A glycopeptide dendrimer inhibitor of the galactose-specific lectin LecA and of Pseudomonas aeruginosa biofilms RU Kadam, M Bergmann, M Hurley, D Garg, M Cacciarini, MA Swiderska, ... Angewandte Chemie (International ed. in English) 50 (45), 10631, 2011 | 193 | 2011 |
A small-molecule fusion inhibitor of influenza virus is orally active in mice MJP van Dongen, RU Kadam, J Juraszek, E Lawson, B Brandenburg, ... Science 363 (6431), eaar6221, 2019 | 119 | 2019 |
CH−π “T-Shape” Interaction with Histidine Explains Binding of Aromatic Galactosides to Pseudomonas aeruginosa Lectin LecA RU Kadam, D Garg, J Schwartz, R Visini, M Sattler, A Stocker, T Darbre, ... ACS chemical biology 8 (9), 1925-1930, 2013 | 112 | 2013 |
Computer-assisted methods in chemical toxicity prediction C Gopi Mohan, T Gandhi, D Garg, R Shinde Mini reviews in medicinal chemistry 7 (5), 499-507, 2007 | 91 | 2007 |
Exploring QSTR and toxicophore of hERG K+ channel blockers using GFA and HypoGen techniques D Garg, T Gandhi, CG Mohan Journal of Molecular Graphics and Modelling 26 (6), 966-976, 2008 | 64 | 2008 |
Novel approaches for targeting thymidylate synthase to overcome the resistance and toxicity of anticancer drugs D Garg, S Henrich, OMH Salo-Ahen, H Myllykallio, MP Costi, RC Wade Journal of medicinal chemistry 53 (18), 6539-6549, 2010 | 61 | 2010 |
Epigallocatechin gallate (EGCG) reduces the intensity of pancreatic amyloid fibrils in human islet amyloid polypeptide (hIAPP) transgenic mice A Franko, DC Rodriguez Camargo, A Böddrich, D Garg, ... Scientific reports 8 (1), 1116, 2018 | 54 | 2018 |
Structure‐Based Optimization of the Terminal Tripeptide in Glycopeptide Dendrimer Inhibitors of Pseudomonas aeruginosa Biofilms Targeting LecA RU Kadam, M Bergmann, D Garg, G Gabrieli, A Stocker, T Darbre, ... Chemistry–A European Journal 19 (50), 17054-17063, 2013 | 47 | 2013 |
Advances in targeting nucleocapsid–nucleic acid interactions in HIV-1 therapy D Garg, BE Torbett Virus research 193, 135-143, 2014 | 37 | 2014 |
hIAPP forms toxic oligomers in plasma DCR Camargo, D Garg, K Buday, A Franko, AR Camargo, F Schmidt, ... Chemical Communications 54 (43), 5426-5429, 2018 | 30 | 2018 |
Identification of phenothiazine derivatives as UHM-binding inhibitors of early spliceosome assembly PKA Jagtap, T Kubelka, K Soni, CL Will, D Garg, C Sippel, TG Kapp, ... Nature Communications 11 (1), 5621, 2020 | 26 | 2020 |
Rational design of cyclic peptide inhibitors of U2AF homology motif (UHM) domains to modulate pre-mRNA splicing PKA Jagtap, D Garg, TG Kapp, CL Will, O Demmer, R Lührmann, ... Journal of medicinal chemistry 59 (22), 10190-10197, 2016 | 26 | 2016 |
Synthesis, biological evaluation and molecular docking of aryl hydrazines and hydrazides for anticancer activity VM Gohil, SK Agrawal, AK Saxena, D Garg, C Gopimohan, KK Bhutani CSIR, 2010 | 16 | 2010 |
Evaluation of proinflammatory cytokine pathway inhibitors for p38 MAPK inhibitory potential RU Kadam, D Garg, AT Paul, KK Bhutani, N Roy Journal of medicinal chemistry 50 (25), 6337-6342, 2007 | 13 | 2007 |
Evaluation of Pseudomonas aeruginosa Deacetylase LpxC Inhibitory Activity of Dual PDE4−TNFα Inhibitors: A Multiscreening Approach RU Kadam, D Garg, A Chavan, N Roy Journal of chemical information and modeling 47 (3), 1188-1195, 2007 | 12 | 2007 |
Translational repression of thymidylate synthase by targeting its mRNA D Garg, AV Beribisky, G Ponterini, A Ligabue, G Marverti, A Martello, ... Nucleic acids research 41 (7), 4159-4170, 2013 | 9 | 2013 |
Conservation and role of electrostatics in thymidylate synthase D Garg, S Skouloubris, J Briffotaux, H Myllykallio, RC Wade Scientific reports 5 (1), 17356, 2015 | 8 | 2015 |
Selective Mapping of Chemical Space for Pseudomonas aeruginosa Deacetylase LpxC Inhibitory Potential RU Kadam, D Garg, N Roy Chemical biology & drug design 71 (1), 45-56, 2008 | 3 | 2008 |
An orally active small molecule fusion inhibitor of influenza virus MJP van Dongen, RU Kadam, J Juraszek, E Lawson, B Brandenburg, ... Science (New York, NY) 363 (6431), 2019 | | 2019 |
CH-π RU Kadam, D Garg, J Schwartz, R Visini, M Sattler, A Stocker, T Darbre, ... ACS chemical biology, 2013 | | 2013 |