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Davide Cirillo
Davide Cirillo
Postdoctoral research, FMP Berlin
在 fmp-berlin.de 的电子邮件经过验证
标题
引用次数
引用次数
年份
Development of selective inhibitors of phosphatidylinositol 3-kinase C2α
WT Lo, H Belabed, M Kücükdisli, J Metag, Y Roske, P Prokofeva, ...
Nature chemical biology 19 (1), 18-27, 2023
162023
Tacrine-xanomeline and tacrine-iperoxo hybrid ligands: Synthesis and biological evaluation at acetylcholinesterase and M1 muscarinic acetylcholine receptors
M Maspero, D Volpato, D Cirillo, NY Chen, R Messerer, C Sotriffer, ...
Bioorganic chemistry 96, 103633, 2020
162020
Structure‐Activity‐Relationship‐Aided Design and Synthesis of xCT Antiporter Inhibitors
D Cirillo, S Sarowar, PØ Enger, HR Bjørsvik
ChemMedChem 16 (17), 2650-2668, 2021
72021
Isoform-selective targeting of PI3K: time to consider new opportunities?
D Cirillo, M Diceglie, M Nazaré
Trends in Pharmacological Sciences, 2023
62023
Functionalization of the Imidazole Backbone by Means of a Tailored and Optimized Oxidative Heck Cross‐Coupling
D Cirillo, F Angelucci, HR Bjørsvik
Advanced Synthesis & Catalysis 362 (22), 5079-5092, 2020
62020
The styryl benzoic acid derivative DC10 potentiates radiotherapy by targeting the xCT-glutathione Axis
S Sarowar, D Cirillo, P Játiva, MH Nilsen, SMA Otragane, J Heggdal, ...
Frontiers in Oncology 12, 786739, 2022
42022
Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition
M Kücükdisli, H Bel-Abed, D Cirillo, WT Lo, NL Efrém, A Horatscheck, ...
Journal of Medicinal Chemistry 66 (20), 14278-14302, 2023
22023
Novel Xanomeline-containing bitopic ligands of muscarinic acetylcholine receptors: design, synthesis and FRET investigation
C Matera, M Kauk, D Cirillo, M Maspero, C Papotto, D Volpato, ...
Molecules 28 (5), 2407, 2023
12023
Imidazole Backbone Functionalization with Olefin Cross‐Metathesis
F Angelucci, D Cirillo, HR Bjørsvik
European Journal of Organic Chemistry 2022 (22), e202200437, 2022
12022
A Scalable High‐Yielding and Selective Oxidative Heck Cross‐Coupling – A Key Step for the Synthesis of trans‐Stilbenes
D Cirillo, S Karlsson, HR Bjørsvik
European Journal of Organic Chemistry 2021 (40), 5519-5529, 2021
12021
Therapy
HR Bjørsvik, PØ Enger, D Cirillo, S Sarowar
US Patent App. 17/763,367, 2022
2022
Styrylbenzoic acid derivative DC10 potentiates radiotherapy by inhibiting glutathione synthesis, leading to increased oxidative stress and cancer cell death
S Sarowar, D Cirillo, P Jativa, MH Nilsen, SMA Otragane, JI Heggdal, ...
Cancer Research 82 (12_Supplement), 214-214, 2022
2022
Front Cover: Structure‐Activity‐Relationship‐Aided Design and Synthesis of xCT Antiporter Inhibitors (ChemMedChem 17/2021)
D Cirillo, S Sarowar, P Øyvind Enger, HR Bjørsvik
ChemMedChem 16 (17), 2546-2546, 2021
2021
Tacrine/Xanomeline hybrid ligands: synthesis and pharmacological evaluation at M1 muscarinic acetylcholine receptors and acetylcholinesterases
M Maspero, D Volpato, D Cirillo, U Holzgrabe, M De Amici, C Dallanoce
2018
Synthesis of a group of novel Xanomeline/77-LH-28-1 hybrid ligands and their FRET investigation at muscarinic acetylcholine receptor subtypes
D Cirillo, M Kauk, C Matera, D Volpato, U Holzgrabe, M De Amici, ...
Congresso Nazionale della Società Chimica Italiana: atti. 4: divisione di …, 2017
2017
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