Convenient Method To Access New 4,4-Dialkoxy- and 4,4-Diaryloxy-diaza-s-indacene Dyes: Synthesis and Spectroscopic Evaluation C Tahtaoui, C Thomas, F Rohmer, P Klotz, G Duportail, Y Mély, D Bonnet, ... The Journal of organic chemistry 72 (1), 269-272, 2007 | 222 | 2007 |
Identification and pharmacological properties of E339–3D6, the first nonpeptidic apelin receptor agonist X Iturrioz, R Alvear‐Perez, N De Mota, C Franchet, F Guillier, V Leroux, ... The FASEB Journal 24 (5), 1506-1517, 2010 | 130 | 2010 |
Proper desensitization of CXCR4 is required for lymphocyte development and peripheral compartmentalization in mice K Balabanian, E Brotin, V Biajoux, L Bouchet-Delbos, E Lainey, ... Blood, The Journal of the American Society of Hematology 119 (24), 5722-5730, 2012 | 128 | 2012 |
Small neutralizing molecules to inhibit actions of the chemokine CXCL12 M Hachet-Haas, K Balabanian, F Rohmer, F Pons, C Franchet, S Lecat, ... Journal of Biological Chemistry 283 (34), 23189-23199, 2008 | 126 | 2008 |
Fluorogenic squaraine dimers with polarity-sensitive folding as bright far-red probes for background-free bioimaging IA Karpenko, M Collot, L Richert, C Valencia, P Villa, Y Mély, M Hibert, ... Journal of the American Chemical Society 137 (1), 405-412, 2015 | 105 | 2015 |
Biased agonist pharmacochaperones of the AVP V2 receptor may treat congenital nephrogenic diabetes insipidus F Jean-Alphonse, S Perkovska, MC Frantz, T Durroux, C Méjean, D Morin, ... Journal of the American Society of Nephrology 20 (10), 2190-2203, 2009 | 104 | 2009 |
α5β1 integrin antagonists reduce chemotherapy‐induced premature senescence and facilitate apoptosis in human glioblastoma cells E Martinkova, A Maglott, DY Leger, D Bonnet, M Stiborova, K Takeda, ... International journal of cancer 127 (5), 1240-1248, 2010 | 89 | 2010 |
Push–pull dioxaborine as fluorescent molecular rotor: far-red fluorogenic probe for ligand–receptor interactions IA Karpenko, Y Niko, VP Yakubovskyi, AO Gerasov, D Bonnet, YP Kovtun, ... Journal of Materials Chemistry C 4 (14), 3002-3009, 2016 | 87 | 2016 |
Neutralization of CXCL12 attenuates established pulmonary hypertension in rats J Bordenave, R Thuillet, L Tu, C Phan, A Cumont, C Marsol, A Huertas, ... Cardiovascular research 116 (3), 686-697, 2020 | 70 | 2020 |
Development of original metabolically stable apelin‐17 analogs with diuretic and cardiovascular effects R Gerbier, R Alvear‐Perez, JF Margathe, A Flahault, P Couvineau, J Gao, ... The FASEB Journal 31 (2), 687-700, 2017 | 68 | 2017 |
Solid-Phase Synthesis of Tetrahydro-β-carbolinehydantoins via the N-Acyliminium Pictet−Spengler Reaction and Cyclative Cleavage D Bonnet, A Ganesan Journal of combinatorial chemistry 4 (6), 546-548, 2002 | 66 | 2002 |
Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays. S Loison, M Cottet, H Orcel, H Adihou, R Rahmeh, L Lamarque, ... Journal of medicinal chemistry 55 (20), 8588-8602, 2012 | 65 | 2012 |
Red fluorescent turn‐on ligands for imaging and quantifying G protein‐coupled receptors in living cells IA Karpenko, R Kreder, C Valencia, P Villa, C Mendre, B Mouillac, Y Mély, ... ChemBioChem 15 (3), 359-363, 2014 | 60 | 2014 |
Squaraine as a bright, stable and environment-sensitive far-red label for receptor-specific cellular imaging IA Karpenko, AS Klymchenko, S Gioria, R Kreder, I Shulov, P Villa, Y Mély, ... Chemical Communications 51 (14), 2960-2963, 2015 | 58 | 2015 |
Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer C Hounsou, JF Margathe, N Oueslati, A Belhocine, E Dupuis, C Thomas, ... ACS chemical biology 10 (2), 466-474, 2015 | 55 | 2015 |
A rapid and versatile method to label receptor ligands using “click” chemistry: Validation with the muscarinic M1 antagonist pirenzepine D Bonnet, B Ilien, JL Galzi, S Riché, C Antheaune, M Hibert Bioconjugate chemistry 17 (6), 1618-1623, 2006 | 54 | 2006 |
Structure–activity relationship studies toward the discovery of selective apelin receptor agonists JF Margathe, X Iturrioz, R Alvear-Perez, C Marsol, S Riché, H Chabane, ... Journal of medicinal chemistry 57 (7), 2908-2919, 2014 | 51 | 2014 |
An antedrug of the CXCL12 neutraligand blocks experimental allergic asthma without systemic effect in mice F Daubeuf, M Hachet-Haas, P Gizzi, V Gasparik, D Bonnet, V Utard, ... Journal of Biological Chemistry 288 (17), 11865-11876, 2013 | 49 | 2013 |
Chemoselective acylation of fully deprotected hydrazino acetyl peptides. Application to the synthesis of lipopeptides D Bonnet, N Ollivier, H Gras-Masse, O Melnyk The Journal of organic chemistry 66 (2), 443-449, 2001 | 47 | 2001 |
Involvement of the TGFβ pathway in the regulation of α5β1 integrins by caveolin‐1 in human glioblastoma EC Cosset, J Godet, N Entz‐Werlé, E Guérin, D Guenot, S Froelich, ... International journal of cancer 131 (3), 601-611, 2012 | 45 | 2012 |