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Ajit Jagtap
Ajit Jagtap
Center of Drug Design, University of Minnesota
在 umn.edu 的电子邮件经过验证
标题
引用次数
引用次数
年份
Ureas: applications in drug design
A Dhananjay Jagtap, N Bharatrao Kondekar, A A Sadani, JW Chern
Current Medicinal Chemistry 24 (6), 622-651, 2017
602017
Novel acylureidoindolin-2-one derivatives as dual Aurora B/FLT3 inhibitors for the treatment of acute myeloid leukemia
AD Jagtap, PT Chang, JR Liu, HC Wang, NB Kondekar, LJ Shen, ...
European Journal of Medicinal Chemistry 85, 268-288, 2014
312014
Bioisosteric replacement of an acylureido moiety attached to an indolin-2-one scaffold with a malonamido or a 2/4-pyridinoylamido moiety produces a selectively potent Aurora-B …
HC Wang, AD Jagtap, PT Chang, JR Liu, CP Liu, HW Tseng, GS Chen, ...
European Journal of Medicinal Chemistry 84, 312-334, 2014
202014
4-Substituted 2-amino-3, 4-dihydroquinazolines with a 3-hairpin turn side chain as novel inhibitors of BACE-1
AD Jagtap, NB Kondekar, PY Hung, CE Hsieh, CR Yang, GS Chen, ...
Bioorganic Chemistry 95, 103135, 2020
102020
Discovery of HDAC6, HDAC8, and 6/8 inhibitors and development of cell-based drug screening models for the treatment of TGF-β-induced idiopathic pulmonary fibrosis
WC Yu, TY Yeh, CH Ye, PCT Chong, YH Ho, DK So, KY Yap, GR Peng, ...
Journal of Medicinal Chemistry 66 (15), 10528-10557, 2023
62023
Indolin-2-one derivatives as protein kinase inhibitors
JW Chern, AD Jagtap, HC Wang, GS Chen
US Patent 8,946,282, 2015
32015
Isoindole-1, 3-dione-based _ampersandsignalpha;, _ampersandsigngamma;-diketo acid bioisosteres as hepatitis C virus NS5B polymerase inhibitors
RR Deore, AD Jagtap, PT Chang, JW Chern
Journal of Asian Association of Schools of Pharmacy 1, 210-225, 2012
12012
Inhibiting HCMV pUL89-C Endonuclease with Metal-Binding Compounds: Miniperspective
AD Jagtap, RJ Geraghty, Z Wang
Journal of medicinal chemistry 66 (20), 13874-13887, 2023
2023
Quinazoline derivatives useful as selective hdac6 inhibitors
YU Chao-Wu, H Pei-Yun, AD Jagtap, HO Yi-Hsun, HY Chaing
US Patent App. 18/001,002, 2023
2023
Quinazoline Derivatives Useful as Selective HDAC6 Inhibitors
HYC Ji-Wang Chern, Chao-Wu Yu, Pei-Yun Hung, Ajit Dhananjay Jagtap, Yi-Hsun Ho
WO Patent WO2021252475A1, 2021
2021
Novel acylureidoindolin-2-one derivatives as dual Aurora B/FLT3 inhibitors for treatment of acute myeloid leukemia
KD Wu, JR Liu, ST Fung, YH Ho, KJ Wang, GY Chen, AD Jagtap, ...
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 250, 2015
2015
Indolin-2-one derivatives as protein kinase inhibitors
GSC Ji-Wang Chern, Ajit Dhananjay Jagtap, Hsiao-Chun Wang
WO Patent WO2013158373A8, 2014
2014
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