Structure− activity relationships of selective estrogen receptor modulators: modifications to the 2-arylbenzothiophene core of raloxifene TA Grese, S Cho, DR Finley, AG Godfrey, CD Jones, CW Lugar, MJ Martin, ... Journal of medicinal chemistry 40 (2), 146-167, 1997 | 230 | 1997 |
A remote-controlled adaptive medchem lab: an innovative approach to enable drug discovery in the 21st Century AG Godfrey, T Masquelin, H Hemmerle Drug Discovery Today 18 (17-18), 795-802, 2013 | 146 | 2013 |
Application of the dakin− west reaction for the synthesis of oxazole-containing dual PPARα/γ agonists AG Godfrey, DA Brooks, LA Hay, M Peters, JR McCarthy, D Mitchell The Journal of Organic Chemistry 68 (7), 2623-2632, 2003 | 126 | 2003 |
Ready oxidation of halides to aldehydes using trimethylamine N-oxide in dimethylsulfoxide AG Godfrey, B Ganem Tetrahedron letters 31 (34), 4825-4826, 1990 | 111 | 1990 |
Reductive deoxygenation by Cp2ZrHCl: Selective formation of imines via zirconation/hydrozirconation of amides DJA Schedler, AG Godfrey, B Ganem Tetrahedron letters 34 (32), 5035-5038, 1993 | 92 | 1993 |
Synergistic methodologies for the synthesis of 3-aroyl-2-arylbenzo[b]thiophene-based selective estrogen receptor modulators. Two concise syntheses of raloxifene DA Bradley, AG Godfrey, CR Schmid Tetrahedron letters 40 (28), 5155-5159, 1999 | 46 | 1999 |
Reductive deoxygenation using hydridozirconium enolates: A new synthesis of α, β-unsaturated esters AG Godfrey, B Ganem Tetrahedron letters 33 (49), 7461-7464, 1992 | 35 | 1992 |
Pyrrole derivatives as pharmaceutical agents DW Beight, TV DeCollo, AG Godfrey, T Goodson Jr, HY Li, WT McMillen, ... US Patent 7,087,626, 2006 | 33 | 2006 |
Imidazo[1,2-a]Pyridine-3-Carboxamides Are Active Antimicrobial Agents against Mycobacterium avium Infection In Vivo GC Moraski, Y Cheng, S Cho, JW Cramer, A Godfrey, T Masquelin, ... Antimicrobial agents and chemotherapy 60 (8), 5018-5022, 2016 | 30 | 2016 |
Oxazolyl-aryloxyacetic acid derivatives and their use as ppar agonists DA Brooks, SE Conner, SJ Dominianni, AG Godfrey, LS Gossett, CJ Rit, ... US Patent 6,982,278, 2006 | 24 | 2006 |
2-amino-3-aroyl-benzo [β] thiophenes and methods for preparing and using same to produce 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)-benzoyl] benzo [β] thiophenes AG Godfrey US Patent 5,466,810, 1995 | 24 | 1995 |
Oxazolyl-aryloxyacetic acid derivatives and their use as PPAR agonists DA Brooks, SE Conner, SJ Dominianni, AG Godfrey, LS Gossett, CJ Rito, ... US Patent 7,351,728, 2008 | 22 | 2008 |
New syntheses of alkenes and alkynes from amines AG Godfrey, B Ganem Journal of the American Chemical Society 112 (9), 3717-3718, 1990 | 17 | 1990 |
Discovery of selective RIO2 kinase small molecule ligand T Varin, AG Godfrey, T Masquelin, CA Nicolaou, DA Evans, M Vieth Biochimica et Biophysica Acta (BBA)-Proteins and Proteomics 1854 (10), 1630-1636, 2015 | 15 | 2015 |
A perspective on innovating the chemistry lab bench AG Godfrey, SG Michael, GS Sittampalam, G Zahoránszky-Köhalmi Frontiers in Robotics and AI 7, 24, 2020 | 13 | 2020 |
New chemistry of diazoesters from thermal rearrangement of n-alkyl-n-nitrosoamides N Nikolaides, AG Godfrey, B Ganem Tetrahedron letters 31 (42), 6009-6012, 1990 | 12 | 1990 |
Arylpiperazines having activity at the serotonin 1A receptor AG Godfrey, DT Kohlman, JC O'toole, YC Xu, TY Zhang US Patent 7,001,908, 2006 | 9 | 2006 |
Compounds as pharmaceutical agents DW Beight, TP Burkholder, TV Decollo, AG Godfrey, CR Heap, CHR King, ... US Patent 7,405,299, 2008 | 7 | 2008 |
Lithiated benzothiophenes and benzofurans require 2-silyl protection to avoid anion migration MM Hansen, MT Clayton, AG Godfrey, JL Grutsch Jr, SS Keast, ... Synlett 2004 (08), 1351-1354, 2004 | 7 | 2004 |
Oxazolyl-arylproplonic acid derivatives and their use as ppar agonists DA Brooks, AG Godfrey, SB Jones, JR McCarthy, CJ Rito, LL Winneroski, ... US Patent 6,930,120, 2005 | 6 | 2005 |