| cis-Peptide bond mimetic tetrazole analogs of the insect kinins identify the active conformation RJ Nachman, J Zabrocki, J Olczak, HJ Williams, G Moyna, AI Scott, ... Peptides 23 (4), 709-716, 2002 | 59 | 2002 |
| Constrained peptidomimetics for TRH: cis-peptide bond analogs Y Tong, J Olczak, J Zabrocki, MC Gershengorn, GR Marshall, KD Moeller Tetrahedron 56 (50), 9791-9800, 2000 | 54 | 2000 |
| Synthesis of quaternary α-amino acid-based arginase inhibitors via the Ugi reaction A Golebiowski, D Whitehouse, RP Beckett, M Van Zandt, MK Ji, TR Ryder, ... Bioorganic & medicinal chemistry letters 23 (17), 4837-4841, 2013 | 51 | 2013 |
| Chitinases and chitinase-like proteins as therapeutic targets in inflammatory diseases, with a special focus on inflammatory bowel diseases M Mazur, A Zielińska, MM Grzybowski, J Olczak, J Fichna International Journal of Molecular Sciences 22 (13), 6966, 2021 | 44 | 2021 |
| Targeting acidic mammalian chitinase is effective in animal model of asthma M Mazur, J Olczak, S Olejniczak, R Koralewski, W Czestkowski, ... Journal of Medicinal Chemistry 61 (3), 695-710, 2018 | 36 | 2018 |
| Discovery and pharmacokinetics of sulfamides and guanidines as potent human arginase 1 inhibitors R Blaszczyk, J Brzezinska, B Dymek, PS Stanczak, M Mazurkiewicz, ... ACS Medicinal Chemistry Letters 11 (4), 433-438, 2020 | 32 | 2020 |
| Development of dual chitinase inhibitors as potential new treatment for respiratory system diseases M Mazur, B Dymek, R Koralewski, P Sklepkiewicz, S Olejniczak, ... Journal of Medicinal Chemistry 62 (15), 7126-7145, 2019 | 28 | 2019 |
| Discovery of OATD-01, a First-in-Class Chitinase Inhibitor as Potential New Therapeutics for Idiopathic Pulmonary Fibrosis R Koralewski, B Dymek, M Mazur, P Sklepkiewicz, S Olejniczak, ... Journal of Medicinal Chemistry 63 (24), 15527-15540, 2020 | 27 | 2020 |
| X-ray and nuclear magnetic resonance (NMR) studies of signalizing the tripeptide sequence (Tyr-D-Ala-Phe) of dermorphin and deltorphins I and II. Comparative analysis in the … MM Słabicki, MJ Potrzebowski, G Bujacz, S Olejniczak, J Olczak The Journal of Physical Chemistry B 108 (14), 4535-4545, 2004 | 26 | 2004 |
| Antarctic, cold-adapted beta-galactosidase of Pseudoalteromonas sp. 22b as an effective tool for alkyl galactopyranosides synthesis K Makowski, A Białkowska, J Olczak, J Kur, M Turkiewicz Enzyme And Microbial Technology 44, 59–64, 2009 | 24 | 2009 |
| Can the 1, 5-disubstituted tetrazole ring modify the co-ordinating ability and biological activity of opiate-like peptides? E Lodyga-Chruscinska, E Brzezinska-Blaszczyk, G Micera, D Sanna, ... Journal of Inorganic Biochemistry 78 (4), 283-291, 2000 | 23 | 2000 |
| OATD-02 validates the benefits of pharmacological inhibition of arginase 1 and 2 in cancer MM Grzybowski, PS Stańczak, P Pomper, R Błaszczyk, B Borek, A Gzik, ... Cancers 14 (16), 3967, 2022 | 20 | 2022 |
| Specific interactions of bovine and human β-casomorphin-7 with Cu (II) ions E Chruścińska, J Olczak, J Zabrocki, M Dyba, G Micera, D Sanna, ... Journal of inorganic biochemistry 69 (1-2), 91-95, 1998 | 19 | 1998 |
| Impact of 1, 5-disubstituted tetrazole ring on chelating ability of δ-selective opioid peptide E Łodyga-Chruścińska, S Ołdziej, G Micera, D Sanna, L Chruściński, ... Journal of inorganic biochemistry 98 (3), 447-458, 2004 | 18 | 2004 |
| Novel glycosylated endomorphin-2 analog produces potent centrally-mediated antinociception in mice after peripheral administration J Fichna, M Mazur, D Grzywacz, W Kamysz, R Perlikowska, J Piekielna, ... Bioorganic & medicinal chemistry letters 23 (24), 6673-6676, 2013 | 17 | 2013 |
| Antinociceptive and antidepressant-like action of endomorphin-2 analogs with proline surrogates in position 2 R Perlikowska, J Piekielna, M Mazur, R Koralewski, J Olczak, JC do Rego, ... Bioorganic & medicinal chemistry 22 (17), 4803-4809, 2014 | 16 | 2014 |
| Effect of the tetrazole cis-amide bond surrogate on the complexing ability of some enkephalin analogues toward Cu (II) ions E Lodyga-Chruscinska, G Micera, D Sanna, J Olczak, J Zabrocki, ... Journal of inorganic biochemistry 76 (1), 1-11, 1999 | 16 | 1999 |
| Consequences of cis-amide bond simulation in opioid peptides J Olczak, K Kaczmarek, I Maszczyńska, M Lisowski, D Stropova, VJ Hruby, ... Letters in Peptide Science 5, 437-440, 1998 | 16 | 1998 |
| Arginase inhibitors and their therapeutic applications R Blaszczyk, J Brzezińska, A Gzik, A Golebiowski, J Nowicka, B Borek, ... US Patent 10,391,077, 2019 | 14 | 2019 |
| Discovery of selective, orally bioavailable inhibitor of mouse chitotriosidase M Mazur, A Bartoszewicz, B Dymek, M Salamon, G Andryianau, ... Bioorganic & medicinal chemistry letters 28 (3), 310-314, 2018 | 14 | 2018 |
Adam GolebiowskiVP Research, OncoArendi Therapeutics在 oncoarendi.com 的电子邮件经过验证
