Involvement of glutamate, oxidative stress and inducible nitric oxide synthase in the convulsant activity of ciprofloxacin in mice AO Abdel-Zaher, AHM Afify, SM Kamel, HM Farghaly, GM El-Osely, ... European journal of pharmacology 685 (1-3), 30-37, 2012 | 19 | 2012 |
Direct, gabapentin-insensitive interaction of a soluble form of the calcium channel subunit α2δ-1 with thrombospondin-4 E El-Awaad, G Pryymachuk, C Fried, J Matthes, J Isensee, T Hucho, ... Scientific Reports 9 (1), 16272, 2019 | 17 | 2019 |
Development of an in vitro screening assay for PIP5K1α lipid kinase and identification of potent inhibitors K Strätker, S Haidar, Á Amesty, E El‐Awaad, C Götz, A Estévez‐Braun, ... The FEBS Journal 287 (14), 3042-3064, 2020 | 10 | 2020 |
Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor E El-Awaad, R Birus, C Marminon, Z Bouaziz, L Ballentin, D Aichele, ... Pharmaceuticals 14 (6), 542, 2021 | 5 | 2021 |
[2.2] Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists R Rajan, D Schepmann, R Steigerwald, JA Schreiber, E El‐Awaad, ... ChemMedChem 16 (20), 3201-3209, 2021 | 4 | 2021 |
4,5,7‐Trisubstituted indeno[1,2‐b]indole inhibits CK2 activity in tumor cells equivalent to CX‐4945 and shows strong anti‐migratory effects R Birus, E El‐Awaad, L Ballentin, F Alchab, D Aichele, L Ettouati, C Götz, ... FEBS Open bio 12 (2), 394-411, 2022 | 2 | 2022 |
Angiotensin II type 1 receptor localizes at the blood–bile barrier in humans and pigs G Pryymachuk, E El-Awaad, N Piekarek, U Drebber, AC Maul, ... Histochemistry and Cell Biology 157 (5), 513-524, 2022 | 1 | 2022 |
Biological evaluation of 4, 5, 7-trisubstituted Indeno [1, 2-b] indoles reveals a potent inhibitor of Protein Kinase CK2 in tumor cells with diverse anti-cancer effects and … R Birus, E El-Awaad, L Ballentin, F Alchab, D Aichele, L Ettouati, C Götz, ... Published online In: 7th International Electronic Conference on Medicinal …, 2021 | 1 | 2021 |
1, 2, 3-Triazole-totarol conjugates as potent PIP5K1α lipid kinase inhibitors S Haidar, Á Amesty, S Oramas-Royo, C Götz, E El-Awaad, J Kaiser, ... Bioorganic & Medicinal Chemistry 105, 117727, 2024 | | 2024 |
Targeting lipid kinase PIP5K1α as a promising strategy for the treatment of castration-resistant prostate cancer E El-Awaad, K Strätker, S Haidar, Á Amesty, C Götz, A Estévez-Braun, ... MDPI, 2020 | | 2020 |
Characterization of the direct interaction between the extracellular matrix protein thrombospondin-4 and the gabapentin receptor α2δ-1 E El-Awaad Universität zu Köln, 2018 | | 2018 |
-Targeting of the thrombospondin-alpha 2 delta-1 interaction-Development of analgesics against neuropathic pain E El-Awaad, C Fried, G Pryymachuk, J Matthes, T Hucho, WF Neiss, ... Naunyn-Schmiedebergs Arch. Pharmacol. 388, S49-1, 2015 | | 2015 |