Anti-Giardia Drug Discovery: Current Status and Gut Feelings A Riches, CJS Hart, KR Trenholme, TS Skinner-Adams Journal of medicinal chemistry 63 (22), 13330-13354, 2020 | 61 | 2020 |
Synthesis of stentorin DW Cameron, AG Riches Tetrahedron letters 36 (13), 2331-2334, 1995 | 41 | 1995 |
A novel in vitro image-based assay identifies new drug leads for giardiasis CJS Hart, T Munro, KT Andrews, JH Ryan, AG Riches, TS Skinner-Adams International Journal for Parasitology: Drugs and Drug Resistance 7 (1), 83-89, 2017 | 33 | 2017 |
Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone TS Skinner-Adams, GM Fisher, AG Riches, OE Hutt, KE Jarvis, T Wilson, ... Communications biology 2 (1), 166, 2019 | 28 | 2019 |
Synthesis of Functionalized Chiral (Racemic) Cyclobutanones AG Riches, LA Wernersbach, LS Hegedus The Journal of Organic Chemistry 63 (14), 4691-4696, 1998 | 25 | 1998 |
Taxane Diterpene Synthesis Studies. Part 2: Towards Taxinine—Enantiospecific Construction of an AB-ring Substructure Incorporating both Quaternary Carbon Centres and Attempts … MG Banwell, MD McLeod, AG Riches Australian journal of chemistry 57 (1), 53-66, 2004 | 17 | 2004 |
Stereoselective reductions of N-Boc-hexahydro-1H-indolin-5 (6H)-ones MA Brodney, ML Cole, JA Freemont, S Kyi, PC Junk, A Padwa, AG Riches, ... Tetrahedron letters 48 (11), 1939-1943, 2007 | 14 | 2007 |
De Novo Synthesis of 4 ‘-Ethoxy Nucleoside Analogues LS Hegedus, L Geisler, AG Riches, SS Salman, G Umbricht The Journal of Organic Chemistry 67 (22), 7649-7655, 2002 | 13 | 2002 |
Scalable synthesis of an integrin-binding peptide mimetic for biomedical applications AG Riches, T Cablewski, V Glattauer, H Thissen, L Meagher Tetrahedron 68 (46), 9448-9455, 2012 | 11 | 2012 |
Control of parasites in animals by N-[(phenyloxy) phenyl]-1, 1, 1-trifluoromethanesulfonamide and N-[(phenylsulfanyl) phenyl]-1, 1, 1-trifluoromethanesulfonamide derivatives A Meyer, K Winzenberg, D Sawutz, A Riches US Patent App. 11/448,421, 2006 | 9 | 2006 |
An image-based Pathogen Box screen identifies new compounds with anti-Giardia activity and highlights the importance of assay choice in phenotypic drug discovery S Tiash, J Saunders, CJS Hart, JH Ryan, AG Riches, TS Skinner-Adams International Journal for Parasitology: Drugs and Drug Resistance 12, 60-67, 2020 | 8 | 2020 |
Discovery of ectoparasiticidal hydrazonotrifluoromethanesulfonanilides A Ali, P Fisara, JA Freemont, S Kyi, AG Meyer, AG Riches, RM Sargent, ... Bioorganic & medicinal chemistry letters 20 (2), 649-652, 2010 | 8 | 2010 |
Reaction of 2-acetoxy-3-chloro and 2, 3-diacetoxy naphthoquinones with 1, 3-dioxy and 1, 1, 3-trioxy butadienes DW Cameron, AG Riches Australian Journal of Chemistry 52 (12), 1165-1171, 1999 | 8 | 1999 |
Immobilisation of a thrombopoietin peptidic mimic by self-assembled monolayers for culture of CD34+ cells EJ Lee, CL Be, AR Vinson, AG Riches, F Fehr, J Gardiner, ... Biomaterials 37, 82-93, 2015 | 7 | 2015 |
N-Phenyl-1, 1, 1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites K Winzenberg, A Meyer, Q Yang, A Riches US Patent App. 11/695,226, 2007 | 6 | 2007 |
Synthesis of 2, 3-Dioxy-1, 4-anthraquinones Related to Tetracenomycins C and X DW Cameron, PG Griffiths, AG Riches Australian Journal of Chemistry 52 (12), 1173-1177, 1999 | 6 | 1999 |
Thieno [3, 2-b] pyrrole 5-carboxamides as potent and selective inhibitors of Giardia duodenalis CJS Hart, AG Riches, S Tiash, R Abraham, K Fayd’Herbe, E Joch, ... International Journal for Parasitology: Drugs and Drug Resistance 23, 54-62, 2023 | 4 | 2023 |
Zinc is not required for activity of TPO agonists acting at the c-Mpl receptor transmembrane domain J Andrade, T Cablewski, G Condie, D Haylock, L Meagher, A Riches, ... ACS Chemical Biology 5 (8), 741-745, 2010 | 4 | 2010 |
Structural reassignment of a dibenz [b, f][1, 4] oxazepin-11 (10H)-one with potent antigiardial activity AG Riches, CJS Hart, M Schmit, EA Debele, S Tiash, E Clapper, ... Australian Journal of Chemistry 75 (10), 839-845, 2022 | 3 | 2022 |
Potent and selective Anti-gardia compound seies: progress and new developments TS Skinner-Adams, CJ Hart, A Riches, J Ryan, S Abraham, R Abraham The American Journal of Tropical Medicine and Hygiene 99 (4 Supp. 1), 655-656, 2018 | 3 | 2018 |