Artemisinin bioactivity and resistance in malaria parasites AM Talman, J Clain, R Duval, R Ménard, F Ariey Trends in parasitology 35 (12), 953-963, 2019 | 115 | 2019 |
Fluorescent natural products as probes and tracers in biology R Duval, C Duplais Natural product reports 34 (2), 161-193, 2017 | 106 | 2017 |
Rapid discovery of triazolobenzylidene-thiazolopyrimidines (TBTP) as CDC25 phosphatase inhibitors by parallel click chemistry and in situ screening R Duval, S Kolb, E Braud, D Genest, C Garbay Journal of Combinatorial Chemistry 11 (6), 947-950, 2009 | 77 | 2009 |
Chamuvarinin, an Acetogenin Bearing a Tetrahydropyran Ring from the Roots of Uvaria chamae D Fall, RA Duval, C Gleye, A Laurens, R Hocquemiller Journal of natural products 67 (6), 1041-1043, 2004 | 52 | 2004 |
Heterocyclic analogues of squamocin as inhibitors of mitochondrial complex I. On the role of the terminal lactone of annonaceous acetogenins RA Duval, G Lewin, E Peris, N Chahboune, A Garofano, S Dröse, ... Biochemistry 45 (8), 2721-2728, 2006 | 46 | 2006 |
Cancer Chemotherapy: A Paclitaxel Prodrug for ADEPT (Antibody‐Directed Enzyme Prodrug Therapy) F Schmidt, I Ungureanu, R Duval, A Pompon, C Monneret European Journal of Organic Chemistry 2001 (11), 2129-2134, 2001 | 44 | 2001 |
Localization of cocaine analog [125I] RTI 82 irreversible binding to transmembrane domain 6 of the dopamine transporter RA Vaughan, DS Sakrikar, ML Parnas, S Adkins, JD Foster, RA Duval, ... Journal of Biological Chemistry 282 (12), 8915-8925, 2007 | 40 | 2007 |
Indium-labeled macrocyclic conjugates of naltrindole: high-affinity radioligands for in vivo studies of peripheral δ opioid receptors RA Duval, RL Allmon, JR Lever Journal of medicinal chemistry 50 (9), 2144-2156, 2007 | 31 | 2007 |
Plasmodium falciparum sexual parasites regulate infected erythrocyte permeability G Bouyer, D Barbieri, F Dupuy, A Marteau, A Sissoko, ME N’dri, G Neveu, ... Communications Biology 3 (1), 726, 2020 | 26 | 2020 |
Radioiodinated azide and isothiocyanate derivatives of cocaine for irreversible labeling of dopamine transporters: synthesis and covalent binding studies JR Lever, MF Zou, ML Parnas, RA Duval, SE Wirtz, JB Justice, ... Bioconjugate chemistry 16 (3), 644-649, 2005 | 24 | 2005 |
Analogues of cytotoxic squamocin using reliable reactions: new insights into the reactivity and role of the α, β-unsaturated lactone of the annonaceous acetogenins RA Duval, E Poupon, V Romero, E Peris, G Lewin, D Cortes, U Brandt, ... Tetrahedron 62 (26), 6248-6257, 2006 | 23 | 2006 |
Semisynthesis of heterocyclic analogues of squamocin, a cytotoxic annonaceous acetogenin, by an unusual oxidative decarboxylation reaction R Duval, G Lewin, R Hocquemiller Bioorganic & medicinal chemistry 11 (16), 3439-3446, 2003 | 21 | 2003 |
Semisynthesis and biological activity of aminoacyl triesters of squamocin, an annonaceous acetogenin RA Duval, P Duret, G Lewin, E Peris, R Hocquemiller Bioorganic & medicinal chemistry 13 (11), 3773-3781, 2005 | 18 | 2005 |
Semisynthesis and Screening of a Small Library of Pro‐Apoptotic Squamocin Analogues: Selection and Study of a Benzoquinone Hybrid with an Improved Biological Profile. S Derbré, R Duval, G Roué, A Garofano, E Poupon, U Brandt, SA Susin, ... ChemMedChem: Chemistry Enabling Drug Discovery 1 (1), 118-129, 2006 | 17 | 2006 |
Remarkable substituent effect: β-aminosquamocin, a potent dual inhibitor of mitochondrial complexes I and III RA Duval, E Poupon, U Brandt, R Hocquemiller Biochimica et Biophysica Acta (BBA)-Bioenergetics 1709 (3), 191-194, 2005 | 17 | 2005 |
Artemisinin-independent inhibitory activity of Artemisia sp. infusions against different Plasmodium stages including relapse-causing hypnozoites K Ashraf, S Tajeri, CS Arnold, N Amanzougaghene, JF Franetich, ... Life Science Alliance 5 (3), 2022 | 15 | 2022 |
A chemically stable fluorescent mimic of dihydroartemisinin, artemether, and arteether with conserved bioactivity and specificity shows high pharmacological relevance to the … A Sissoko, P Vásquez-Ocmín, A Maciuk, D Barbieri, G Neveu, ... ACS Infectious Diseases 6 (7), 1532-1547, 2020 | 14 | 2020 |
Artemisinin and its derivatives target mitochondrial c-type cytochromes in yeast and human cells A Laleve, C Panozzo, I Kühl, A Bourand-Plantefol, J Ostojic, A Sissoko, ... Biochimica et Biophysica Acta (BBA)-Molecular Cell Research 1867 (5), 118661, 2020 | 13 | 2020 |
Fischer indole synthesis in water: simple, efficient preparation of naltrindole, naltriben and analogs RA Duval, JR Lever Green Chemistry 12 (2), 304-309, 2010 | 13 | 2010 |
Ultraspecific live imaging of the dynamics of zebrafish neutrophil granules by a histopermeable fluorogenic benzochalcone probe E Colucci-Guyon, AS Batista, SDS Oliveira, M Blaud, IC Bellettini, ... Chemical Science 10 (12), 3654-3670, 2019 | 12 | 2019 |