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Abdelfattah Faouzi
Abdelfattah Faouzi
Scientist, Exploratory Chemistry
在 ucsd.edu 的电子邮件经过验证
标题
引用次数
引用次数
年份
Biased opioid ligands
A Faouzi, BR Varga, S Majumdar
Molecules 25 (18), 4257, 2020
962020
Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site
R Uprety, T Che, SA Zaidi, SG Grinnell, BR Varga, A Faouzi, ST Slocum, ...
Elife 10, e56519, 2021
492021
Structure-based design of bitopic ligands for the µ-opioid receptor
A Faouzi, H Wang, SA Zaidi, JF DiBerto, T Che, Q Qu, MJ Robertson, ...
Nature 613 (7945), 767-774, 2023
422023
A novel mitragynine analog with low-efficacy mu opioid receptor agonism displays antinociception with attenuated adverse effects
S Chakraborty, JF DiBerto, A Faouzi, SM Bernhard, AM Gutridge, ...
Journal of medicinal chemistry 64 (18), 13873-13892, 2021
412021
Site selective C–H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy
S Bhowmik, J Galeta, V Havel, M Nelson, A Faouzi, B Bechand, ...
Nature communications 12 (1), 3858, 2021
282021
Synthesis and biological evaluation of thiophene and benzo [b] thiophene analogs of combretastatin A-4 and isocombretastatin A-4: A comparison between the linkage positions of …
CV Do, A Faouzi, C Barette, A Farce, MO Fauvarque, E Colomb, L Catry, ...
Bioorganic & medicinal chemistry letters 26 (1), 174-180, 2016
262016
Synthesis and pharmacology of a novel μ–δ opioid receptor heteromer-selective agonist based on the carfentanyl template
A Faouzi, R Uprety, I Gomes, N Massaly, AI Keresztes, V Le Rouzic, ...
Journal of medicinal chemistry 63 (22), 13618-13637, 2020
252020
Combretastatin A-4 sulfur-containing heterocyclic derivatives: Synthesis, antiproliferative activities and molecular docking studies
A Faouzi, A Arnaud, A Bancet, C Barette, J Preto, CV Do, LP Jordheim, ...
European Journal of Medicinal Chemistry 215, 113275, 2021
82021
Think big, start small: How nanomedicine could alleviate the burden of rare CNS diseases
A Faouzi, VG Roullin
Pharmaceuticals 14 (2), 109, 2021
42021
Design of first in class bitopic ligands targeting the sodium binding pocket in opioid receptors
A Faouzi, S Zaidi, T Che, C Kormos, T Zhang, M Madasu, S Eans, ...
The FASEB Journal 34 (S1), 1-1, 2020
22020
Syntheses and biological evaluations of combretastatine A-4 analogs and DYRK kinases inhibitors
A Faouzi
Université de Lyon, 2017
2017
Synthèses et évaluations biologiques d’analogues de la combrétastatine A-4 et d’inhibiteurs de kinases DYRK
A Faouzi
Université de Lyon, 2017
2017
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