A multitiered analysis platform for genome sequencing: Design and initial findings of the Australian Genomics Cardiovascular Disorders Flagship R Austin, JS Brown, S Casauria, EO Madelli, T Mattiske, T Boughtwood, ... Genetics in Medicine Open 2, 101842, 2024 | | 2024 |
Compounds and their use in treating cancer IN Michaelides, U Börjesson, TGC Hayhow, JG Kettle, GW Collie, ... US Patent App. 18/247,014, 2023 | | 2023 |
The role of allylic strain for conformational control in medicinal chemistry H Zhao, J Brånalt, M Perry, C Tyrchan Journal of Medicinal Chemistry 66 (12), 7730-7755, 2023 | 6 | 2023 |
Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3-3 Protein–Protein Interaction JS Pallesen, CC Munier, F Bosica, SA Andrei, K Edman, A Gunnarsson, ... Journal of medicinal chemistry 65 (24), 16818-16828, 2022 | 6 | 2022 |
Surprising lipophilicity observations identify unexpected conformational effects MWD Perry, U Börjesson, A Nikitidis, C Tyrchan Bioorganic & Medicinal Chemistry Letters 69, 128786, 2022 | 1 | 2022 |
Novel inhibitors of phosphatidylinositol 3-kinase gamma M Mogemark, N Pemberton, J Petersen, M Perry, K Karabelas, ... | | 2021 |
PI3K inhibitors are finally coming of age B Vanhaesebroeck, MWD Perry, JR Brown, F André, K Okkenhaug Nature reviews Drug discovery 20 (10), 741-769, 2021 | 300 | 2021 |
Dual inhibitors of phosphatidylinositol 3-kinase delta & gamma M Perry, C Tyrchan, K Karabelas, A Nikitidis, M Mogemark, J Petersen, ... US Patent App. 17/173,826, 2021 | | 2021 |
Discovery of AZD8154, a dual PI3Kγδ inhibitor for the treatment of asthma MWD Perry, K Bjorhall, P Bold, M Brulls, U Borjesson, J Carlsson, ... Journal of Medicinal Chemistry 64 (12), 8053-8075, 2021 | 25 | 2021 |
Derivados de 5-[2-(piridin-2-ilamino)-1, 3-tiazol-5-il]-2, 3-dihidro-1H-isoindol-1-ona y su uso como inhibidores dobles de fosfatidilinositol·· 3-cinasa delta y gamma M Perry, K Karabelas, M Mogemark, P Bold, C Tyrchan, A Nikitidis, ... ES Patent App. 17,772,381 T, 2021 | | 2021 |
(S)-2-(1-cyclopropylethyl)-5-(4-methyl-2-((6-(2-oxopyrrolidin-1-yl) pyridin-2-yl) amino) thiazol-5-yl)-7-(methylsulfonyl) isoindolin-1-one as a phosphatidylinositol 3-kinase … M Perry, C Tyrchan, K Karabelas, A Nikitidis, M Mogemark, J Petersen, ... US Patent 10,961,236, 2021 | | 2021 |
Pochodne 5-[2-(pirydyn-2-yloamino)-1, 3-tiazol-5-ilo]-2, 3-dihydro-1h-izoindol-1-onu i ich zastosowanie jako podwójnych inhibitorów 3-kinazy fosfatydyloinozytolu delta i gamma M Perry, K Karabelas, M Mogemark, P Bold, C Tyrchan, A Nikitidis, ... | | 2021 |
The Cascade Reactions of Indigo with Propargyl Substrates for Heterocyclic and Photophysical Diversity PM McCosker, NM Butler, A Shakoori, MK Volland, MJ Perry, JW Mullen, ... Chemistry–A European Journal 27 (11), 3708-3721, 2021 | 6 | 2021 |
Inhibitors of phosphatidylinositol 3-kinase gamma M Mogemark, N Pemberton, J Petersen, M Perry, K Karabelas, ... US Patent App. 17/088,689, 2021 | | 2021 |
Glucocorticoid receptor Thr524 phosphorylation by MINK1 induces interactions with 14-3-3 protein regulators CC Munier, L De Maria, K Edman, A Gunnarsson, M Longo, ... Journal of Biological Chemistry 296, 2021 | 12 | 2021 |
The API B Bonn, M Perry Inhaled Medicines, 13-34, 2021 | 4 | 2021 |
14-3-3 modulation of the inflammatory response CC Munier, C Ottmann, MWD Perry Pharmacological research 163, 105236, 2021 | 62 | 2021 |
Inhibitors of phosphatidylinositol 3-kinase gamma M Mogemark, N Pemberton, J Petersen, M Perry, K Karabelas, ... US Patent 10,858,355, 2020 | | 2020 |
Derivati 5-[2-(piridin-2-ilamino)-1, 3-tiazol-5-il]-2, 3-dihidro-1h-izoindol-1-ona i njihova upotreba kao dvostrukih inhibitora fosfatidilinozitola 3-kinaze delta i gama M Perry, K Karabelas, M Mogemark, P Bold, C Tyrchan, A Nikitidis, ... HR Patent App. P20201175T T, 2020 | | 2020 |
5-[2-(piridin-2-ilamino)-1, 3-tiazol-5-il]-2, 3-dihidro-1h-izoindol-1-ono dariniai ir jų naudojimas kaip fosfatatidilitinozitol 3-kinazės delta ir gama dvejopų inhibitorių M Perry, K Karabelas, M Mogemark, P Bold, C Tyrchan, A Nikitidis, ... | | 2020 |