Tetrazoles via multicomponent reactions CG Neochoritis, T Zhao, A Domling Chemical reviews 119 (3), 1970-2042, 2019 | 511 | 2019 |
One-pot microwave assisted synthesis under green chemistry conditions, antioxidant screening, and cytotoxicity assessments of benzimidazole Schiff bases and pyrimido [1, 2-a … CG Neochoritis, T Zarganes-Tzitzikas, CA Tsoleridis, ... European journal of medicinal chemistry 46 (1), 297-306, 2011 | 128 | 2011 |
How to design a successful p53–MDM2/X interaction inhibitor: a thorough overview based on crystal structures N Estrada‐Ortiz, CG Neochoritis, A Dömling ChemMedChem 11 (8), 757-772, 2016 | 101 | 2016 |
Efficient isocyanide-less isocyanide-based multicomponent reactions CG Neochoritis, S Stotani, B Mishra, A Dömling Organic letters 17 (8), 2002-2005, 2015 | 100 | 2015 |
1, 5-Benzoxazepines vs 1, 5-benzodiazepines. One-pot microwave-assisted synthesis and evaluation for antioxidant activity and lipid peroxidation inhibition CG Neochoritis, CA Tsoleridis, J Stephanidou-Stephanatou, ... Journal of medicinal chemistry 53 (23), 8409-8420, 2010 | 90 | 2010 |
Versatile multicomponent reaction macrocycle synthesis using α-isocyano-ω-carboxylic acids GP Liao, EMM Abdelraheem, CG Neochoritis, K Kurpiewska, ... Organic letters 17 (20), 4980-4983, 2015 | 72 | 2015 |
Atorvastatin (lipitor) by MCR T Zarganes-Tzitzikas, CG Neochoritis, A Dömling ACS medicinal chemistry letters 10 (3), 389-392, 2019 | 71 | 2019 |
Dimethyl acetylenedicarboxylate: a versatile tool in organic synthesis CG Neochoritis, T Zarganes-Tzitzikas, J Stephanidou-Stephanatou Synthesis 46 (05), 537-585, 2014 | 71 | 2014 |
Repurposing the HCV NS3–4A protease drug boceprevir as COVID-19 therapeutics R Oerlemans, AJ Ruiz-Moreno, Y Cong, ND Kumar, ... RSC medicinal chemistry 12 (3), 370-379, 2021 | 69 | 2021 |
Rational Development of a Potent 15-Lipoxygenase-1 Inhibitor with in Vitro and ex Vivo Anti-inflammatory Properties N Eleftheriadis, CG Neochoritis, NGJ Leus, PE van der Wouden, ... Journal of medicinal chemistry 58 (19), 7850-7862, 2015 | 60 | 2015 |
TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics VBK Kunig, M Potowski, M Akbarzadeh, M Klika Škopić, ... Angewandte Chemie 132 (46), 20518-20522, 2020 | 59 | 2020 |
Rational design and synthesis of 1, 5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction E Surmiak, CG Neochoritis, B Musielak, A Twarda-Clapa, K Kurpiewska, ... European Journal of Medicinal Chemistry 126, 384-407, 2017 | 53 | 2017 |
Leuckart–Wallach route toward isocyanides and some applications CG Neochoritis, T Zarganes-Tzitzikas, S Stotani, A Dömling, ... ACS combinatorial science 17 (9), 493-499, 2015 | 51 | 2015 |
2, 3′-Bis (1′ H-indole) heterocycles: New p53/MDM2/MDMX antagonists CG Neochoritis, K Wang, N Estrada-Ortiz, E Herdtweck, K Kubica, ... Bioorganic & medicinal chemistry letters 25 (24), 5661-5666, 2015 | 50 | 2015 |
Artificial macrocycles as potent p53–MDM2 inhibitors N Estrada-Ortiz, CG Neochoritis, A Twarda-Clapa, B Musielak, TA Holak, ... ACS medicinal chemistry letters 8 (10), 1025-1030, 2017 | 48 | 2017 |
Multicomponent reactions:“kinderleicht” CG Neochoritis, T Zarganes-Tzitzikas, K Katsampoxaki-Hodgetts, ... Journal of chemical education 97 (10), 3739-3745, 2020 | 46 | 2020 |
Design of a novel thiophene inhibitor of 15-lipoxygenase-1 with both anti-inflammatory and neuroprotective properties N Eleftheriadis, H Poelman, NGJ Leus, B Honrath, CG Neochoritis, ... European journal of medicinal chemistry 122, 786-801, 2016 | 43 | 2016 |
Multicomponent peptide stapling as a diversity‐driven tool for the development of inhibitors of protein–protein interactions MG Ricardo, AM Ali, J Plewka, E Surmiak, B Labuzek, CG Neochoritis, ... Angewandte Chemie International Edition 59 (13), 5235-5241, 2020 | 39 | 2020 |
One-pot microwave assisted synthesis of new 2-alkoxycarbonylmethylene-4-oxo-1, 5-benzo-, naphtho-, and pyridodiazepines and assessment of their cytogenetic activity N Eleftheriadis, CG Neochoritis, CA Tsoleridis, ... European journal of medicinal chemistry 67, 302-309, 2013 | 38 | 2013 |
Multicomponent reaction–derived covalent inhibitor space F Sutanto, S Shaabani, CG Neochoritis, T Zarganes-Tzitzikas, P Patil, ... Science advances 7 (6), eabd9307, 2021 | 35 | 2021 |