| A small-molecule P2RX7 activator promotes anti-tumor immune responses and sensitizes lung tumor to immunotherapy L Douguet, S Janho dit Hreich, J Benzaquen, L Seguin, T Juhel, ... Nature Communications 12 (1), 653, 2021 | 54 | 2021 |
| From conventional Lewis acids to heterogeneous montmorillonite K10: eco‐friendly plant‐based catalysts used as green Lewis acids M Hechelski, A Ghinet, B Louvel, P Dufrénoy, B Rigo, A Daïch, C Waterlot ChemSusChem 11 (8), 1249-1277, 2018 | 54 | 2018 |
| Synthesis and anticancer activity of analogues of phenstatin, with a phenothiazine A-ring, as a new class of microtubule-targeting agents CM Abuhaie, E Bîcu, B Rigo, P Gautret, D Belei, A Farce, J Dubois, ... Bioorganic & medicinal chemistry letters 23 (1), 147-152, 2013 | 50 | 2013 |
| Involvement of the P2X7 purinergic receptor in inflammation: an update of antagonists series since 2009 and their promising therapeutic potential D Baudelet, E Lipka, R Millet, A Ghinet Current Medicinal Chemistry 22 (6), 713-729, 2015 | 48 | 2015 |
| New farnesyltransferase inhibitors in the phenothiazine series D Belei, C Dumea, A Samson, A Farce, J Dubois, E Bîcu, A Ghinet Bioorganic & medicinal chemistry letters 22 (14), 4517-4522, 2012 | 48 | 2012 |
| Studies on indolizines. Evaluation of their biological properties as microtubule-interacting agents and as melanoma targeting compounds A Ghinet, CM Abuhaie, P Gautret, B Rigo, J Dubois, A Farce, D Belei, ... European Journal of Medicinal Chemistry 89, 115-127, 2015 | 44 | 2015 |
| Synthesis and biological evaluation of phenstatin metabolites A Ghinet, B Rigo, JP Hénichart, D Le Broc-Ryckewaert, J Pommery, ... Bioorganic & medicinal chemistry 19 (20), 6042-6054, 2011 | 40 | 2011 |
| Design, synthesis and evaluation of hydrazine and acyl hydrazone derivatives of 5-pyrrolidin-2-one as antifungal agents AE Dascalu, A Ghinet, E Lipka, C Furman, B Rigo, A Fayeulle, ... Bioorganic & Medicinal Chemistry Letters 30 (13), 127220, 2020 | 37 | 2020 |
| Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin A Ghinet, A Tourteau, B Rigo, V Stocker, M Leman, A Farce, J Dubois, ... Bioorganic & medicinal chemistry 21 (11), 2932-2940, 2013 | 36 | 2013 |
| New indolizine–chalcones as potent inhibitors of human farnesyltransferase: design, synthesis and biological evaluation IM Moise, A Ghinet, D Belei, J Dubois, A Farce, E Bîcu Bioorganic & Medicinal Chemistry Letters 26 (15), 3730-3734, 2016 | 34 | 2016 |
| Synthesis of triazoloquinazolinone based compounds as tubulin polymerization inhibitors and vascular disrupting agents M Driowya, J Leclercq, V Verones, A Barczyk, M Lecoeur, N Renault, ... European journal of medicinal chemistry 115, 393-405, 2016 | 34 | 2016 |
| Pyroglutamide-based P2X7 receptor antagonists targeting inflammatory bowel disease G Homerin, S Jawhara, X Dezitter, D Baudelet, P Dufrénoy, B Rigo, ... Journal of Medicinal Chemistry 63 (5), 2074-2094, 2019 | 32 | 2019 |
| Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors CM Abuhaie, A Ghinet, A Farce, J Dubois, P Gautret, B Rigo, D Belei, ... European Journal of Medicinal Chemistry 59, 101-110, 2013 | 32 | 2013 |
| Studies on phenothiazines: New microtubule-interacting compounds with phenothiazine A-ring as potent antineoplastic agents A Ghinet, IM Moise, B Rigo, G Homerin, A Farce, J Dubois, E Bicu Bioorganic & Medicinal Chemistry 24 (10), 2307-2317, 2016 | 31 | 2016 |
| Synthesis and biological evaluation of new phenothiazine derivatives bearing a pyrazole unit as protein farnesyltransferase inhibitors L Baciu-Atudosie, A Ghinet, A Farce, J Dubois, D Belei, E Bîcu Bioorganic & medicinal chemistry letters 22 (22), 6896-6902, 2012 | 31 | 2012 |
| Discovery of indolizines containing triazine moiety as new leads for the development of antitumoral agents targeting mitotic events L Lucescu, A Ghinet, D Belei, B Rigo, J Dubois, E Bîcu Bioorganic & Medicinal Chemistry Letters 25 (18), 3975-3979, 2015 | 30 | 2015 |
| Conformational Restriction Leading to a Selective CB2 Cannabinoid Receptor Agonist Orally Active Against Colitis J El Bakali, GG Muccioli, M Body-Malapel, M Djouina, F Klupsch, A Ghinet, ... ACS Medicinal Chemistry Letters 6 (2), 198-203, 2015 | 30 | 2015 |
| Novel indolizine derivatives with unprecedented inhibitory activity on human farnesyltransferase C Dumea, D Belei, A Ghinet, J Dubois, A Farce, E Bîcu Bioorganic & Medicinal Chemistry Letters 24 (24), 5777-5781, 2014 | 29 | 2014 |
| Enantioseparation of pyroglutamide derivatives on polysaccharide based chiral stationary phases by high-performance liquid chromatography and supercritical fluid chromatography … D Baudelet, N Schifano-Faux, A Ghinet, X Dezitter, F Barbotin, P Gautret, ... Journal of Chromatography A 1363, 257-269, 2014 | 25 | 2014 |
| The receptor for advanced glycation end products is a sensor for cell‐free heme O May, L Yatime, NS Merle, F Delguste, M Howsam, MV Daugan, ... The FEBS Journal 288 (11), 3448-3464, 2021 | 22 | 2021 |
