关注
Peter Keov
Peter Keov
在 monash.edu 的电子邮件经过验证
标题
引用次数
引用次数
年份
Allosteric modulation of G protein-coupled receptors: a pharmacological perspective
P Keov, PM Sexton, A Christopoulos
Neuropharmacology 60 (1), 24-35, 2011
2992011
The TRPV4 agonist GSK1016790A regulates the membrane expression of TRPV4 channels
S Baratchi, P Keov, WG Darby, A Lai, K Khoshmanesh, P Thurgood, ...
Frontiers in pharmacology 10, 6, 2019
792019
Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptor
P Keov, L Lopez, SM Devine, C Valant, JR Lane, PJ Scammells, ...
Journal of Biological Chemistry 289 (34), 23817-23837, 2014
732014
Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor
A Abdul-Ridha, L Lopez, P Keov, DM Thal, SN Mistry, PM Sexton, ...
Journal of Biological Chemistry 289 (9), 6067-6079, 2014
732014
Development of a human vasopressin V1a-receptor antagonist from an evolutionary-related insect neuropeptide
MG Di Giglio, M Muttenthaler, K Harpsøe, Z Liutkeviciute, P Keov, T Eder, ...
Scientific Reports 7 (1), 41002, 2017
422017
Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M1 muscarinic acetylcholine receptor
P Keov, C Valant, SM Devine, JR Lane, PJ Scammells, PM Sexton, ...
Molecular Pharmacology 84 (3), 425-437, 2013
402013
Contractility measurements of human uterine smooth muscle to aid drug development
S Arrowsmith, P Keov, M Muttenthaler, CW Gruber
JoVE (Journal of Visualized Experiments), e56639, 2018
372018
AM833 is a novel agonist of calcitonin family G protein–coupled receptors: pharmacological comparison with six selective and nonselective agonists
MM Fletcher, P Keov, TT Truong, G Mennen, CA Hick, P Zhao, ...
Journal of Pharmacology and Experimental Therapeutics 377 (3), 417-440, 2021
332021
Cyclotides isolated from an ipecac root extract antagonize the corticotropin releasing factor type 1 receptor
M Fahradpour, P Keov, C Tognola, E Perez-Santamarina, PJ McCormick, ...
Frontiers in Pharmacology 8, 616, 2017
322017
Discovery of peptide probes to modulate oxytocin-type receptors of insects
P Keov, Z Liutkevičiūtė, R Hellinger, RJ Clark, CW Gruber
Scientific reports 8 (1), 10020, 2018
172018
Nature-inspired dimerization as a strategy to modulate neuropeptide pharmacology exemplified with vasopressin and oxytocin
Z Dekan, T Kremsmayr, P Keov, M Godin, N Teakle, L Dürrauer, H Xiang, ...
Chemical Science 12 (11), 4057-4062, 2021
162021
Orphan receptor GPR37L1 remains unliganded
T Ngo, BP Wilkins, SS So, P Keov, KK Chahal, AM Finch, JLJ Coleman, ...
Nature chemical biology 17 (4), 383-386, 2021
102021
Tackling the complexities of orphan GPCR ligand discovery with rationally assisted approaches
SS So, T Ngo, P Keov, NJ Smith, I Kufareva
GPCRs, 295-334, 2020
92020
I8-arachnotocin–an arthropod-derived G protein-biased ligand of the human vasopressin V2 receptor
L Duerrauer, E Muratspahić, J Gattringer, P Keov, HC Mendel, ...
Scientific Reports 9 (1), 19295, 2019
82019
Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor
N Tomašević, FS Emser, E Muratspahić, J Gattringer, S Hasinger, ...
Journal of Biological Chemistry 300 (6), 107330, 2024
2024
Development of a Novel Assay for Direct Assessment of Selective Amylin Receptor Activation Reveals Novel Differences in Behavior of Selective and Nonselective Peptide Agonists
P Keov, G Christopoulos, CA Hick, T Glendorf, B Ballarín-González, ...
Molecular Pharmacology 105 (5), 359-373, 2024
2024
Role of G protein‐coupled receptor kinases (GRKs) in β2‐adrenoceptor‐mediated glucose uptake
S Ham, S Mukaida, M Sato, P Keov, T Bengtsson, S Furness, ND Holliday, ...
Pharmacology Research & Perspectives 12 (1), e1176, 2024
2024
Orphan G protein-coupled receptor, GPR37L1: pharmacological toolbox empty once again
T Ngo, BP Wilkins, SS So, P Keov, KK Chahal, AM Finch, JLJ Coleman, ...
bioRxiv, 2020.09. 11.290486, 2020
2020
Pharmacological Characterisation of the Cyclotide Kalata B7 At Insect Orthologues of the Oxytocin/vasopressin Receptors
P Keov, Z Liutkeviciute, R Clark, C Gruber
Journal Of Peptide Science 22, S86-S86, 2016
2016
Structural and mechanistic studies of novel selective agonists of the M1 muscarinic acetylcholine receptor
P Keov
Monash University, 2014
2014
系统目前无法执行此操作,请稍后再试。
文章 1–20