Congo red protects against toxicity of β-amyloid peptides on rat hippocampal neurones MC Burgevin, M Passat, N Daniel, M Capet, A Doble Neuroreport 5 (18), 2429-2432, 1994 | 70 | 1994 |
Histamine and tele-methylhistamine quantification in cerebrospinal fluid from narcoleptic subjects by liquid chromatography tandem mass spectrometry with precolumn derivatization M Croyal, Y Dauvilliers, O Labeeuw, M Capet, JC Schwartz, P Robert Analytical biochemistry 409 (1), 28-36, 2011 | 51 | 2011 |
Azetidine derivatives, their preparation and medicaments containing them D Achard, H Bouchard, J Bouquerel, M Capet, S Grisoni, JL Malleron, ... US Patent 6,518,264, 2003 | 49 | 2003 |
Refined Docking as a Valuable Tool for Lead Optimization: Application to Histamine H3 Receptor Antagonists N Levoin, T Calmels, O Poupardin‐Olivier, O Labeeuw, D Danvy, ... Archiv der Pharmazie 341 (10), 610-623, 2008 | 44 | 2008 |
Farnesyl transferase inhibitors, their preparation, the pharmaceutical compositions which contain them and their use in the preparation of medicaments JD Bourzat, A Commerçon, N Dereu, P Mailliet, F Sounigo-Thompson, ... US Patent 6,013,662, 2000 | 41 | 2000 |
Pharmacological properties of ureido-acetamides, new potent and selective non-peptide CCKB/gastrin receptor antagonists P Bertrand, GA Böhme, C Durieux, C Guyon, M Capet, B Jeantaud, ... European journal of pharmacology 262 (3), 233-245, 1994 | 39 | 1994 |
Fluorinated non-imidazole histamine H3 receptor antagonists K Isensee, M Amon, A Galaparti, X Ligneau, JC Camelin, M Capet, ... Bioorganic & medicinal chemistry letters 19 (8), 2172-2175, 2009 | 35 | 2009 |
Unexpected formation of aryl ketones by palladium-catalyzed coupling of aryl bromides with vinylic acetates M Jean, J Renault, P Uriac, M Capet, P van de Weghe Organic Letters 9 (18), 3623-3625, 2007 | 35 | 2007 |
6, 11-dihydro-5H-benzo [d] imidazo [1, 2-a] azepines derivatives as histamine H4 receptor ligands I Berrebi-Bertrand, X Billot, T Calmels, M Capet, S Krief, O Labeeuw, ... US Patent 9,255,101, 2016 | 31 | 2016 |
Interaction of brain cannabinoid receptors with guanine nucleotide binding protein: A radioligand binding study F Petitet, B Jeantaud, M Capet, A Doble Biochemical pharmacology 54 (11), 1267-1270, 1997 | 29 | 1997 |
Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity N Levoin, O Labeeuw, T Calmels, O Poupardin-Olivier, I Berrebi-Bertrand, ... Bioorganic & medicinal chemistry letters 21 (18), 5378-5383, 2011 | 24 | 2011 |
Parallel synthesis and dopamine D3/D2 receptor screening of novel {4-[4-(2-methoxyphenyl) piperazin-1-yl] butyl} carboxamides P Heidler, V Zohrabi-Kalantari, T Calmels, M Capet, I Berrebi-Bertrand, ... Bioorganic & medicinal chemistry 13 (6), 2009-2014, 2005 | 23 | 2005 |
Homology model versus X-ray structure in receptor-based drug design: A retrospective analysis with the dopamine D3 receptor N Levoin, T Calmels, S Krief, D Danvy, I Berrebi-Bertrand, JM Lecomte, ... ACS Medicinal Chemistry Letters 2 (4), 293-297, 2011 | 22 | 2011 |
Exploring occupancy of the histamine H3 receptor by pitolisant in humans using PET P Rusjan, P Sabioni, P Di Ciano, E Mansouri, I Boileau, A Laveillé, ... British journal of pharmacology 177 (15), 3464-3472, 2020 | 21 | 2020 |
Pyrrole derivatives, and pharmaceutical compositions which contain them and pharmacological methods of use JD Bourzat, M Capet, C Cotrel, R Labaudiniere, P Pitchen, G Roussel US Patent 4,960,779, 1990 | 20 | 1990 |
Determination of the binding mode and interacting amino-acids for dibasic H3 receptor antagonists N Levoin, O Labeeuw, S Krief, T Calmels, O Poupardin-Olivier, ... Bioorganic & medicinal chemistry 21 (15), 4526-4529, 2013 | 19 | 2013 |
Pyrrolidine and thiazolidine derivatives, their preparation and medicaments containing them M Capet, C Cotrel, C Guyon, M Joannic, F Manfre, G erard Roussel, ... US Patent 5,610,144, 1997 | 16 | 1997 |
N-phenylglycinamide CCK antagonists and pharmaceutical compositions containing them JD Bourzat, M Capet, C Cotrel, C Guyon, F Manfre, G Roussel US Patent 5,475,106, 1995 | 16 | 1995 |
Arylvinylazacycloalkane compounds and methods of preparation and use thereof JD Schmitt, GM Dull, CH Miller, A Genevois-Borella, M Capet, M Cheve US Patent 8,063,068, 2011 | 15* | 2011 |
3-Ureidobenzodiazepinones useful as antagonists of CCK or of gastrin M Capet, C Cotrel, MC Dubroeuco, C Guyon, JP Martin US Patent 5,563,136, 1996 | 15 | 1996 |