Enantioselective (4+ 2) Annulation of Donor–Acceptor Cyclobutanes by N‐Heterocyclic Carbene Catalysis A Levens, A Ametovski, DW Lupton Angewandte Chemie 128 (52), 16370-16374, 2016 | 51 | 2016 |
Cannabichromene, related phytocannabinoids, and 5-fluoro-cannabichromene have anticonvulsant properties in a mouse model of Dravet Syndrome LL Anderson, A Ametovski, J Lin Luo, D Everett-Morgan, IS McGregor, ... ACS chemical neuroscience 12 (2), 330-339, 2021 | 47 | 2021 |
Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB‐4en‐PICA, MDMB‐4en‐PINACA, ADB‐4en‐PINACA, and MMB‐4CN‐BUTINACA using … KE Grafinger, MM Vandeputte, A Cannaert, A Ametovski, E Sparkes, ... Drug testing and analysis 13 (7), 1412-1429, 2021 | 39 | 2021 |
Enantioselective Total Synthesis of (−)-Δ9-Tetrahydrocannabinol via N-Heterocyclic Carbene Catalysis A Ametovski, DW Lupton Organic letters 21 (4), 1212-1215, 2019 | 36 | 2019 |
Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB‐4en‐PICA, MDMB‐4en‐PINACA, ADB‐4en‐PINACA, and MMB‐4CN‐BUTINACA using … E Pike, KE Grafinger, A Cannaert, A Ametovski, JL Luo, E Sparkes, ... Drug testing and analysis 13 (7), 1383-1401, 2021 | 26 | 2021 |
Biomimetic and biocatalytic synthesis of bruceol AJ Day, JHZ Lee, QD Phan, HC Lam, A Ametovski, CJ Sumby, SG Bell, ... Angewandte Chemie International Edition 58 (5), 1427-1431, 2019 | 21 | 2019 |
Exploring stereochemical and conformational requirements at cannabinoid receptors for synthetic cannabinoids related to SDB-006, 5F-SDB-006, CUMYL-PICA, and 5F-CUMYL-PICA A Ametovski, C Macdonald, JJ Manning, SAS Haneef, M Santiago, ... ACS Chemical Neuroscience 11 (21), 3672-3682, 2020 | 18 | 2020 |
NNL-3: a synthetic intermediate or a new class of hydroxybenzotriazole esters with cannabinoid receptor activity? A Ametovski, EA Cairns, KE Grafinger, A Cannaert, MH Deventer, S Chen, ... ACS Chemical Neuroscience 12 (21), 4020-4036, 2021 | 8 | 2021 |
Putative Synthetic Cannabinoids MEPIRAPIM, 5F-BEPIRAPIM (NNL-2), and Their Analogues Are T-Type Calcium Channel (CaV3) Inhibitors RC Kevin, S Mirlohi, JJ Manning, R Boyd, EA Cairns, A Ametovski, F Lai, ... ACS Chemical Neuroscience 13 (9), 1395-1409, 2022 | 6 | 2022 |
In vitro evaluation of the interaction of the cannabis constituents cannabichromene and cannabichromenic acid with ABCG2 and ABCB1 transporters MG Etchart, LL Anderson, A Ametovski, PM Jones, AM George, ... European Journal of Pharmacology 922, 174836, 2022 | 5 | 2022 |
Comprehensive Characterization of a Systematic Library of Alkyl and Alicyclic Synthetic Cannabinoids Related to CUMYL-PICA, CUMYL-BUTICA, CUMYL-CBMICA, and CUMYL-PINACA LK Janssens, A Ametovski, E Sparkes, R Boyd, F Lai, CJ Maloney, ... ACS chemical neuroscience 14 (1), 35-52, 2022 | 4 | 2022 |
Synthesis and pharmacological evaluation of newly detected synthetic cannabinoid receptor agonists AB-4CN-BUTICA, MMB-4CN-BUTINACA, MDMB-4F-BUTICA, MDMB-4F-BUTINACA and their … E Sparkes, R Boyd, S Chen, JW Markham, JL Luo, T Foyzun, H Zaman, ... Frontiers in Psychiatry 13, 1010501, 2022 | 3 | 2022 |
Structure–Activity Relationships, Deuteration, and Fluorination of Synthetic Cannabinoid Receptor Agonists Related to AKB48, 5F-AKB-48, and AFUBIATA E Sparkes, CJ Maloney, JW Markham, C Dane, R Boyd, J Gilchrist, M Moir, ... ACS Chemical Neuroscience, 2024 | | 2024 |
Synthesis and Functional Evaluation of Synthetic Cannabinoid Receptor Agonists Related to ADB-HEXINACA E Sparkes, A Timmerman, JW Markham, R Boyd, R Gordon, KA Walker, ... ACS Chemical Neuroscience 15 (9), 1787-1812, 2024 | | 2024 |
Synthesis and functional evaluation of proteinogenic amino acid-derived synthetic cannabinoid receptor agonists related to MPP-5F-PICA, MMB-5F-PICA, and MDMB-5F-PICA E Sparkes, JW Markham, R Boyd, M Udoh, R Gordon, H Zaman, ... RSC Medicinal Chemistry, 2024 | | 2024 |
MEPIRAPIM-derived synthetic cannabinoids inhibit T-type calcium channels with divergent effects on seizures in rodent models of epilepsy T Harman, M Udoh, DL McElroy, LL Anderson, RC Kevin, SD Banister, ... Frontiers in Physiology 14, 1086243, 2023 | | 2023 |
Azaindole E Pike, KE Grafinger, A Cannaert, A Ametovski, JL Luo, E Sparkes, ... | | |
Novel N-Heterocyclic Carbene Catalysed (4+ 2) Annulations for the Synthesis of Natural Products A AMETOVSKI Monash University, 0 | | |