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Kamala K Vasu
Kamala K Vasu
Assistant Director, B.V.Patel PERD Centre, Ahmedabad, India
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标题
引用次数
引用次数
年份
Synthesis of 4-benzyl-1, 3-thiazole derivatives as potential anti-inflammatory agents: an analogue-based drug design approach
RN Sharma, FP Xavier, KK Vasu, SC Chaturvedi, SS Pancholi
Journal of enzyme inhibition and medicinal chemistry 24 (3), 890-897, 2009
2582009
Design, synthesis and characterization of novel 2-(2, 4-disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one derivatives as inhibitors of NF-κB and AP-1 mediated …
RS Giri, HM Thaker, T Giordano, J Williams, D Rogers, V Sudersanam, ...
European journal of medicinal chemistry 44 (5), 2184-2189, 2009
2322009
Novel drug designing approach for dual inhibitors as anti-inflammatory agents: implication of pyridine template
AD Pillai, PD Rathod, PX Franklin, M Patel, M Nivsarkar, KK Vasu, H Padh, ...
Biochemical and Biophysical Research Communications 301 (1), 183-186, 2003
1302003
2-Amino-5-thiazolyl motif: A novel scaffold for designing anti-inflammatory agents of diverse structures
PX Franklin, AD Pillai, PD Rathod, S Yerande, M Nivsarkar, H Padh, ...
European journal of medicinal chemistry 43 (1), 129-134, 2008
1242008
Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents
KI Molvi, KK Vasu, SG Yerande, V Sudarsanam, N Haque
European journal of medicinal chemistry 42 (8), 1049-1058, 2007
962007
Tetra substituted thiophenes as anti-inflammatory agents: exploitation of analogue-based drug design
AD Pillai, PD Rathod, FP Xavier, H Padh, V Sudarsanam, KK Vasu
Bioorganic & medicinal chemistry 13 (24), 6685-6692, 2005
912005
Investigation of microemulsion system for transdermal delivery of itraconazole
A Chudasama, V Patel, M Nivsarkar, K Vasu, C Shishoo
Journal of advanced pharmaceutical technology & research 2 (1), 30-38, 2011
892011
QSAR studies on some thiophene analogs as anti-inflammatory agents: enhancement of activity by electronic parameters and its utilization for chemical lead optimization
AD Pillai, S Rani, PD Rathod, FP Xavier, KK Vasu, H Padh, ...
Bioorganic & medicinal chemistry 13 (4), 1275-1283, 2005
732005
Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-кB and AP-1 mediated transcriptional …
RS Giri, HM Thaker, T Giordano, J Williams, D Rogers, KK Vasu, ...
Bioorganic & Medicinal Chemistry 18 (7), 2796-2808, 2010
642010
Dissolution test for site-specific release isoniazid pellets in USP apparatus 3 (reciprocating cylinder): Optimization using response surface methodology
A Joshi, S Pund, M Nivsarkar, K Vasu, C Shishoo
European journal of pharmaceutics and biopharmaceutics 69 (2), 769-775, 2008
632008
Gastroretentive delivery of rifampicin: In vitro mucoadhesion and in vivo gamma scintigraphy
S Pund, A Joshi, K Vasu, M Nivsarkar, C Shishoo
International journal of pharmaceutics 411 (1-2), 106-112, 2011
592011
Design, synthesis, and pharmacological evaluation of some 2-[4-morpholino]-3-aryl-5-substituted thiophenes as novel anti-inflammatory agents: generation of a novel anti …
AD Pillai, PD Rathod, FP Xavier, KK Vasu, H Padh, V Sudarsanam
Bioorganic & medicinal chemistry 12 (17), 4667-4671, 2004
562004
Design, synthesis, and SAR studies of some 5-aliphatic oximino esters of thiophene as potential anti-inflammatory leads: comparative biological activity profile of aliphatic …
AD Pillai, PD Rathod, PX Franklin, H Padh, KK Vasu, V Sudarsanam
Biochemical and biophysical research communications 317 (4), 1067-1074, 2004
472004
Synthesis and evaluation of quinazolinone derivatives as inhibitors of NF-κB, AP-1 mediated transcription and eIF-4E mediated translational activation: Inhibitors of multi …
RS Giri, HM Thaker, T Giordano, B Chen, S Nuthalapaty, KK Vasu, ...
European journal of medicinal chemistry 45 (9), 3558-3563, 2010
422010
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists
AB Scheiff, SG Yerande, A El-Tayeb, W Li, GS Inamdar, KK Vasu, ...
Bioorganic & Medicinal Chemistry 18 (6), 2195-2203, 2010
392010
Design, synthesis and biological evaluation of novel pyrazolo-pyrimidinones as DPP-IV inhibitors in diabetes
SR Sagar, JK Agarwal, DH Pandya, RP Dash, M Nivsarkar, KK Vasu
Bioorganic & Medicinal Chemistry Letters 25 (20), 4428-4433, 2015
362015
Multivariate optimization of formulation and process variables influencing physico-mechanical characteristics of site-specific release isoniazid pellets
S Pund, A Joshi, K Vasu, M Nivsarkar, C Shishoo
International journal of pharmaceutics 388 (1-2), 64-72, 2010
362010
New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1, 3-thiazol-2-yl] benzamides and furamides
GS Inamdar, AN Pandya, HM Thakar, V Sudarsanam, S Kachler, ...
European Journal of Medicinal Chemistry 63, 924-934, 2013
332013
A convenient synthesis of di-and trisubstituted 2-aminoimidazoles from 1-amidino-3-trityl-thioureas
JC Kaila, AB Baraiya, AN Pandya, HB Jalani, KK Vasu, V Sudarsanam
Tetrahedron Letters 50 (27), 3955-3958, 2009
302009
A novel lipid-based oral drug delivery system of nevirapine
A Chudasama, V Patel, M Nivsarkar, K Vasu, C Shishoo
Int. J. Pharm. Tech. Res 3 (2), 1159-1168, 2011
292011
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