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Agostino Cilibrizzi
Agostino Cilibrizzi
在 kcl.ac.uk 的电子邮件经过验证 - 首页
标题
引用次数
引用次数
年份
Diversity-oriented synthesis of macrocyclic peptidomimetics
A Isidro-Llobet, T Murillo, P Bello, A Cilibrizzi, JT Hodgkinson, ...
Proceedings of the National Academy of Sciences 108 (17), 6793-6798, 2011
1312011
Hydroxypyridinone journey into metal chelation
A Cilibrizzi, V Abbate, YL Chen, Y Ma, T Zhou, RC Hider
Chemical reviews 118 (16), 7657-7701, 2018
752018
6-Methyl-2,4-Disubstituted Pyridazin-3(2H)-ones: A Novel Class of Small-Molecule Agonists for Formyl Peptide Receptors
A Cilibrizzi, MT Quinn, LN Kirpotina, IA Schepetkin, J Holderness, RD Ye, ...
Journal of medicinal chemistry 52 (16), 5044-5057, 2009
622009
An overview of PDE4 inhibitors in clinical trials: 2010 to early 2022
L Crocetti, G Floresta, A Cilibrizzi, MP Giovannoni
Molecules 27 (15), 4964, 2022
612022
Optimization of N-Benzoylindazole Derivatives as Inhibitors of Human Neutrophil Elastase
L Crocetti, IA Schepetkin, A Cilibrizzi, A Graziano, C Vergelli, D Giomi, ...
Journal of medicinal chemistry 56 (15), 6259-6272, 2013
612013
Development of small molecule non-peptide formyl peptide receptor (FPR) ligands and molecular modeling of their recognition
IA Schepetkin, AI Khlebnikov, MP Giovannoni, LN Kirpotina, A Cilibrizzi, ...
Current medicinal chemistry 21 (13), 1478-1504, 2014
592014
Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain
C Biancalani, MP Giovannoni, S Pieretti, N Cesari, A Graziano, C Vergelli, ...
Journal of medicinal chemistry 52 (23), 7397-7409, 2009
512009
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase
L Crocetti, MP Giovannoni, IA Schepetkin, MT Quinn, AI Khlebnikov, ...
Bioorganic & medicinal chemistry 19 (15), 4460-4472, 2011
462011
Cinnoline derivatives as human neutrophil elastase inhibitors
MP Giovannoni, IA Schepetkin, L Crocetti, G Ciciani, A Cilibrizzi, ...
Journal of enzyme inhibition and medicinal chemistry 31 (4), 628-639, 2016
442016
Further studies on 2-arylacetamide pyridazin-3 (2H)-ones: Design, synthesis and evaluation of 4, 6-disubstituted analogs as formyl peptide receptors (FPRs) agonists
MP Giovannoni, IA Schepetkin, A Cilibrizzi, L Crocetti, AI Khlebnikov, ...
European journal of medicinal chemistry 64, 512-528, 2013
402013
3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation
G Floresta, A Cilibrizzi, V Abbate, A Spampinato, C Zagni, A Rescifina
Bioorganic Chemistry 84, 276-284, 2019
332019
Analytical characterization of three cathinone derivatives, 4‐MPD, 4F–PHP and bk‐EPDP, purchased as bulk powder from online vendors
O Apirakkan, A Frinculescu, T Shine, MC Parkin, A Cilibrizzi, N Frascione, ...
Drug Testing and Analysis 10 (2), 372-378, 2018
322018
Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists
A Cilibrizzi, IA Schepetkin, G Bartolucci, L Crocetti, V Dal Piaz, ...
Bioorganic & medicinal chemistry 20 (12), 3781-3792, 2012
292012
Functionalized pyrazoles and pyrazolo [3, 4-d] pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity
P Biagini, C Biancalani, A Graziano, N Cesari, MP Giovannoni, A Cilibrizzi, ...
Bioorganic & Medicinal Chemistry 18 (10), 3506-3517, 2010
272010
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists
C Vergelli, IA Schepetkin, G Ciciani, A Cilibrizzi, L Crocetti, ...
Bioorganic & medicinal chemistry 24 (11), 2530-2543, 2016
262016
Synthesis and pharmacological evaluation of new pyridazin‐based thioderivatives as formyl peptide receptor (FPR) agonists
L Crocetti, C Vergelli, A Cilibrizzi, A Graziano, AI Khlebnikov, LN Kirpotina, ...
Drug Development Research 74 (4), 259-271, 2013
242013
A case of extensive protein platination: The reaction of lysozyme with a Pt (II)–terpyridine complex
G Ferraro, T Marzo, T Infrasca, A Cilibrizzi, R Vilar, L Messori, A Merlino
Dalton Transactions 47 (26), 8716-8723, 2018
232018
Further studies on pyrazolo [1′, 5′: 1, 6] pyrimido [4, 5-d] pyridazin-4 (3H)-ones as potent and selective human A1 adenosine receptor antagonists
MP Giovannoni, G Ciciani, A Cilibrizzi, L Crocetti, S Daniele, ...
European Journal of Medicinal Chemistry 89, 32-41, 2015
222015
FABP4 inhibitors 3D-QSAR model and isosteric replacement of BMS309403 datasets
G Floresta, A Cilibrizzi, V Abbate, A Spampinato, C Zagni, A Rescifina
Data in brief 22, 471-483, 2019
212019
The role of mitochondrial labile iron in Friedreich's ataxia skin fibroblasts sensitivity to ultraviolet A
O Reelfs, V Abbate, A Cilibrizzi, MA Pook, RC Hider, C Pourzand
Metallomics 11 (3), 656-665, 2019
202019
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