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Roberta Ettari
Roberta Ettari
Associate Professor of Medicinal Chemistry, Messina University
在 unime.it 的电子邮件经过验证 - 首页
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引用次数
引用次数
年份
Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors
R Ettari, E Nizi, ME Di Francesco, MA Dude, G Pradel, R Vicík, ...
Journal of medicinal chemistry 51 (4), 988-996, 2008
2372008
Falcipain‐2 inhibitors
R Ettari, F Bova, M Zappalà, S Grasso, N Micale
Medicinal research reviews 30 (1), 136-167, 2010
1542010
BAY 11-7082 inhibits the NF-κB and NLRP3 inflammasome pathways and protects against IMQ-induced psoriasis
N Irrera, M Vaccaro, A Bitto, G Pallio, G Pizzino, M Lentini, V Arcoraci, ...
Clinical Science 131 (6), 487-498, 2017
1302017
Immunoproteasome-selective and non-selective inhibitors: A promising approach for the treatment of multiple myeloma
R Ettari, M Zappalà, S Grasso, C Musolino, V Innao, A Allegra
Pharmacology & Therapeutics 182, 176-192, 2018
1012018
Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents
N Micale, AP Kozikowski, R Ettari, S Grasso, M Zappalà, JJ Jeong, ...
Journal of medicinal chemistry 49 (11), 3064-3067, 2006
1002006
Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis
R Ettari, L Tamborini, IC Angelo, N Micale, A Pinto, C De Micheli, P Conti
Journal of Medicinal Chemistry 56 (14), 5637-5658, 2013
992013
Novel peptidomimetics containing a vinyl ester moiety as highly potent and selective falcipain-2 inhibitors
R Ettari, N Micale, T Schirmeister, C Gelhaus, M Leippe, E Nizi, ...
Journal of Medicinal Chemistry 52 (7), 2157-2160, 2009
922009
Peptide‐based proteasome inhibitors in anticancer drug design
N Micale, K Scarbaci, V Troiano, R Ettari, S Grasso, M Zappala
Medicinal research reviews 34 (5), 1001-1069, 2014
662014
Development of novel peptidomimetics containing a vinyl sulfone moiety as proteasome inhibitors
R Ettari, C Bonaccorso, N Micale, C Heindl, T Schirmeister, ML Calabrò, ...
ChemMedChem 6 (7), 1228-1237, 2011
612011
Development of novel peptide-based Michael acceptors targeting rhodesain and falcipain-2 for the treatment of Neglected Tropical Diseases (NTDs)
S Previti, R Ettari, S Cosconati, G Amendola, K Chouchene, A Wagner, ...
Journal of Medicinal Chemistry 60 (16), 6911-6923, 2017
572017
The inhibition of cysteine proteases rhodesain and TbCatB: A valuable approach to treat Human African Trypanosomiasis
R Ettari, S Previti, L Tamborini, G Cullia, S Grasso, M Zappalà
Mini reviews in medicinal chemistry 16 (17), 1374-1391, 2016
562016
Nonpeptidic vinyl and allyl phosphonates as falcipain-2 inhibitors
R Ettari, E Nizi, ME Di Francesco, N Micale, S Grasso, M Zappalà, R Vicík, ...
ChemMedChem 3 (7), 1030-1033, 2008
522008
Design and synthesis of novel isoxazole-based HDAC inhibitors
P Conti, L Tamborini, A Pinto, L Sola, R Ettari, C Mercurio, C De Micheli
European journal of medicinal chemistry 45 (9), 4331-4338, 2010
512010
Lead discovery of SARS-CoV-2 main protease inhibitors through covalent docking-based virtual screening
G Amendola, R Ettari, S Previti, C Di Chio, A Messere, S Di Maro, ...
Journal of Chemical Information and Modeling 61 (4), 2062-2073, 2021
472021
Immunoproteasome-selective inhibitors: a promising strategy to treat hematologic malignancies, autoimmune and inflammatory diseases
R Ettari, S Previti, A Bitto, S Grasso, M Zappala
Current medicinal chemistry 23 (12), 1217-1238, 2016
462016
Development of rhodesain inhibitors with a 3‐bromoisoxazoline warhead
R Ettari, L Tamborini, IC Angelo, S Grasso, T Schirmeister, L Lo Presti, ...
ChemMedChem 8 (12), 2070-2076, 2013
462013
Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain
R Ettari, M Zappalà, N Micale, T Schirmeister, C Gelhaus, M Leippe, ...
European journal of medicinal chemistry 45 (7), 3228-3233, 2010
462010
Novel 2H-isoquinolin-3-ones as antiplasmodial falcipain-2 inhibitors
N Micale, R Ettari, T Schirmeister, A Evers, C Gelhaus, M Leippe, ...
Bioorganic & medicinal chemistry 17 (18), 6505-6511, 2009
432009
Development of peptidomimetic boronates as proteasome inhibitors
N Micale, R Ettari, A Lavecchia, C Di Giovanni, K Scarbaci, V Troiano, ...
European journal of medicinal chemistry 64, 23-34, 2013
422013
Formaldehyde exposure and acute myeloid leukemia: a review of the literature
A Allegra, G Spatari, S Mattioli, S Curti, V Innao, R Ettari, AG Allegra, ...
Medicina 55 (10), 638, 2019
412019
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