Fluorine in pharmaceutical industry: fluorine-containing drugs introduced to the market in the last decade (2001–2011) J Wang, M Sánchez-Roselló, JL Aceña, C Del Pozo, AE Sorochinsky, ... Chemical reviews 114 (4), 2432-2506, 2014 | 4615 | 2014 |
Next generation of fluorine-containing pharmaceuticals, compounds currently in phase II–III clinical trials of major pharmaceutical companies: new structural trends and … Y Zhou, J Wang, Z Gu, S Wang, W Zhu, JL Aceña, VA Soloshonok, ... Chemical reviews 116 (2), 422-518, 2016 | 2482 | 2016 |
Enantioselective synthesis of beta-amino acids E Juaristi, VA Soloshonok John Wiley & Sons, 2005 | 1067 | 2005 |
Modern approaches for asymmetric construction of carbon–fluorine quaternary stereogenic centers: synthetic challenges and pharmaceutical needs Y Zhu, J Han, J Wang, N Shibata, M Sodeoka, VA Soloshonok, ... Chemical reviews 118 (7), 3887-3964, 2018 | 562 | 2018 |
Recent advances in the trifluoromethylation methodology and new CF3-containing drugs W Zhu, J Wang, S Wang, Z Gu, JL Aceña, K Izawa, H Liu, VA Soloshonok Journal of Fluorine Chemistry 167, 37-54, 2014 | 468 | 2014 |
Fluorine‐containing drugs approved by the FDA in 2018 H Mei, J Han, S Fustero, M Medio‐Simon, DM Sedgwick, C Santi, ... Chemistry–A European Journal 25 (51), 11797-11819, 2019 | 435 | 2019 |
Fluorine-containing Amino Acids: Synthesis and Properties VA Soloshonok, VP Kukhar John Wiley & Sons, 1995 | 422* | 1995 |
Chemical aspects of human and environmental overload with fluorine J Han, L Kiss, H Mei, AM Remete, M Ponikvar-Svet, DM Sedgwick, ... Chemical Reviews 121 (8), 4678-4742, 2021 | 285 | 2021 |
Enantiocontrolled synthesis of fluoro-organic compounds: stereochemical challenges and biomedical targets VA Soloshonok (No Title), 1999 | 272 | 1999 |
Remarkable amplification of the self‐disproportionation of enantiomers on achiral‐phase chromatography columns VA Soloshonok Angewandte Chemie International Edition 45 (5), 766-769, 2006 | 247 | 2006 |
Chiral sulfoxides: advances in asymmetric synthesis and problems with the accurate determination of the stereochemical outcome J Han, VA Soloshonok, KD Klika, J Drabowicz, A Wzorek Chemical Society Reviews 47 (4), 1307-1350, 2018 | 240 | 2018 |
Next generation organofluorine containing blockbuster drugs J Han, AM Remete, LS Dobson, L Kiss, K Izawa, H Moriwaki, ... Journal of Fluorine Chemistry 239, 109639, 2020 | 228 | 2020 |
Applications of fluorine-containing amino acids for drug design H Mei, J Han, KD Klika, K Izawa, T Sato, NA Meanwell, VA Soloshonok European journal of medicinal chemistry 186, 111826, 2020 | 195 | 2020 |
Phenomenon of optical self-purification of chiral non-racemic compounds VA Soloshonok, H Ueki, M Yasumoto, S Mekala, JS Hirschi, DA Singleton Journal of the American Chemical Society 129 (40), 12112-12113, 2007 | 191 | 2007 |
Fluorine-containing drugs approved by the FDA in 2019 H Mei, AM Remete, Y Zou, H Moriwaki, S Fustero, L Kiss, VA Soloshonok, ... Chinese Chemical Letters 31 (9), 2401-2413, 2020 | 189 | 2020 |
Asymmetric synthesis of fluorine-containing amines, amino alcohols, α-and β-amino acids mediated by chiral sulfinyl group AE Sorochinsky, VA Soloshonok Journal of Fluorine Chemistry 131 (2), 127-139, 2010 | 178 | 2010 |
Self-disproportionation of enantiomers via achiral chromatography: a warning and an extra dimension in optical purifications VA Soloshonok, C Roussel, O Kitagawa, AE Sorochinsky Chemical Society Reviews 41 (11), 4180-4188, 2012 | 176 | 2012 |
Recent advances in the synthesis of fluorinated aminophosphonates and aminophosphonic acids KV Turcheniuk, VP Kukhar, GV Röschenthaler, JL Aceña, VA Soloshonok, ... RSC advances 3 (19), 6693-6716, 2013 | 166 | 2013 |
Asymmetric synthesis of α-amino acids via homologation of Ni (II) complexes of glycine Schiff bases; Part 1: alkyl halide alkylations AE Sorochinsky, JL Aceña, H Moriwaki, T Sato, VA Soloshonok Amino Acids 45, 691-718, 2013 | 155 | 2013 |
Recent advances in the asymmetric synthesis of α-(trifluoromethyl)-containing α-amino acids JL Aceña, AE Sorochinsky, VA Soloshonok Synthesis 44 (11), 1591-1602, 2012 | 153 | 2012 |