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Raveendra Dayam
Raveendra Dayam
Excelra Knowledge Solutions Private Limited
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标题
引用次数
引用次数
年份
Rational design and synthesis of novel dimeric diketoacid-containing inhibitors of HIV-1 integrase: implication for binding to two metal ions on the active site of integrase
YQ Long, XH Jiang, R Dayam, T Sanchez, R Shoemaker, S Sei, ...
Journal of medicinal chemistry 47 (10), 2561-2573, 2004
2402004
Discovery of structurally diverse HIV-1 integrase inhibitors based on a chalcone pharmacophore
J Deng, T Sanchez, LQ Al-Mawsawi, R Dayam, RA Yunes, A Garofalo, ...
Bioorganic & medicinal chemistry 15 (14), 4985-5002, 2007
2142007
Design and synthesis of novel indole β-diketo acid derivatives as HIV-1 integrase inhibitors
M Sechi, M Derudas, R Dallocchio, A Dessì, A Bacchi, L Sannia, F Carta, ...
Journal of medicinal chemistry 47 (21), 5298-5310, 2004
1752004
Discovery of small molecule integrin αvβ3 antagonists as novel anticancer agents
R Dayam, F Aiello, J Deng, Y Wu, A Garofalo, X Chen, N Neamati
Journal of medicinal chemistry 49 (15), 4526-4534, 2006
1572006
β-Diketo acid pharmacophore hypothesis. 1. Discovery of a novel class of HIV-1 integrase inhibitors
R Dayam, T Sanchez, O Clement, R Shoemaker, S Sei, N Neamati
Journal of medicinal chemistry 48 (1), 111-120, 2005
1572005
Discovery of novel small-molecule inhibitors of human epidermal growth factor receptor-2: Combined ligand and target-based approach
R Gundla, R Kazemi, R Sanam, R Muttineni, JARP Sarma, R Dayam, ...
Journal of medicinal chemistry 51 (12), 3367-3377, 2008
1522008
Discovery of a small-molecule HIV-1 integrase inhibitor-binding site
LQ Al-Mawsawi, V Fikkert, R Dayam, M Witvrouw, TR Burke Jr, ...
Proceedings of the National Academy of Sciences 103 (26), 10080-10085, 2006
1372006
HIV‐1 integrase inhibitors: 2005–2006 update
R Dayam, R Gundla, LQ Al‐Mawsawi, N Neamati
Medicinal Research Reviews 28 (1), 118-154, 2008
1252008
Quinolone 3-carboxylic acid pharmacophore: design of second generation HIV-1 integrase inhibitors
R Dayam, LQ Al-Mawsawi, Z Zawahir, M Witvrouw, Z Debyser, N Neamati
Journal of medicinal chemistry 51 (5), 1136-1144, 2008
1182008
Small-molecule HIV-1 integrase inhibitors: the 2001-2002 update
R Dayam, N Neamati
Current pharmaceutical design 9 (22), 1789-1802, 2003
1112003
HIV‐1 integrase inhibitors: 2003–2004 update
R Dayam, J Deng, N Neamati
Medicinal research reviews 26 (3), 271-309, 2006
982006
Diketo acid pharmacophore. 2. Discovery of structurally diverse inhibitors of HIV-1 integrase
R Dayam, T Sanchez, N Neamati
Journal of medicinal chemistry 48 (25), 8009-8015, 2005
852005
Discovery of novel non-cytotoxic salicylhydrazide containing HIV-1 integrase inhibitors
LQ Al-Mawsawi, R Dayam, L Taheri, M Witvrouw, Z Debyser, N Neamati
Bioorganic & medicinal chemistry letters 17 (23), 6472-6475, 2007
802007
Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors
M Sechi, G Rizzi, A Bacchi, M Carcelli, D Rogolino, N Pala, TW Sanchez, ...
Bioorganic & medicinal chemistry 17 (7), 2925-2935, 2009
782009
Pharmacophore guided discovery of small-molecule human apurinic/apyrimidinic endonuclease 1 inhibitors
Z Zawahir, R Dayam, J Deng, C Pereira, N Neamati
Journal of medicinal chemistry 52 (1), 20-32, 2009
782009
Active site binding modes of the β-diketoacids: a multi-active site approach in HIV-1 integrase inhibitor design
R Dayam, N Neamati
Bioorganic & medicinal chemistry 12 (24), 6371-6381, 2004
772004
HIV-1 integrase inhibitors: an emerging clinical reality
R Dayam, LQ Al-Mawsawi, N Neamati
Drugs in R & D 8, 155-168, 2007
702007
Inhibitory profile of a LEDGF/p75 peptide against HIV-1 integrase: Insight into integrase–DNA complex formation and catalysis
LQ Al-Mawsawi, F Christ, R Dayam, Z Debyser, N Neamati
FEBS letters 582 (10), 1425-1430, 2008
692008
Discovery and preclinical evaluation of a novel class of small-molecule compounds in hormone-dependent and-independent cancer cell lines
C Plasencia, R Dayam, Q Wang, J Pinski, TR Burke Jr, DI Quinn, ...
Molecular cancer therapeutics 4 (7), 1105-1113, 2005
642005
Fibroblast growth factor receptor inhibitors
S Kumar BVS, L Narasu, R Gundla, R Dayam, S JARP
Current pharmaceutical design 19 (4), 687-701, 2013
472013
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