A Copper‐Catalyzed Tandem Synthesis of Indolo‐ and Pyrrolo[2,1‐a]isoquinolines AK Verma, T Kesharwani, J Singh, V Tandon, RC Larock Angewandte Chemie 121 (6), 1158-1163, 2009 | 222 | 2009 |
Synthesis of 3,4-Disubstituted 2H-Benzopyrans through C−C Bond Formation via Electrophilic Cyclization SA Worlikar, T Kesharwani, T Yao, RC Larock The Journal of organic chemistry 72 (4), 1347-1353, 2007 | 182 | 2007 |
Synthesis of 2,3-Disubstituted Benzo[b]selenophenes via Electrophilic Cyclization T Kesharwani, SA Worlikar, RC Larock The Journal of organic chemistry 71 (6), 2307-2312, 2006 | 164 | 2006 |
Discovery of Clinical Candidate (1R,4r)-4-((R)-2-((S)-6-Fluoro-5H-imidazo[5,1-a]isoindol-5-yl)-1-hydroxyethyl)cyclohexan-1-ol (Navoximod), a Potent and … S Kumar, JP Waldo, FA Jaipuri, A Marcinowicz, C Van Allen, J Adams, ... Journal of medicinal chemistry 62 (14), 6705-6733, 2019 | 65 | 2019 |
IDO inhibitors M Mautino, F Jaipuri, A Marcinowicz-Flick, T Kesharwani, J Waldo US Patent 10,047,066, 2018 | 59 | 2018 |
Studies in acyl C− H activation via aryl and alkyl to acyl “through space” migration of palladium T Kesharwani, AK Verma, D Emrich, JA Ward, RC Larock Organic letters 11 (12), 2591-2593, 2009 | 59 | 2009 |
Benzylic C–H activation and C–O bond formation via aryl to benzylic 1, 4-palladium migrations T Kesharwani, RC Larock Tetrahedron 64 (26), 6090-6102, 2008 | 56 | 2008 |
Fused imidazole derivatives useful as IDO inhibitors M Mautino, S Kumar, J Waldo, F Jaipuri, T Kesharwani, X Zhang US Patent 9,260,434, 2016 | 48 | 2016 |
Environmentally benign process for the synthesis of 2, 3-disubstituted benzo [b] thiophenes using electrophilic cyclization S Kim, N Dahal, T Kesharwani Tetrahedron Letters 54 (33), 4373-4376, 2013 | 47 | 2013 |
IDO inhibitors MR Mautino, S Kumar, F Jaipuri, J Waldo, T Kesharwani, NN Vahanian, ... US Patent 8,748,469, 2014 | 31 | 2014 |
Green synthesis of halogenated thiophenes, selenophenes and benzo [b] selenophenes using sodium halides as a source of electrophilic halogens T Kesharwani, KA Giraudy, JL Morgan, C Kornman, AD Olaitan Tetrahedron letters 58 (7), 638-641, 2017 | 29 | 2017 |
Variable temperature NMR experiment studying restricted bond rotation MT Huggins, T Kesharwani, J Buttrick, C Nicholson Journal of chemical education 97 (5), 1425-1429, 2020 | 27 | 2020 |
Imidazole derivatives as IDO inhibitors MR Mautino, S Kumar, F Jaipuri, J Waldo, T Kesharwani US Patent 8,722,720, 2014 | 27 | 2014 |
Synthesis of pyrrolo-[2, 1-j] quinolone framework via intramolecular electrophilic ipso-cyclization L Low-Beinart, X Sun, E Sidman, T Kesharwani Tetrahedron Letters 54 (11), 1344-1347, 2013 | 26 | 2013 |
Green synthesis of benzo [b] thiophenes via iron (III) mediated 5-endo-dig iodocyclization of 2-alkynylthioanisoles T Kesharwani, CT Kornman, AL Tonnaer, AD Royappa Tetrahedron Letters 57 (3), 411-414, 2016 | 22 | 2016 |
Sodium halides as the source of electrophilic halogens in green synthesis of 3-halo-and 3, n-dihalobenzo [b] thiophenes T Kesharwani, C Kornman, A Tonnaer, A Hayes, S Kim, N Dahal, ... Tetrahedron 74 (24), 2973-2984, 2018 | 20 | 2018 |
IDO Inhibitors M Mautino, F Jaipuri, A Marcinowicz-Flick, T Kesharwani, J Waldo US Patent App. 13/801,268, 2013 | 15 | 2013 |
Copper-catalyzed electrophilic chlorocyclization reaction using sodium chloride as the source of electrophilic chlorine C Walter, N Fallows, T Kesharwani ACS omega 4 (4), 6538-6545, 2019 | 13 | 2019 |
Synthesis of 3-iodobenzo [b] thiophenes via iodocyclization/etherification reaction sequence T Kesharwani, J Craig, C Del Rosario, R Shavnore, C Kornman Tetrahedron letters 55 (50), 6812-6816, 2014 | 13 | 2014 |
Comprehensive Organic Transformations, 4 Volume Set: A Guide to Functional Group Preparations AV Dubrovskiy, T Kesharwani, NA Markina, AA Pletnev, C Raminelli, ... John Wiley & Sons, 2018 | 12 | 2018 |