Moderating strain without sacrificing reactivity: design of fast and tunable noncatalyzed alkyne–azide cycloadditions via stereoelectronically controlled transition state … B Gold, GB Dudley, IV Alabugin Journal of the American Chemical Society 135 (4), 1558-1569, 2013 | 156 | 2013 |
Selective transition state stabilization via hyperconjugative and conjugative assistance: stereoelectronic concept for copper-free click chemistry B Gold, NE Shevchenko, N Bonus, GB Dudley, IV Alabugin The Journal of organic chemistry 77 (1), 75-89, 2012 | 138 | 2012 |
“Two functional groups in one package”: using both alkyne π-bonds in cascade transformations IV Alabugin, B Gold The Journal of Organic Chemistry 78 (16), 7777-7784, 2013 | 119 | 2013 |
Alkenes as Alkyne Equivalents in Radical Cascades Terminated by Fragmentations: Overcoming Stereoelectronic Restrictions on Ring Expansions For the Preparation of Expanded … R Mohamed, S Mondal, B Gold, CJ Evoniuk, T Banerjee, K Hanson, ... Journal of the American Chemical Society 137 (19), 6335-6349, 2015 | 92 | 2015 |
1, 3-Dipolar cycloadditions of diazo compounds in the presence of azides MR Aronoff, B Gold, RT Raines Organic letters 18 (7), 1538-1541, 2016 | 86 | 2016 |
Fine-tuning strain and electronic activation of strain-promoted 1, 3-dipolar cycloadditions with endocyclic sulfamates in SNO-OCTs EG Burke, B Gold, TT Hoang, RT Raines, JM Schomaker Journal of the American Chemical Society 139 (23), 8029-8037, 2017 | 72 | 2017 |
Design of Leaving Groups in Radical C C Fragmentations: Through‐Bond 2c–3e Interactions in Self‐Terminating Radical Cascades S Mondal, B Gold, RK Mohamed, IV Alabugin Chemistry–A European Journal 20 (28), 8664-8669, 2014 | 71 | 2014 |
Sub-picomolar inhibition of HIV-1 protease with a boronic acid IW Windsor, MJ Palte, JC Lukesh III, B Gold, KT Forest, RT Raines Journal of the American Chemical Society 140 (43), 14015-14018, 2018 | 64 | 2018 |
Boronic acid with high oxidative stability and utility in biological contexts BJ Graham, IW Windsor, B Gold, RT Raines Proceedings of the National Academy of Sciences 118 (10), e2013691118, 2021 | 63 | 2021 |
Divergent Cyclizations of 1-R-Ethynyl-9,10-anthraquinones: Use of Thiourea as a “S2–” Equivalent in an “Anchor-Relay” Addition Mediated by Formal C–H Activation DS Baranov, B Gold, SF Vasilevsky, IV Alabugin The Journal of Organic Chemistry 78 (5), 2074-2082, 2013 | 42 | 2013 |
1, 3-Dipolar cycloaddition with diazo groups: Noncovalent interactions overwhelm strain B Gold, MR Aronoff, RT Raines Organic letters 18 (18), 4466-4469, 2016 | 39 | 2016 |
Decreasing distortion energies without strain: Diazo-selective 1, 3-dipolar cycloadditions B Gold, MR Aronoff, RT Raines The Journal of organic chemistry 81 (14), 5998-6006, 2016 | 39 | 2016 |
Alkynyl crown ethers as a scaffold for hyperconjugative assistance in noncatalyzed azide–alkyne click reactions: ion sensing through enhanced transition-state stabilization B Gold, P Batsomboon, GB Dudley, IV Alabugin The Journal of Organic Chemistry 79 (13), 6221-6232, 2014 | 39 | 2014 |
Single-Crystal X-ray Structure of 1,3- dimethylcyclobutadiene IV Alabugin, B Gold, M Shatruk, K Kovnir Science 330, 1047, 2010 | 36* | 2010 |
Rerouting radical cascades: intercepting the homoallyl ring expansion in enyne cyclizations via C–S scission S Mondal, B Gold, RK Mohamed, H Phan, IV Alabugin The Journal of Organic Chemistry 79 (16), 7491-7501, 2014 | 32 | 2014 |
Strain control in nucleophilic cyclizations: reversal of exo‐selectivity in cyclizations of hydrazides of acetylenyl carboxylic acids by annealing to a pyrazole scaffold SF Vasilevsky, B Gold, TF Mikhailovskaya, IV Alabugin Journal of Physical Organic Chemistry 25 (11), 998-1005, 2012 | 31 | 2012 |
Chameleonic reactivity of vicinal diazonium salt of acetylenyl-9, 10-anthraquinones: Synthetic application toward two heterocyclic targets AA Stepanov, LM Gornostaev, SF Vasilevsky, EV Arnold, VI Mamatyuk, ... The Journal of Organic Chemistry 76 (21), 8737-8748, 2011 | 31 | 2011 |
An n→π* Interaction in the Bound Substrate of Aspartic Proteases Replicates the Oxyanion Hole IW Windsor, B Gold, RT Raines ACS catalysis 9 (2), 1464-1471, 2018 | 28 | 2018 |
Rapid cycloaddition of a diazo group with an unstrained dipolarophile MR Aronoff, B Gold, RT Raines Tetrahedron letters 57 (22), 2347-2350, 2016 | 28 | 2016 |
Urea as an organic solvent and reagent for the addition/cyclization/fragmentation cascades leading to 2-R-7 H-dibenzo [de, h] quinolin-7-one analogues of Aporphinoid alkaloids DS Baranov, SF Vasilevsky, B Gold, IV Alabugin RSC advances 1 (9), 1745-1750, 2011 | 28 | 2011 |