Residue-specific peptide modification: a chemist’s guide JN deGruyter, LR Malins, PS Baran Biochemistry 56 (30), 3863-3873, 2017 | 474 | 2017 |
Electrochemically driven, Ni-catalyzed aryl amination: scope, mechanism, and applications Y Kawamata, JC Vantourout, DP Hickey, P Bai, L Chen, Q Hou, W Qiao, ... Journal of the American Chemical Society 141 (15), 6392-6402, 2019 | 284 | 2019 |
Unlocking P (V): Reagents for chiral phosphorothioate synthesis KW Knouse, JN deGruyter, MA Schmidt, B Zheng, JC Vantourout, ... Science 361 (6408), 1234-1238, 2018 | 190 | 2018 |
Peptide macrocyclization inspired by non-ribosomal imine natural products LR Malins, JN deGruyter, KJ Robbins, PM Scola, MD Eastgate, ... Journal of the American Chemical Society 139 (14), 5233-5241, 2017 | 119 | 2017 |
Alkyl sulfinates: radical precursors enabling drug discovery: Miniperspective JM Smith, JA Dixon, JN deGruyter, PS Baran Journal of Medicinal Chemistry 62 (5), 2256-2264, 2018 | 117 | 2018 |
Direct carbon isotope exchange through decarboxylative carboxylation C Kingston, MA Wallace, AJ Allentoff, JN deGruyter, JS Chen, SX Gong, ... Journal of the American Chemical Society 141 (2), 774-779, 2019 | 76 | 2019 |
Serine-selective bioconjugation JC Vantourout, SR Adusumalli, KW Knouse, DT Flood, A Ramirez, ... Journal of the American Chemical Society 142 (41), 17236-17242, 2020 | 72 | 2020 |
CITU: a peptide and decarboxylative coupling reagent JN Degruyter, LR Malins, L Wimmer, KJ Clay, J Lopez-Ogalla, T Qin, ... Organic letters 19 (22), 6196-6199, 2017 | 38 | 2017 |
The taumycin A macrocycle: Asymmetric total synthesis and revision of relative stereochemistry JN deGruyter, WA Maio Organic letters 16 (19), 5196-5199, 2014 | 17 | 2014 |
Magnesiate Addition/Ring-Expansion Strategy To Access the 6–7–6 Tricyclic Core of Hetisine-Type C20-Diterpenoid Alkaloids JJ Pflueger, LC Morrill, JN deGruyter, MA Perea, R Sarpong Organic letters 19 (17), 4632-4635, 2017 | 10 | 2017 |
Iminoboronate-mediated peptide cyclization with lysine homologues K Li, J Gao Synlett 28 (15), 1913-1916, 2017 | 7 | 2017 |
Synthesis of Tryptophan–Folate Conjugates K Maruyama, KJ Malawska, N Konoue, K Oisaki, M Kanai Synlett 31 (08), 784-787, 2020 | 6 | 2020 |
Solid-phase zincke reaction for the synthesis of peptide-4, 4′-bipyridinium Conjugates P Cortón, P Novo, V López-Sobrado, MD Garcia, C Peinador, E Pazos Synthesis 52 (04), 537-543, 2020 | 5 | 2020 |
E Vs Z Selectivity in Olefin Metathesis through Catalyst Design Q Michaudel, SJ Kempel, TW Hsu, N Justine Elsevier, 2022 | 4 | 2022 |
Peptide Cyclization at High Concentration RD Wills, VT Adebomi, M Raj Synlett 31 (16), 1537-1542, 2020 | 4 | 2020 |
α-Chymotrypsin-Induced Acetalization of Aldehydes and Ketones with Alcohols J Lan, G Jiang, J Yang, H Zhu, Z Le, Z Xie Synthesis 52 (14), 2121-2126, 2020 | 2 | 2020 |
Functionalized Peptides: Ideal Targets for Collaborative Chemistry JN deGruyter Biochemistry 57 (19), 2745-2746, 2018 | 1 | 2018 |
Phosphorous (v)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (v) compounds MA Schmidt, B Zheng, K Knouse, J Degruyter, MD Eastgate, P Baran, ... US Patent App. 18/167,772, 2023 | | 2023 |
Phosphorous (V)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (V) compounds MA Schmidt, B Zheng, K Knouse, J Degruyter, MD Eastgate, P Baran, ... US Patent 11,613,554, 2023 | | 2023 |
Novel phosphorous (v)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (v) compounds MA Schmidt, B Zheng, K Knouse, J Degruyter, MD Eastgate, P Baran, ... US Patent App. 16/382,692, 2019 | | 2019 |