Peptidomimetic toolbox for drug discovery E Lenci, A Trabocchi Chemical Society Reviews 49 (11), 3262-3277, 2020 | 249 | 2020 |
A new family of cinchona-derived amino phosphine precatalysts: application to the highly enantio-and diastereoselective silver-catalyzed isocyanoacetate aldol reaction F Sladojevich, A Trabocchi, A Guarna, DJ Dixon Journal of the American Chemical Society 133 (6), 1710-1713, 2011 | 240 | 2011 |
Suzuki Reaction of Vinyl Triflates from Six- and Seven-Membered N-Alkoxycarbonyl Lactams with Boronic Acids and Esters EG Occhiato, A Trabocchi, A Guarna The Journal of Organic Chemistry 66 (7), 2459-2465, 2001 | 114 | 2001 |
Structural diversity of bicyclic amino acids A Trabocchi, D Scarpi, A Guarna Amino acids 34, 1-24, 2008 | 103 | 2008 |
γ-and δ-amino acids: synthetic strategies and relevant applications A Trabocchi, F Guarna, A Guarna Current Organic Chemistry 9 (12), 1127-1153, 2005 | 95 | 2005 |
Peptidomimetics in Organic and Medicinal Chemistry: the art of transforming peptides in drugs A Guarna, A Trabocchi John Wiley & Sons, 2014 | 86 | 2014 |
Diversity-oriented synthesis: Basics and applications in organic synthesis, drug discovery, and chemical biology A Trabocchi John Wiley & Sons, 2013 | 80 | 2013 |
Click-chemistry-derived triazole ligands of arginine− glycine− aspartate (RGD) integrins with a broad capacity to inhibit adhesion of melanoma cells and both in vitro and in … A Trabocchi, G Menchi, N Cini, F Bianchini, S Raspanti, A Bottoncetti, ... Journal of medicinal chemistry 53 (19), 7119-7128, 2010 | 63 | 2010 |
Synthesis and Conformational Analysis of Small Peptides Containing 6-Endo-BT(t)L Scaffolds as Reverse Turn Mimetics A Trabocchi, EG Occhiato, D Potenza, A Guarna The Journal of Organic Chemistry 67 (21), 7483-7492, 2002 | 60 | 2002 |
Synthesis and reactivity of bicycles derived from tartaric acid and α-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3 … A Guarna, A Guidi, F Machetti, G Menchi, EG Occhiato, D Scarpi, S Sisi, ... The Journal of Organic Chemistry 64 (20), 7347-7364, 1999 | 56 | 1999 |
Exploring the chemical space and the bioactivity profile of lactams: a chemoinformatic study FI Saldívar-González, E Lenci, A Trabocchi, JL Medina-Franco RSC advances 9 (46), 27105-27116, 2019 | 55 | 2019 |
Carbohydrates in diversity-oriented synthesis: challenges and opportunities E Lenci, G Menchi, A Trabocchi Organic & Biomolecular Chemistry 14 (3), 808-825, 2016 | 53 | 2016 |
Occurrence of morpholine in central nervous system drug discovery E Lenci, L Calugi, A Trabocchi ACS Chemical Neuroscience 12 (3), 378-390, 2021 | 49 | 2021 |
Novel small molecules for the treatment of infections caused by Candida albicans: a patent review (2002 – 2010) C Calugi, A Trabocchi, A Guarna Expert opinion on therapeutic patents 21 (3), 381-397, 2011 | 43 | 2011 |
Diversity-oriented synthesis of morpholine-containing molecular scaffolds C Lalli, A Trabocchi, F Sladojevich, G Menchi, A Guarna Chemistry-a European Journal 15, 7871-7875, 2009 | 42 | 2009 |
Convenient route to enantiopure fmoc-protected morpholine-3-carboxylic acid F Sladojevich, A Trabocchi, A Guarna The Journal of Organic Chemistry 72 (11), 4254-4257, 2007 | 42 | 2007 |
Diversity-oriented synthesis as a tool for chemical genetics E Lenci, A Guarna, A Trabocchi Molecules 19 (10), 16506-16528, 2014 | 38 | 2014 |
Synthesis of a new enantiopure bicyclic γ/δ-amino acid (BTKa) derived from tartaric acid and α-amino acetophenone A Guarna, I Bucelli, F Machetti, G Menchi, EG Occhiato, D Scarpi, ... Tetrahedron 58 (49), 9865-9870, 2002 | 38 | 2002 |
Stereoselective cyclopropanation of serine-and threonine-derived oxazines to access new morpholine-based scaffolds F Sladojevich, A Trabocchi, A Guarna Organic & Biomolecular Chemistry 6 (18), 3328-3336, 2008 | 37 | 2008 |
Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds A Trabocchi, C Mannino, F Machetti, F De Bernardis, S Arancia, R Cauda, ... Journal of medicinal chemistry 53 (6), 2502-2509, 2010 | 36 | 2010 |