Coumarins effectively inhibit bacterial α-carbonic anhydrases S Giovannuzzi, CS Hewitt, A Nocentini, C Capasso, DP Flaherty, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 333-338, 2022 | 31 | 2022 |
Inhibition studies of bacterial α-carbonic anhydrases with phenols S Giovannuzzi, CS Hewitt, A Nocentini, C Capasso, G Costantino, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 666-671, 2022 | 22 | 2022 |
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae S Giovannuzzi, NS Abutaleb, CS Hewitt, F Carta, A Nocentini, MN Seleem, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1-8, 2022 | 21 | 2022 |
4-(3-Alkyl/benzyl-guanidino) benzenesulfonamides as selective carbonic anhydrase VII inhibitors M Abdoli, S Giovannuzzi, CT Supuran, R Žalubovskis Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1568-1576, 2022 | 16 | 2022 |
Aromatic sulfonamides including a sulfonic acid tail: new membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer-associated isoforms S Giovannuzzi, M D’Ambrosio, C Luceri, SM Osman, M Pallecchi, ... International Journal of Molecular Sciences 23 (1), 461, 2021 | 15 | 2021 |
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful … V De Luca, S Giovannuzzi, CT Supuran, C Capasso International Journal of Molecular Sciences 23 (22), 13827, 2022 | 12 | 2022 |
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum S Giovannuzzi, V De Luca, A Nocentini, C Capasso, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 680-685, 2022 | 11 | 2022 |
Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties S Saied, M Shaldam, MM Elbadawi, S Giovannuzzi, A Nocentini, ... European Journal of Medicinal Chemistry 259, 115707, 2023 | 9 | 2023 |
1, 5-diaryl-1, 2, 4-triazole ureas as new SLC-0111 analogues endowed with dual carbonic anhydrase and VEGFR-2 inhibitory activities AE Elsawi, MM Elbadawi, A Nocentini, H Almahli, S Giovannuzzi, ... Journal of Medicinal Chemistry 66 (15), 10558-10578, 2023 | 9 | 2023 |
Continued structural exploration of sulfocoumarin as selective inhibitor of tumor-associated human carbonic anhydrases ix and XII S Giovannuzzi, C Capasso, A Nocentini, CT Supuran Molecules 27 (13), 4076, 2022 | 7 | 2022 |
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates S Giovannuzzi, AK Marapaka, NS Abutaleb, F Carta, HW Liang, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2284119, 2023 | 6 | 2023 |
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ S Giovannuzzi, V De Luca, C Capasso, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2173748, 2023 | 5 | 2023 |
Boron-containing carbonic anhydrases inhibitors S Giovannuzzi, A Nikitjuka, BRP Resende, M Smietana, A Nocentini, ... Bioorganic Chemistry, 106976, 2023 | 4 | 2023 |
Potent inhibitors of tumor associated carbonic anhydrases endowed with cathepsin B inhibition A Kumar, P Arya, V Sharma, S Giovannuzzi, N Raghav, CT Supuran, ... Archiv der Pharmazie 356 (11), 2300349, 2023 | 4 | 2023 |
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae A Bonardi, A Nocentini, S Giovannuzzi, N Paoletti, A Ammara, S Bua, ... Journal of Medicinal Chemistry, 2024 | 3 | 2024 |
Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: design, synthesis and anti-proliferative activity S Higazy, N Samir, A El-Khouly, S Giovannuzzi, P Begines, HM Gaber, ... Bioorganic Chemistry 144, 107089, 2024 | 3 | 2024 |
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides S Akocak, N Lolak, S Giovannuzzi, CT Supuran Bioorganic & Medicinal Chemistry Letters 95, 129479, 2023 | 3 | 2023 |
Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR-2 as Potential Agents for Solid Tumors: X-ray, In Vitro, In Vivo, and In Silico … SM Hefny, TF El-Moselhy, N El-Din, S Giovannuzzi, T Bin Traiki, ... Journal of Medicinal Chemistry 67 (9), 7406-7430, 2024 | 2 | 2024 |
1, 2, 3‐Triazole‐based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition K Siwach, M Rani, L Vats, S Giovannuzzi, AK Paul, M Brahma, N Kumari, ... Archiv der Pharmazie 357 (3), 2300372, 2024 | 2 | 2024 |
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies P Begines, A Bonardi, A Nocentini, P Gratteri, S Giovannuzzi, R Ronca, ... Bioorganic & Medicinal Chemistry 94, 117467, 2023 | 2 | 2023 |