Treatment-induced tumor dormancy through YAP-mediated transcriptional reprogramming of the apoptotic pathway KJ Kurppa, Y Liu, C To, T Zhang, M Fan, A Vajdi, EH Knelson, Y Xie, ... Cancer cell 37 (1), 104-122. e12, 2020 | 385 | 2020 |
CuI/oxalic diamide catalyzed coupling reaction of (hetero) aryl chlorides and amines W Zhou, M Fan, J Yin, Y Jiang, D Ma Journal of the American Chemical Society 137 (37), 11942-11945, 2015 | 233 | 2015 |
Palladium-catalyzed direct functionalization of 2-aminobutanoic acid derivatives: application of a convenient and versatile auxiliary. M Fan, D Ma Angewandte Chemie International Edition 52 (46), 2013 | 180 | 2013 |
Assembly of primary (hetero) arylamines via CuI/oxalic diamide-catalyzed coupling of aryl chlorides and ammonia M Fan, W Zhou, Y Jiang, D Ma Organic letters 17 (23), 5934-5937, 2015 | 143 | 2015 |
CuI/Oxalamide catalyzed couplings of (Hetero) aryl chlorides and phenols for diaryl ether formation M Fan, W Zhou, Y Jiang, D Ma Angewandte Chemie International Edition 55 (21), 6211-6215, 2016 | 133 | 2016 |
Copper-catalyzed diaryl ether formation from (hetero) aryl halides at low catalytic loadings Y Zhai, X Chen, W Zhou, M Fan, Y Lai, D Ma The Journal of Organic Chemistry 82 (9), 4964-4969, 2017 | 60 | 2017 |
Assembly of Indoline-2-carboxylate-Embodied Dipeptides via Pd-Catalyzed C(sp2)–H Bond Direct Functionalization YP He, C Zhang, M Fan, Z Wu, D Ma Organic letters 17 (3), 496-499, 2015 | 57 | 2015 |
Covalent disruptor of YAP-TEAD association suppresses defective Hippo signaling M Fan, W Lu, J Che, NP Kwiatkowski, Y Gao, HS Seo, SB Ficarro, ... Elife 11, e78810, 2022 | 45 | 2022 |
Total Synthesis of Lapidilectine B Enabled by Manganese (III)‐Mediated Oxidative Cyclization of Indoles Y Gao, M Fan, Q Geng, D Ma Chemistry–A European Journal 24 (25), 6547-6550, 2018 | 29 | 2018 |
Depletion of creatine phosphagen energetics with a covalent creatine kinase inhibitor N Darabedian, W Ji, M Fan, S Lin, HS Seo, EV Vinogradova, TM Yaron, ... Nature chemical biology 19 (7), 815-824, 2023 | 28 | 2023 |
Structure-based design of Y-shaped covalent TEAD inhibitors W Lu, M Fan, W Ji, J Tse, I You, SB Ficarro, I Tavares, J Che, AY Kim, ... Journal of medicinal chemistry 66 (7), 4617-4632, 2023 | 14 | 2023 |
Spatiotemporal quantification of HER2-targeting antibody–drug conjugate bystander activity and enhancement of solid tumor penetration Q Wei, T Yang, J Zhu, Z Zhang, L Yang, Y Zhang, C Hu, J Chen, J Wang, ... Clinical Cancer Research 30 (5), 984-997, 2024 | 9 | 2024 |
Amino pyrimidine compounds useful as SSAO inhibitors M Fan, L Qin, Y Wei, G Zhou, J Zhou US Patent 10,278,970, 2019 | 6 | 2019 |
Discovery and optimization of thieno [3, 2-d] pyrimidine derivatives as highly selective inhibitors of cyclin-dependent kinase 7 H Zhang, G Lin, S Jia, Y Zhang, J Wu, Y Tao, W Huang, M Song, K Ding, ... European Journal of Medicinal Chemistry 263, 115955, 2024 | 4 | 2024 |
Transcriptional enhanced associate doman (tead) transcription factor inhibitors and uses thereof NS Gray, T Zhang, J Che, NP Kwiatkowski, FAN Mengyang, W Lu | 3 | 2021 |
Design, synthesis and evaluation of thieno [3, 2-d] pyrimidine derivatives as novel potent CDK7 inhibitors H Zhang, G Lin, S Jia, J Wu, Y Zhang, Y Tao, W Huang, M Song, K Ding, ... Bioorganic Chemistry 148, 107456, 2024 | 2 | 2024 |
Discovery of novel macrocyclic derivatives as potent and selective cyclin-dependent kinase 2 inhibitors P Niu, Y Tao, Q Meng, Y Huang, S Li, K Ding, D Ma, Z Ye, M Fan Bioorganic & Medicinal Chemistry 104, 117711, 2024 | 2 | 2024 |
Discovery and optimization of (2-naphthylthio) acetic acid derivative as selective Bfl-1 inhibitor P Niu, H Xu, M Fan Bioorganic & Medicinal Chemistry Letters 101, 129658, 2024 | 2 | 2024 |
Amino pyrimidine compounds useful as SSAO inhibitors M Fan, L Qin, Y Wei, G Zhou, J Zhou US Patent 10,471,060, 2019 | 2 | 2019 |
Transcriptional enhanced associated domain (tead) transcription factor inhibitors and uses thereof NS Gray, T Zhang, M Fan, J Che, W Lu, S Dhe-Paganon, NP Kwiatkowski US Patent App. 18/553,988, 2024 | 1 | 2024 |