Novel 4-(piperazin-1-yl) quinolin-2 (1H)-one bearing thiazoles with antiproliferative activity through VEGFR-2-TK inhibition A Hassan, M Badr, HA Hassan, D Abdelhamid, GEDA Abuo‐Rahma Bioorganic & Medicinal Chemistry 40, 116168, 2021 | 29 | 2021 |
Design, synthesis, anticonvulsant activity, and pharmacophore study of new 1,5-diaryl-1H-1,2,4-triazole-3-carboxamide derivatives AH Abuelhassan, MM Badran, HA Hassan, D Abdelhamed, S Elnabtity, ... Medicinal Chemistry Research 27, 928-938, 2018 | 22 | 2018 |
Design and biological evaluation of 3-substituted quinazoline-2,4(1H,3H)-dione derivatives as dual c-Met/VEGFR-2-TK inhibitors A Hassan, FAF Mubarak, IA Shehadi, AM Mosallam, H Temairk, M Badr, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2189578, 2023 | 20 | 2023 |
Novel 3-phenylquinazolin-2,4(1H,3H)-diones as dual VEGFR-2/c-Met-TK inhibitors: design, synthesis, and biological evaluation A Hassan, AM Mosallam, AOA Ibrahim, M Badr, AH Abdelmonsef Scientific Reports 13 (1), 18567, 2023 | 16 | 2023 |
Design, synthesis, in vitro antiproliferative evaluation and in silico studies of new VEGFR-2 inhibitors based on 4-piperazinylquinolin-2 (1H)-one scaffold A Hassan, M Badr, D Abdelhamid, HA Hassan, MAS Abourehab, ... Bioorganic Chemistry 120, 105631, 2022 | 15 | 2022 |
New quinazolin-2, 4-dione derivatives incorporating acylthiourea, pyrazole and/or oxazole moieties as antibacterial agents via DNA gyrase inhibition AOA Ibrahim, A Hassan, AM Mosallam, A Khodairy, HRM Rashdan, ... RSC advances 14 (24), 17158-17169, 2024 | 11 | 2024 |
SYNTHETIC APPROACHES TOWARD CERTAIN STRUCTURALLY RELATED ANTIMICROBIAL THIAZOLE DERIVATIVES (2010-2020) A Hassan, HA Hassan, D Abdelhamid, GEDA Abuo-Rahma Heterocycles: an international journal for reviews and communications in …, 2021 | 5 | 2021 |
Synthesis of new thiazole-privileged chalcones as tubulin polymerization inhibitors with potential anticancer activities H Hashem, A Hassan, WM Abdelmagid, AGK Habib, MAA Abdel-Aal, ... Pharmaceuticals 17 (9), 1154, 2024 | 3 | 2024 |
New 1, 3-diphenyl-1H-pyrazol-5-ols as anti-methicillin resistant Staphylococcus aureus agents: Synthesis, antimicrobial evaluation and in silico studies MAMA Reheim, ISA Hafiz, HM Reffat, HSA Rady, IA Shehadi, ... Heliyon 10 (13), 2024 | 2 | 2024 |
New S-and N-alkyl functionalized bis-1, 2, 4-Triazolyl-based derivatives as potential dual EGFRWT and EGFRT790M inhibitors: Synthesis, anti-proliferative evaluation, molecular … AM Ahmed, MO Aboelez, HAA Ezelarab, A Khodairy, A Hassan, MA User, ... Journal of Molecular Structure 1324, 140720, 2025 | | 2025 |
Design, synthesis in vitro and in vivo evaluation of new diaryltriazoles carboxylic and hydroxamic acid derivatives as inhibitors of tumor necrosis alpha converting enzyme (TACE) A Hassan, MM Badran, HA Hassan, D Abdelhamid, O Aly Octahedron Drug Research 2 (1), 44-62, 2023 | | 2023 |