| In vitro assessment of the risk of ABCB1-mediated drug-drug interaction between rivaroxaban and tacrolimus in HEK293 recombinant cell lines G Mahieu, AL Sennesael, L Pochet, V Haufroid, F Van Bambeke, ... Research and Practice in Thrombosis and Haemostasis, 102521, 2024 | | 2024 |
| Advances in Targeting Kainic Acid Receptors: Developing Selective Positive Allosteric Modulators from the 1, 2, 4-Benzothiadiazine 1, 1-Dioxide scaffold T Colson, M Piette, Y Bay, DS Pickering, AS Kristensen, G Baudino, ... CIRM Day 2024, 2024 | | 2024 |
| Kainic Acid Receptors: Innovating Selective Positive Allosteric Modulators based on 1, 2, 4-Benzothiadiazine 1, 1-Dioxides T Colson, M Piette, Y Bay, DS Pickering, AS Kristensen, G Baudino, ... MedChem 2023, 2023 | | 2023 |
| Coumarins as factor XIIa inhibitors: Potency and selectivity improvements using a fragment-based strategy C Davoine, A Traina, J Evrard, S Lanners, M Fillet, L Pochet European Journal of Medicinal Chemistry 259, 115636, 2023 | 4 | 2023 |
| Activity and affinity assays by capillary electrophoresis in the context of drug screening C Davoine, L Pochet, M Fillet Jinan University, 2023 | | 2023 |
| Intérêt de l’EC dans le contexte du développement de médicaments pour le screening de ligands et la caractérisation de leur interaction avec la cible thérapeutique C Davoine, L Pochet, M Fillet Conférence «La Chimie Analytique au service de la Santé», 2023 | | 2023 |
| Advances in analytical technologies detecting and characterizing noncovalent interactions for fragment-based drug discovery C Davoine, L Pochet, M Fillet TrAC Trends in Analytical Chemistry, 117161, 2023 | 2 | 2023 |
| Affinity Capillary Electrophoresis for Fragment-based Drug Discovery Projects: Hit Discovery and Binding Site Characterization C Davoine, L Pochet, M Fillet 12th International Symposium on Drug Analysis and the 32nd International …, 2022 | | 2022 |
| Affinity Capillary Electrophoresis in Fragment-based Drug Discovery Projects, A tool for Hit discovery and Binding site Characterization C Davoine, L Pochet, M Fillet 38th International Symposium on Microscale Separations and Bioanalysis (MSB …, 2022 | | 2022 |
| Discovery of Potent FXIIa Inhibitors using a Fragment-based Strategy C Davoine, M Fillet, L Pochet FNRS Med Chem Meeting, 2022 | | 2022 |
| Development of Factor XIIa Inhibitors Assisted by Affinity Capillary Electrophoresis, A Fragment-based Lead Discovery Project C Davoine, L Pochet, M Fillet CIRM day 2022, 2022 | | 2022 |
| Fragment hit discovery and binding site characterization by indirect affinity capillary electrophoresis: application to factor XIIa C Davoine, A Pardo, L Pochet, M Fillet Analytical Chemistry 93 (44), 14802-14809, 2021 | 12 | 2021 |
| Key amino acid residues in homoserine-acetyltransferase from M. tuberculosis give insight into the evolution of MetX family of enzymes–HAT, SAT and HST B Maurya, M Colaço, J Wouters, L Pochet, S Misquith Biochimie 189, 13-25, 2021 | 2 | 2021 |
| Using Biochemical Assay and Capillary Electrophoresis to Explore Fragments against Coagulation Factor XIIa C Davoine, F Simon, C Bouckaert, M Fillet, L Pochet 8th EFMC Young Medicinal Chemists' Symposium, 2021 | | 2021 |
| Exploring Fragments to Design FXIIa Inhibitors with Biochemical Assay and Capillary Electrophoresis C Davoine, F Simon, S Lanners, M Fillet, L Pochet FNRS Med Chem Meeting, 2021 | | 2021 |
| Uncovering biochemical assay’s false positives by counter-screening a fragment library with affinity capillary electrophoresis C Davoine, M Fillet, L Pochet CIRM-day 2021, 2021 | | 2021 |
| Capillary electrophoresis as a fragment screening tool to cross-validate hits from chromogenic assay: Application to FXIIa C Davoine, M Fillet, L Pochet Talanta 226, 122163, 2021 | 8 | 2021 |
| Factor XII/XIIa inhibitors: Their discovery, development, and potential indications C Davoine, C Bouckaert, M Fillet, L Pochet European Journal of Medicinal Chemistry 208, 112753, 2020 | 50 | 2020 |
| Integrated synthesis using isothiocyanate-substituted aryllithiums by flow chemistry HJ Lee, D Torii, Y Jeon, J Yoshida, H Kim Synlett 31 (19), 1899-1902, 2020 | 6 | 2020 |
| MetA (Rv3341) from Mycobacterium tuberculosis H37Rv strain exhibits substrate dependent dual role of transferase and hydrolase activity B Maurya, L Pochet, J Wouters, M Colaço, S Misquith Biochimie 179, 113-126, 2020 | 5 | 2020 |
