Synthesis of indolo/pyrroloazepinone-oxindoles as potential cytotoxic, DNA-intercalating and Topo I inhibitors M Kadagathur, AS Shaikh, B Panda, J George, R Phanindranath, ... Bioorganic Chemistry 122, 105706, 2022 | 15 | 2022 |
Exploration of mercaptoacetamide-linked pyrimidine-1, 3, 4-oxadiazole derivatives as DNA intercalative topo II inhibitors: Cytotoxicity and apoptosis induction AS Shaikh, G Kiranmai, GP Devi, PN Makhal, DK Sigalapalli, R Tokala, ... Bioorganic & Medicinal Chemistry Letters 65, 128697, 2022 | 13 | 2022 |
Design, synthesis of DNA-interactive 4-thiazolidinone-based indolo-/pyrroloazepinone conjugates as potential cytotoxic and topoisomerase I inhibitors M Kadagathur, S Patra, G Devabattula, J George, R Phanindranath, ... European Journal of Medicinal Chemistry 238, 114465, 2022 | 12 | 2022 |
Cyclodesulfurization: an enabling protocol for synthesis of various heterocycles M Kadagathur, AS Shaikh, GS Jadhav, DK Sigalapalli, N Shankaraiah, ... ChemistrySelect 6 (10), 2621-2640, 2021 | 11 | 2021 |
Insights into the pharmacophore-based 3D-QSAR modeling, molecular dynamics simulation studies of certain dihydroxy pyrrolidine/piperidine and aza-flavanone derivatives as α … DK Sigalapalli, V Yele, S Jupudi, AS Shaikh, M Kadagathur, ... Journal of Molecular Structure 1223, 129243, 2021 | 5 | 2021 |
Oxyberberine an oxoderivative of berberine confers neuroprotective effects in controlled-cortical impact mouse model of traumatic brain injury PM Tentu, MR Bazaz, T Pasam, AS Shaikh, Z Rahman, A Mourya, ... International Journal of Neuroscience, 1-16, 2023 | 4 | 2023 |
Disulfiram prevents collagen crosslinking and inhibits renal fibrosis by inhibiting lysyl oxidase enzymes MA Saifi, AS Shaikh, VR Kaki, C Godugu Journal of Cellular Physiology 237 (5), 2516-2527, 2022 | 4 | 2022 |
TBHP‐Mediated Selenocyclization of N‐Allylbenzamides/Benzthioamides via In‐Situ Generation of “PhSeOH” Species** PN Makhal, SR Dannarm, AS Shaikh, R Sonti, VR Kaki ChemistrySelect 7 (14), e202200933, 2022 | 3 | 2022 |
Microwave‐assisted TBHP‐mediated synthesis of 2‐amino‐1, 3, 4‐oxadiazoles in water D Kumar Sigalapalli, M Kadagathur, A Sujat Shaikh, GS Jadhav, B Bakchi, ... ChemistrySelect 5 (42), 13248-13258, 2020 | 3 | 2020 |
Design, synthesis, anti-cancer activity and in-silico studies of some novel 4,5-dihydroisoxazole-5-carboxamide derivatives S Endoori, KC Gulipalli, S Bodige, AS Shaikh, D Vemula, SR Surapureddi, ... Synthetic Communications 51 (22), 3416-3426, 2021 | 2 | 2021 |
Quest for selective MMP9 inhibitors: a computational approach AS Shaikh, A Sethi, PN Makhal, B Rathi, VR Kaki Journal of Biomolecular Structure and Dynamics 41 (24), 15053-15066, 2023 | 1 | 2023 |
Naringenin-capped silver nanoparticles amalgamated gel for the treatment of cutaneous candidiasis C Katta, AS Shaikh, N Bhale, VGSS Jyothi, VR Kaki, AG Dikundwar, ... AAPS PharmSciTech 24 (5), 126, 2023 | 1 | 2023 |
Naringenin-Zinc Oxide Nanocomposites Amalgamated Polymeric Gel Augmented Drug Delivery and Attenuated Experimental Cutaneous Candidiasis in Balb/c Mice: In Vitro and In Vivo … C Katta, D Bahuguna, H Veerabomma, S Gollapalli, AS Shaikh, NA Bhale, ... AAPS PharmSciTech 25 (5), 130, 2024 | | 2024 |
Oxyberberine protects middle cerebral artery occlusion triggered cerebral injury through TLR4/NLRP3 pathway in rats Z Rahman, AS Shaikh, KV Rao, MP Dandekar Journal of Chemical Neuroanatomy 136, 102393, 2024 | | 2024 |
Development of trisubstituted thiophene-3-arboxamide selenide derivatives as novel EGFR kinase inhibitors with cytotoxic activity PN Makhal, A Sood, AS Shaikh, LN Dayare, DK Khatri, VR Kaki RSC Medicinal Chemistry 14 (12), 2677-2698, 2023 | | 2023 |
Exo-trig selenocyclization of secondary allylic carboxamides using Woollins’ reagent: en route to 2, 5-disubstituted selenazolines PN Makhal, SR Dannarm, AS Shaikh, R Ahmed, S Chilvery, LN Dayare, ... Chemical Communications 59 (25), 3767-3770, 2023 | | 2023 |
Research Philosophy, Ethics, and Environmental Aspects PN Makhal, AS Shaikh, LN Dayare, VR Kaki Principles of Research Methodology and Ethics in Pharmaceutical Sciences …, 0 | | |