, ... Metabolites 10 (10), 412, 2020 | 128 | 2020 |
| New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors HI Gul, C Yamali, H Sakagami, A Angeli, J Leitans, A Kazaks, K Tars, ... Bioorganic Chemistry 77, 411-419, 2018 | 110 | 2018 |
| Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase A Nocentini, A Angeli, F Carta, JY Winum, R Zalubovskis, S Carradori, ... Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 561-580, 2021 | 89 | 2021 |
| Synthesis of coumarin-sulfonamide derivatives and determination of their cytotoxicity, carbonic anhydrase inhibitory and molecular docking studies BZ Kurt, F Sonmez, D Ozturk, A Akdemir, A Angeli, CT Supuran European Journal of Medicinal Chemistry 183, 111702, 2019 | 74 | 2019 |
| Synthesis and anti-inflammatory activity of sulfonamides and carboxylates incorporating trimellitimides: dual cyclooxygenase/carbonic anhydrase inhibitory actions AM Alaa, A Angeli, AS El-Azab, MEA Hammouda, MA El-Sherbeny, ... Bioorganic chemistry 84, 260-268, 2019 | 70 | 2019 |
| Selenols: A new class of carbonic anhydrase inhibitors A Angeli, D Tanini, A Nocentini, A Capperucci, M Ferraroni, P Gratteri, ... Chemical communications 55 (5), 648-651, 2019 | 68 | 2019 |
| Discovery of novel nonsteroidal anti-inflammatory drugs and carbonic anhydrase inhibitors hybrids (NSAIDs–CAIs) for the management of rheumatoid arthritis O Akgul, L Di Cesare Mannelli, D Vullo, A Angeli, C Ghelardini, ... Journal of Medicinal Chemistry 61 (11), 4961-4977, 2018 | 66 | 2018 |
| Discovery of new selenoureido analogues of 4-(4-fluorophenylureido) benzenesulfonamide as carbonic anhydrase inhibitors A Angeli, D Tanini, TS Peat, L Di Cesare Mannelli, G Bartolucci, ... ACS medicinal chemistry letters 8 (9), 963-968, 2017 | 64 | 2017 |
| Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1, 2, 4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and … M Krasavin, A Shetnev, T Sharonova, S Baykov, T Tuccinardi, S Kalinin, ... Bioorganic Chemistry 76, 88-97, 2018 | 62 | 2018 |
| Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo [d] thiazole-5-and 6-sulfonamides M Abdoli, A Angeli, M Bozdag, F Carta, A Kakanejadifard, H Saeidian, ... Journal of Enzyme Inhibition and Medicinal Chemistry 32 (1), 1071-1078, 2017 | 61 | 2017 |
| Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines NMA Gawad, NH Amin, MT Elsaadi, FMM Mohamed, A Angeli, V De Luca, ... Bioorganic & medicinal chemistry 24 (13), 3043-3051, 2016 | 61 | 2016 |
| Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases L De Luca, F Mancuso, S Ferro, MR Buemi, A Angeli, S Del Prete, ... European journal of medicinal chemistry 143, 276-282, 2018 | 60 | 2018 |
| Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors C Melis, R Meleddu, A Angeli, S Distinto, G Bianco, C Capasso, ... Journal of enzyme inhibition and medicinal chemistry 32 (1), 68-73, 2017 | 58 | 2017 |
| Microwave-assisted extraction, HPLC analysis, and inhibitory effects on carbonic anhydrase I, II, VA, and VII isoforms of 14 blueberry Italian cultivars A Mollica, M Locatelli, G Macedonio, S Carradori, AP Sobolev, ... Journal of enzyme inhibition and medicinal chemistry 31 (sup4), 1-6, 2016 | 58 | 2016 |
| Synthesis, biological activity and multiscale molecular modeling studies of bis-coumarins as selective carbonic anhydrase IX and XII inhibitors with effective cytotoxicity … BZ Kurt, A Dag, B Doğan, S Durdagi, A Angeli, A Nocentini, CT Supuran, ... Bioorganic Chemistry 87, 838-850, 2019 | 56 | 2019 |
| Discovery of New Potential Anti‐Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target‐Focused Repurposing Approaches G Annunziato, A Angeli, F D'Alba, A Bruno, M Pieroni, D Vullo, V De Luca, ... ChemMedChem 11 (17), 1904-1914, 2016 | 55 | 2016 |
| Synthesis and biological evaluation of coumarin-1, 3, 4-oxadiazole hybrids as selective carbonic anhydrase IX and XII inhibitors SG Narella, MG Shaik, A Mohammed, M Alvala, A Angeli, CT Supuran Bioorganic chemistry 87, 765-772, 2019 | 52 | 2019 |
| Structural investigations on coumarins leading to chromeno [4, 3-c] pyrazol-4-ones and pyrano [4, 3-c] pyrazol-4-ones: New scaffolds for the design of the tumor-associated … A Bonardi, M Falsini, D Catarzi, F Varano, LDC Mannelli, B Tenci, ... European Journal of Medicinal Chemistry 146, 47-59, 2018 | 52 | 2018 |
| Bioactive isoflavones from Pueraria lobata root and starch: Different extraction techniques and carbonic anhydrase inhibition A Mocan, S Carradori, M Locatelli, D Secci, S Cesa, A Mollica, S Riga, ... Food and chemical toxicology 112, 441-447, 2018 | 52 | 2018 |
| Discovery of benzenesulfonamides with potent human carbonic anhydrase inhibitory and effective anticonvulsant action: design, synthesis, and pharmacological assessment CB Mishra, S Kumari, A Angeli, SM Monti, M Buonanno, M Tiwari, ... Journal of Medicinal Chemistry 60 (6), 2456-2469, 2017 | 52 | 2017 |
Fabrizio CartaUniversita' di Firenze-Dept. Neurofarba在 unifi.it 的电子邮件经过验证
