| Recent progress in the development of anti-malarial quinolones RM Beteck, FJ Smit, RK Haynes, DD N’Da Malaria journal 13, 1-10, 2014 | 95 | 2014 |
| Synthesis, in vitro antimalarial activity and cytotoxicity of novel 4-aminoquinolinyl-chalcone amides FJ Smit, DD N’Da Bioorganic & Medicinal Chemistry 22 (3), 1128-1138, 2014 | 71 | 2014 |
| Synthesis and in vitro biological evaluation of dihydroartemisinyl-chalcone esters FJ Smit, RA van Biljon, LM Birkholtz, DND David European journal of medicinal chemistry 90, 33-44, 2015 | 60 | 2015 |
| Synthesis and in vitro biological evaluation of aminoacridines and artemisinin–acridine hybrids JP Joubert, FJ Smit, L Du Plessis, PJ Smith, DD N’Da European Journal of Pharmaceutical Sciences 56, 16-27, 2014 | 55 | 2014 |
| Synthesis, in vitro antimalarial activities and cytotoxicities of amino-artemisinin-ferrocene derivatives C De Lange, D Coertzen, FJ Smit, JF Wentzel, HN Wong, LM Birkholtz, ... Bioorganic & medicinal chemistry letters 28 (3), 289-292, 2018 | 42 | 2018 |
| Synthesis, antimalarial activities and cytotoxicities of amino-artemisinin-1, 2-disubstituted ferrocene hybrids C De Lange, D Coertzen, FJ Smit, JF Wentzel, HN Wong, LM Birkholtz, ... Bioorganic & Medicinal Chemistry Letters 28 (19), 3161-3163, 2018 | 35 | 2018 |
| Accessible and distinct decoquinate derivatives active against Mycobacterium tuberculosis and apicomplexan parasites RM Beteck, R Seldon, D Coertzen, ME van der Watt, J Reader, ... Communications Chemistry 1 (1), 62, 2018 | 34 | 2018 |
| Single-step synthesis and in vitro anti-mycobacterial activity of novel nitrofurantoin analogues NH Zuma, FJ Smit, R Seldon, J Aucamp, A Jordaan, DF Warner, ... Bioorganic chemistry 96, 103587, 2020 | 24 | 2020 |
| Synthesis and antimycobacterial activity of disubstituted benzyltriazoles FJ Smit, R Seldon, J Aucamp, A Jordaan, DF Warner, DD N’Da Medicinal Chemistry Research 28, 2279-2293, 2019 | 24 | 2019 |
| Synthesis and in vitro biological activities of ferrocenyl–chalcone amides FJ Smit, JJ Bezuidenhout, CC Bezuidenhout, DD N’Da Medicinal Chemistry Research 25, 568-584, 2016 | 24 | 2016 |
| The case for development of 11-aza-artemisinins for malaria R Harmse, H Ning Wong, F Smit, R K Haynes, DD N’Da Current medicinal chemistry 22 (31), 3607-3630, 2015 | 21 | 2015 |
| Synthesis and biological evaluation of a series of non-hemiacetal ester derivatives of artemisinin NH Zuma, FJ Smit, C de Kock, J Combrinck, PJ Smith, DND David European Journal of Medicinal Chemistry 122, 635-646, 2016 | 20 | 2016 |
| Straightforward conversion of decoquinate into inexpensive tractable new derivatives with significant antimalarial activities RM Beteck, D Coertzen, FJ Smit, LM Birkholtz, RK Haynes, DD N’Da Bioorganic & Medicinal Chemistry Letters 26 (13), 3006-3009, 2016 | 20 | 2016 |
| Design, synthesis, and antimycobacterial activity of novel ciprofloxacin derivatives P Cilliers, R Seldon, FJ Smit, J Aucamp, A Jordaan, DF Warner, DD N'Da Chemical biology & drug design 94 (2), 1518-1536, 2019 | 19 | 2019 |
| Activities of 11‐Azaartemisinin and N‐Sulfonyl Derivatives against Neospora caninum and Comparative Cytotoxicities R Harmse, HN Wong, FJ Smit, J Müller, A Hemphill, DD N'Da, RK Haynes ChemMedChem 12 (24), 2094-2098, 2017 | 18 | 2017 |
| Preliminary evaluation of artemisinin–cholesterol conjugates as potential drugs for the treatment of intractable forms of malaria and tuberculosis M Morake, D Coertzen, A Ngwane, JF Wentzel, HN Wong, FJ Smit, ... ChemMedChem 13 (1), 67-77, 2018 | 17 | 2018 |
| Synthesis and comparison of in vitro dual anti-infective activities of novel naphthoquinone hybrids and atovaquone C Erasmus, J Aucamp, FJ Smit, R Seldon, A Jordaan, DF Warner, ... Bioorganic Chemistry 114, 105118, 2021 | 16 | 2021 |
| Synthesis and in vitro antimycobacterial and antileishmanial activities of hydroquinone-triazole hybrids CM Horn, J Aucamp, FJ Smit, R Seldon, A Jordaan, DF Warner, DD N’Da Medicinal Chemistry Research 29, 1387-1399, 2020 | 16 | 2020 |
| Activities of 11‐Azaartemisinin and N‐Sulfonyl Derivatives against Asexual and Transmissible Malaria Parasites R Harmse, D Coertzen, HN Wong, FJ Smit, ME van der Watt, J Reader, ... ChemMedChem 12 (24), 2086-2093, 2017 | 16 | 2017 |
| Synthesis and in vitro antimalarial activity of novel chalcone derivatives FJ Smit | 3 | 2014 |
