Synthesis and evaluation of phosphorus containing, specific CDK9/CycT1 inhibitors G Németh, Z Greff, A Sipos, Z Varga, R Székely, M Sebestyén, Z Jászay, ... Journal of medicinal chemistry 57 (10), 3939-3965, 2014 | 81 | 2014 |
Oxaphosphinanes: new therapeutic perspectives for glioblastoma L Clarion, C Jacquard, O Sainte-Catherine, S Loiseau, D Filippini, ... Journal of Medicinal Chemistry 55 (5), 2196-2211, 2012 | 76 | 2012 |
Regio-and stereoselective synthesis of 2-amino-1-hydroxy-2-aryl ethylphosphonic esters HJ Cristau, JL Pirat, M Drag, P Kafarski Tetrahedron Letters 41 (50), 9781-9785, 2000 | 67 | 2000 |
Oxaphospholene and oxaphosphinene heterocycles via RCM using unsymmetrical phosphonates or functional phosphinates P Fourgeaud, C Midrier, JP Vors, JN Volle, JL Pirat, D Virieux Tetrahedron 66 (3), 758-764, 2010 | 65 | 2010 |
Fatty hydroxamic acid biosynthesis in aqueous medium in the presence of the lipase-acyltransferase from Candida parapsilosis L Vaysse, E Dubreucq, JL Pirat, P Galzy Journal of biotechnology 53 (1), 41-46, 1997 | 58 | 1997 |
A convenient one-pot synthesis of phosphino-dipeptide analogs HJ Cristau, A Coulombeau, A Genevois-Borella, JL Pirat Tetrahedron Letters 42 (27), 4491-4494, 2001 | 46 | 2001 |
Enantioselective reactions catalyzed by phosphine oxides T Ayad, A Gernet, JL Pirat, D Virieux Tetrahedron 75 (33), 4385-4418, 2019 | 45 | 2019 |
NMDA receptor channels: Labeling of MK-801 with iodine-125 and fluorine-18 DM Wieland, MR Kilbourn, DJ Yang, E Laborde, DL Gildersleeve, ... International Journal of Radiation Applications and Instrumentation. Part A …, 1988 | 43 | 1988 |
Double [3+ 2]-dimerisation cascade synthesis of bis (triazolyl) bisphosphanes, a new scaffold for bidentate bisphosphanes C Laborde, MM Wei, A van Der Lee, E Deydier, JC Daran, JN Volle, ... Dalton Transactions 44 (28), 12539-12545, 2015 | 41 | 2015 |
C-Glycoside Mimetics Inhibit Glioma Stem Cell Proliferation, Migration, and Invasion L Clarion, C Jacquard, O Sainte-Catherine, M Decoux, S Loiseau, ... Journal of Medicinal Chemistry 57 (20), 8293-8306, 2014 | 41 | 2014 |
Pallado-catalysed P-arylations and P-vinylation of 2-hydrogeno-2-oxo-1, 4, 2-oxazaphosphinanes JL Pirat, J Monbrun, D Virieux, HJ Cristau Tetrahedron 61 (29), 7029-7036, 2005 | 40 | 2005 |
Diastereoselective Addition of 2H-2-Oxo-1,4,2-oxazaphosphinanes to Aldehydes and Imines JL Pirat, J Monbrun, D Virieux, JN Volle, M Tillard, HJ Cristau The Journal of Organic Chemistry 70 (18), 7035-7041, 2005 | 39 | 2005 |
Neuroprotection in non-transgenic and transgenic mouse models of Alzheimer's disease by positive modulation of σ1 receptors T Maurice, JN Volle, M Strehaiano, L Crouzier, C Pereira, N Kaloyanov, ... Pharmacological Research 144, 315-330, 2019 | 38 | 2019 |
Novel easily recyclable bifunctional phosphonic acid carrying tripeptides for the stereoselective michael addition of aldehydes with nitroalkenes M Cortes‐Clerget, O Gager, M Monteil, JL Pirat, E Migianu‐Griffoni, ... Advanced Synthesis & Catalysis 358 (1), 34-40, 2016 | 37 | 2016 |
Hydrophosphonylation of alkenes or nitriles by double radical transfer mediated by titanocene/propylene oxide C Midrier, M Lantsoght, JN Volle, JL Pirat, D Virieux, CV Stevens Tetrahedron letters 52 (50), 6693-6696, 2011 | 37 | 2011 |
Synthesis and biological applications of phosphinates and derivatives D Virieux, JN Volle, N Bakalara, JL Pirat Phosphorus Chemistry I: Asymmetric Synthesis and Bioactive Compounds, 39-114, 2015 | 36 | 2015 |
Synthesis, reactivity and stereochemistry of new phosphorus heterocycles with 5-or 6-membered rings HJ Cristau, JL Pirat, D Virieux, J Monbrun, C Ciptadi, YA Bekro Journal of organometallic chemistry 690 (10), 2472-2481, 2005 | 36 | 2005 |
Preparation of phosphinodipeptide analogs as building blocks for pseudopeptides synthesis HJ Cristau, A Coulombeau, A Genevois-Borella, F Sanchez, JL Pirat Journal of organometallic chemistry 643, 381-391, 2002 | 35 | 2002 |
A convenient synthesis of tetrazole, precursors of α-dialkylated α-amino acids, by reaction of trimethylsilyl azide with α-dialkylated β-ketoesters HJ Cristau, X Marat, JP Vors, JL Pirat Tetrahedron letters 44 (15), 3179-3181, 2003 | 34 | 2003 |
Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group JN Volle, D Filippini, B Krawczy, N Kaloyanov, A Van der Lee, T Maurice, ... Organic & Biomolecular Chemistry 8 (6), 1438-1444, 2010 | 33 | 2010 |