Discovery of antimycobacterial spiro-piperidin-4-ones: An atom economic, stereoselective synthesis, and biological intervention RR Kumar, S Perumal, P Senthilkumar, P Yogeeswari, D Sriram Journal of Medicinal Chemistry 51 (18), 5731-5735, 2008 | 273 | 2008 |
A facile synthesis and antimycobacterial evaluation of novel spiro-pyrido-pyrrolizines and pyrrolidines RR Kumar, S Perumal, P Senthilkumar, P Yogeeswari, D Sriram European journal of medicinal chemistry 44 (9), 3821-3829, 2009 | 190 | 2009 |
An atom efficient, solvent-free, green synthesis and antimycobacterial evaluation of 2-amino-6-methyl-4-aryl-8-[(E)-arylmethylidene]-5, 6, 7, 8-tetrahydro-4H-pyrano [3, 2-c … RR Kumar, S Perumal, P Senthilkumar, P Yogeeswari, D Sriram Bioorganic & Medicinal Chemistry Letters 17 (23), 6459-6462, 2007 | 177 | 2007 |
A highly atom economic, chemo-, regio-and stereoselective synthesis, and discovery of spiro-pyrido-pyrrolizines and pyrrolidines as antimycobacterial agents RR Kumar, S Perumal, P Senthilkumar, P Yogeeswari, D Sriram Tetrahedron 64 (13), 2962-2971, 2008 | 94 | 2008 |
Synthesis and antimycobacterial activities of novel 6-nitroquinolone-3-carboxylic acids P Senthilkumar, M Dinakaran, P Yogeeswari, D Sriram, A China, ... European journal of medicinal chemistry 44 (1), 345-358, 2009 | 89 | 2009 |
Novel ofloxacin derivatives: Synthesis, antimycobacterial and toxicological evaluation M Dinakaran, P Senthilkumar, P Yogeeswari, A China, V Nagaraja, ... Bioorganic & Medicinal Chemistry Letters 18 (3), 1229-1236, 2008 | 87 | 2008 |
Conventional and microwave assisted synthesis of pyrazolone Mannich bases possessing anti-inflammatory, analgesic, ulcerogenic effect and antimicrobial properties KK Sivakumar, A Rajasekaran, P Senthilkumar, PP Wattamwar Bioorganic & Medicinal Chemistry Letters 24 (13), 2940-2944, 2014 | 69 | 2014 |
5-Nitrofuran-2-yl derivatives: synthesis and inhibitory activities against growing and dormant mycobacterium species D Sriram, P Yogeeswari, P Dhakla, P Senthilkumar, D Banerjee, ... Bioorganic & Medicinal Chemistry Letters 19 (4), 1152-1154, 2009 | 61 | 2009 |
Antimycobacterial activities of novel 1-(cyclopropyl/tert-butyl/4-fluorophenyl)-1, 4-dihydro-6-nitro-4-oxo-7-(substituted secondary amino)-1, 8-naphthyridine-3-carboxylic acid D Sriram, P Senthilkumar, M Dinakaran, P Yogeeswari, A China, ... Journal of medicinal chemistry 50 (24), 6232-6239, 2007 | 60 | 2007 |
Antimycobacterial activities of novel 2-(sub)-3-fluoro/nitro-5, 12-dihydro-5-oxobenzothiazolo [3, 2-a] quinoline-6-carboxylic acid M Dinakaran, P Senthilkumar, P Yogeeswari, A China, V Nagaraja, ... Bioorganic & medicinal chemistry 16 (6), 3408-3418, 2008 | 59 | 2008 |
5-Nitro-2-furoic acid hydrazones: design, synthesis and in vitro antimycobacterial evaluation against log and starved phase cultures D Sriram, P Yogeeswari, DRK Vyas, P Senthilkumar, P Bhat, M Srividya Bioorganic & medicinal chemistry letters 20 (15), 4313-4316, 2010 | 58 | 2010 |
Synthesis and Antimycobacterial Evaluation of Novel Phthalazin‐4‐ylacetamides Against log‐and Starved Phase Cultures D Sriram, P Yogeeswari, P Senthilkumar, D Sangaraju, R Nelli, ... Chemical biology & drug design 75 (4), 381-391, 2010 | 45 | 2010 |
Antimycobacterial activities of novel fluoroquinolones P Senthilkumar, M Dinakaran, P Yogeeswari, A China, V Nagaraja, ... Biomedicine & Pharmacotherapy 63 (1), 27-35, 2009 | 45 | 2009 |
Synthesis and in vitro antitubercular activity of 4-aryl/alkylsulfonylmethylcoumarins as inhibitors of Mycobacterium tuberculosis M Jeyachandran, P Ramesh, D Sriram, P Senthilkumar, P Yogeeswari Bioorganic & medicinal chemistry letters 22 (14), 4807-4809, 2012 | 41 | 2012 |
Synthesis and antimycobacterial evaluation of newer 1-cyclopropyl-1, 4-dihydro-6-fluoro-7-(substituted secondary amino)-8-methoxy-5-(sub)-4-oxoquinoline-3-carboxylic acids P Senthilkumar, M Dinakaran, D Banerjee, RV Devakaram, P Yogeeswari, ... Bioorganic & medicinal chemistry 16 (5), 2558-2569, 2008 | 34 | 2008 |
Synthesis of various 3-nitropropionamides as Mycobacterium tuberculosis isocitrate lyase inhibitor D Sriram, P Yogeeswari, S Methuku, DRK Vyas, P Senthilkumar, M Alvala, ... Bioorganic & medicinal chemistry letters 21 (18), 5149-5154, 2011 | 31 | 2011 |
N-Hydroxythiosemicarbazones: Synthesis and in vitro antitubercular activity D Sriram, P Yogeeswari, P Dhakla, P Senthilkumar, D Banerjee Bioorganic & medicinal chemistry letters 17 (7), 1888-1891, 2007 | 31 | 2007 |
Antitubercular activities of novel benzothiazolo naphthyridone carboxylic acid derivatives endowed with high activity toward multi-drug resistant tuberculosis M Dinakaran, P Senthilkumar, P Yogeeswari, D Sriram Biomedicine & Pharmacotherapy 63 (1), 11-18, 2009 | 30 | 2009 |
Novel pthalazinyl derivatives: synthesis, antimycobacterial activities, and inhibition of Mycobacterium tuberculosis isocitrate lyase enzyme D Sriram, P Yogeeswari, P Senthilkumar, S Dewakar, N Rohit, B Debjani, ... Medicinal Chemistry 5 (5), 422-422, 2009 | 26 | 2009 |
Antimycobacterial and phototoxic evaluation of novel 6-fluoro/nitro-4-oxo-7-(sub)-4H-[1, 3] thiazeto [3, 2-a] quinoline-3-carboxylic acid D Murugesan, S Palaniappan, Y Perumal, N Valakunja, D Sriram International journal of antimicrobial agents 31 (4), 337-344, 2008 | 26 | 2008 |