受强制性开放获取政策约束的文章 - Tomi Sawyer了解详情
无法在其他位置公开访问的文章：3 篇
9-(Arenethenyl) purines as dual Src/Abl kinase inhibitors targeting the inactive conformation: design, synthesis, and biological evaluation
WS Huang, X Zhu, Y Wang, M Azam, D Wen, R Sundaramoorthi, ...
Journal of medicinal chemistry 52 (15), 4743-4756, 2009
强制性开放获取政策： US National Institutes of Health
Renaissance in peptide drug discovery: the third wave
TK Sawyer
强制性开放获取政策： A*Star, Singapore
Liposome click membrane permeability assay for identifying permeable peptides
TJ Desai, B Habulihaz, JR Cannon, A Chandramohan, HYK Kaan, ...
Pharmaceutical Research 38, 843-850, 2021
强制性开放获取政策： A*Star, Singapore
可在其他位置公开访问的文章：14 篇
AP24534, a pan-BCR-ABL inhibitor for chronic myeloid leukemia, potently inhibits the T315I mutant and overcomes mutation-based resistance
T O'Hare, WC Shakespeare, X Zhu, CA Eide, VM Rivera, F Wang, ...
Cancer cell 16 (5), 401-412, 2009
强制性开放获取政策： Howard Hughes Medical Institute
Incorporation of putative helix-breaking amino acids in the design of novel stapled peptides: Exploring biophysical and cellular permeability properties
AW Partridge, HYK Kaan, YC Juang, A Sadruddin, S Lim, CJ Brown, S Ng, ...
Molecules 24 (12), 2292, 2019
强制性开放获取政策： A*Star, Singapore
NanoClick: a high throughput, target-agnostic peptide cell permeability assay
A Peier, L Ge, N Boyer, J Frost, R Duggal, K Biswas, S Edmondson, ...
ACS Chemical Biology 16 (2), 293-309, 2021
强制性开放获取政策： A*Star, Singapore
Targeting anti-cancer agents to bone using bisphosphonates
L Xing, FH Ebetino, RK Boeckman Jr, V Srinivasan, J Tao, TK Sawyer, J Li, ...
Bone 138, 115492, 2020
强制性开放获取政策： US National Institutes of Health
Macrocyclization of an all-d linear α-helical peptide imparts cellular permeability
S Kannan, PGA Aronica, S Ng, DTG Lian, Y Frosi, S Chee, J Shimin, ...
Chemical Science 11 (21), 5577-5591, 2020
强制性开放获取政策： A*Star, Singapore
De-risking drug discovery of intracellular targeting peptides: screening strategies to eliminate false-positive hits
S Ng, YC Juang, A Chandramohan, HYK Kaan, A Sadruddin, TY Yuen, ...
ACS Medicinal Chemistry Letters 11 (10), 1993-2001, 2020
强制性开放获取政策： A*Star, Singapore
AP24163 Inhibits the Gatekeeper Mutant of BCR‐ABL and Suppresses In vitro Resistance
M Azam, JT Powers, W Einhorn, WS Huang, WC Shakespeare, X Zhu, ...
Chemical biology & drug design 75 (2), 223-227, 2010
强制性开放获取政策： US National Institutes of Health
Discovery of cell active macrocyclic peptides with on-target inhibition of KRAS signaling
S Lim, N Boyer, N Boo, C Huang, G Venkatachalam, YCA Juang, ...
Chemical Science 12 (48), 15975-15987, 2021
强制性开放获取政策： A*Star, Singapore
Design-rules for stapled peptides with in vivo activity and their application to Mdm2/X antagonists
A Chandramohan, H Josien, TY Yuen, R Duggal, D Spiegelberg, L Yan, ...
Nature Communications 15 (1), 489, 2024
强制性开放获取政策： A*Star, Singapore
Demonstration of a Common DPhe7 to DNal(2′)7 Peptide Ligand Antagonist Switch for Melanocortin-3 and Melanocortin-4 Receptors Identifies the Systematic …
LE Gimenez, TA Noblin, SY Williams, S Mullick Bagchi, RL Ji, YX Tao, ...
Journal of Medicinal Chemistry 65 (8), 5990-6000, 2022
强制性开放获取政策： US National Institutes of Health
Inhibition of the melanocortin-3 receptor (MC3R) causes generalized sensitization to anorectic agents
NS Dahir, Y Gui, Y Wu, PR Sweeney, SY Williams, LE Gimenez, ...
bioRxiv, 2023
强制性开放获取政策： US National Institutes of Health
Aqueous remote loading of setmelanotide in poly (lactic-co-glycolic acid) microspheres for long-term obesity treatment
S Wang, G Downing, KF Olsen, TK Sawyer, RD Cone, SP Schwendeman
Journal of Controlled Release 364, 589-600, 2023
强制性开放获取政策： US National Institutes of Health
Design-Rules for Stapled Alpha-Helical Peptides with On-Target In Vivo Activity: Application to Mdm2/X dual antagonists
A Chandramohan, H Josien, TY Yuen, R Duggal, D Spiegelberg, L Yan, ...
Biorxiv, 2023.02. 25.530030, 2023
强制性开放获取政策： A*Star, Singapore
Macrocyclization of an all-D linear peptide improves target affinity and imparts cellular activity: A novel stapled α-helical peptide modality
S Kannan, PGA Aronica, S Ng, D Thean, Y Frosi, S Chee, J Shimin, ...
bioRxiv, 767673, 2019
强制性开放获取政策： A*Star, Singapore
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